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IN2014DN07797A - - Google Patents

Info

Publication number
IN2014DN07797A
IN2014DN07797A IN7797DEN2014A IN2014DN07797A IN 2014DN07797 A IN2014DN07797 A IN 2014DN07797A IN 7797DEN2014 A IN7797DEN2014 A IN 7797DEN2014A IN 2014DN07797 A IN2014DN07797 A IN 2014DN07797A
Authority
IN
India
Prior art keywords
disintegrating
components
tablet
wet granulation
component
Prior art date
Application number
Other languages
English (en)
Inventor
Takahiro Hiramura
Kiyoshi Ikura
Sae Ishikawa
Tomohito Okabayashi
Naohiro Hashikawa
Tetsuro Morita
Kimiko Ikeda
Haruka WAKAYAMA
Original Assignee
Daicel Corp
Nichirin Chemical Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49260166&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014DN07797(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Daicel Corp, Nichirin Chemical Ind filed Critical Daicel Corp
Publication of IN2014DN07797A publication Critical patent/IN2014DN07797A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
IN7797DEN2014 2012-03-29 2013-03-27 IN2014DN07797A (fr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2012075832 2012-03-29
JP2012206895 2012-09-20
JP2012206896 2012-09-20
JP2012275942 2012-12-18
PCT/JP2013/059083 WO2013146917A1 (fr) 2012-03-29 2013-03-27 Procédé de production d'une composition de particules délitantes comprenant de la carboxyméthylcellulose de type acide, composition de particules délitantes comprenant de la carboxyméthylcellulose de type acide, et comprimé à dissolution orale contenant une composition de particules délitantes comprenant de la carboxyméthylcellulose de type acide

Publications (1)

Publication Number Publication Date
IN2014DN07797A true IN2014DN07797A (fr) 2015-05-15

Family

ID=49260166

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7797DEN2014 IN2014DN07797A (fr) 2012-03-29 2013-03-27

Country Status (8)

Country Link
US (2) US20150174075A2 (fr)
EP (1) EP2832350B1 (fr)
JP (1) JP5996633B2 (fr)
KR (1) KR101707938B1 (fr)
CN (1) CN104080443B (fr)
IN (1) IN2014DN07797A (fr)
TW (1) TWI610691B (fr)
WO (1) WO2013146917A1 (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN2014DN07797A (fr) 2012-03-29 2015-05-15 Daicel Corp
WO2014046035A1 (fr) 2012-09-20 2014-03-27 株式会社ダイセル Composition de particule se désintégrant contenant de la carboxyméthylcellulose de type acide et de la cellulose cristalline, et comprimé se désintégrant oralement contenant ladite composition
CN105517576A (zh) * 2013-07-06 2016-04-20 株式会社大赛璐 超速崩解片剂及其制备方法
CN105555316B (zh) * 2013-09-27 2020-07-07 株式会社大赛璐 通过二阶段的湿式制粒工序制备的崩解性颗粒组合物及含有该组合物的口腔内崩解片剂
US20160213619A1 (en) * 2013-09-27 2016-07-28 Daicel Corporation Intraorally disintegrable tablet comprising disintegrable granular composition
JP2017036214A (ja) * 2013-12-10 2017-02-16 株式会社ダイセル 炭酸塩を含む口腔内崩壊錠剤用組成物及び口腔内崩壊錠剤
EP3135300B1 (fr) 2014-04-21 2022-03-30 Daicel Corporation Composition particulaire apte à se désagréger comprenant de la cellulose microfibreuse
JP2017226600A (ja) * 2014-10-16 2017-12-28 株式会社ダイセル 超速崩壊錠剤
KR102377914B1 (ko) 2014-11-24 2022-03-22 주식회사 다이셀 분쇄 유당 또는 조립 유당을 포함하는 붕해성 입자 조성물
WO2016098459A1 (fr) * 2014-12-17 2016-06-23 株式会社ダイセル Composition particulaire à désintégration retardée
CN106999437A (zh) * 2014-12-25 2017-08-01 株式会社大赛璐 超速崩解片剂及其制备方法
JP5897196B1 (ja) * 2015-10-05 2016-03-30 大同化成工業株式会社 糖又は糖アルコール、膨潤型結合剤、崩壊剤及び高吸収性賦形剤を含む複合化造粒物及びその製造方法
WO2018021265A1 (fr) 2016-07-27 2018-02-01 沢井製薬株式会社 Composition d'additif pour comprimé à désintégration orale
JP6651638B2 (ja) 2016-09-06 2020-02-19 沢井製薬株式会社 口腔内崩壊錠添加用組成物
WO2020022053A1 (fr) * 2018-07-25 2020-01-30 株式会社ダイセル Composition particulaire se délitant contenant de la cellulose microfibreuse mais ne contenant pas d'excipient
WO2020246120A1 (fr) * 2019-06-07 2020-12-10 あゆみ製薬株式会社 Comprimé à désintégration buccale et son procédé de production

