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IN2014MN02574A - - Google Patents

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Publication number
IN2014