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2851453A (en) * 1954-08-09 1958-09-09 Smith Kline French Lab Cellulose derivative product, compositions comprising the same and their preparation
JPH10182436A (ja) 1996-10-31 1998-07-07 Takeda Chem Ind Ltd 固形医薬製剤
JP2000273039A (ja) 1999-01-20 2000-10-03 Taisho Pharmaceut Co Ltd 口腔内崩壊性組成物
JP4284017B2 (ja) * 2000-10-06 2009-06-24 武田薬品工業株式会社 固形製剤
AU2001294192A1 (en) 2000-10-06 2002-04-22 Takeda Chemical Industries Ltd. Solid preparations
JP4551627B2 (ja) 2003-02-28 2010-09-29 東和薬品株式会社 口腔内崩壊錠剤の製造方法
KR20080083071A (ko) 2003-08-08 2008-09-12 아지노모토 가부시키가이샤 나테글리니드 함유 제제
EP1923074A4 (fr) * 2005-08-10 2011-09-14 Shionogi & Co Comprimé pouvant être désintégré par voie orale
JP5123517B2 (ja) 2005-11-14 2013-01-23 帝人ファーマ株式会社 アンブロキソール口腔内速崩性錠剤
WO2008061226A2 (fr) * 2006-11-17 2008-05-22 Supernus Pharmaceuticals Inc. Formulations de topiramate à libération prolongée
JP5766899B2 (ja) * 2007-04-11 2015-08-19 ニプロ株式会社 口腔内崩壊剤及びその製造方法
JP2008285434A (ja) 2007-05-16 2008-11-27 Taisho Pharm Ind Ltd 口腔内速崩壊錠
CA2686964A1 (fr) 2007-06-06 2008-12-11 Basf Se Preparation pharmaceutique pour produire des comprimes a delitement rapide
JP4989733B2 (ja) * 2008-02-13 2012-08-01 大日本住友製薬株式会社 口腔内崩壊錠
US20110229570A1 (en) * 2008-11-25 2011-09-22 Masaaki Sugimoto Orally rapidly disintegrating tablet and process for producing same
WO2011019045A1 (fr) 2009-08-11 2011-02-17 富士化学工業株式会社 Composition de particules se désintégrant et comprimé se désintégrant rapidement dans la cavité buccale
US8591955B2 (en) 2009-08-11 2013-11-26 Dainippon Sumitomo Pharma Co., Ltd. Orally rapidly disintegrating tablet that contains two or more types of particles
US20110150989A1 (en) 2009-12-22 2011-06-23 Mallinkckrodt Inc. Methods of Producing Stabilized Solid Dosage Pharmaceutical Compositions Containing Morphinans
US9198861B2 (en) * 2009-12-22 2015-12-01 Mallinckrodt Llc Methods of producing stabilized solid dosage pharmaceutical compositions containing morphinans
JP6073543B2 (ja) * 2010-07-08 2017-02-01 沢井製薬株式会社 ロラタジン含有口腔内崩壊錠の製造方法
JP5630902B2 (ja) * 2010-08-26 2014-11-26 沢井製薬株式会社 ゾルピデム酒石酸塩含有口腔内崩壊錠の製造方法
JP6245677B2 (ja) 2012-01-20 2017-12-13 ニプロ株式会社 口腔内崩壊錠
IN2014DN07797A (fr) 2012-03-29 2015-05-15 Daicel Corp
WO2014046035A1 (fr) 2012-09-20 2014-03-27 株式会社ダイセル Composition de particule se désintégrant contenant de la carboxyméthylcellulose de type acide et de la cellulose cristalline, et comprimé se désintégrant oralement contenant ladite composition
CN105555316B (zh) * 2013-09-27 2020-07-07 株式会社大赛璐 通过二阶段的湿式制粒工序制备的崩解性颗粒组合物及含有该组合物的口腔内崩解片剂
KR102377914B1 (ko) * 2014-11-24 2022-03-22 주식회사 다이셀 분쇄 유당 또는 조립 유당을 포함하는 붕해성 입자 조성물
TWI690333B (zh) * 2015-06-29 2020-04-11 日商大賽璐股份有限公司 易服用性固態製劑(有核錠)之製造方法及易服用性固態製劑

Also Published As

Publication number Publication date
EP2832350B1 (fr) 2019-07-17
EP2832350A1 (fr) 2015-02-04
WO2013146917A1 (fr) 2013-10-03
US12059501B2 (en) 2024-08-13
CN104080443B (zh) 2017-12-12
JP5996633B2 (ja) 2016-09-21
EP2832350A4 (fr) 2015-11-18
TWI610691B (zh) 2018-01-11
US20150174075A2 (en) 2015-06-25
CN104080443A (zh) 2014-10-01
US20150045452A1 (en) 2015-02-12
KR20140144249A (ko) 2014-12-18
JPWO2013146917A1 (ja) 2015-12-14
TW201400145A (zh) 2014-01-01
KR101707938B1 (ko) 2017-02-17
US20200038332A1 (en) 2020-02-06

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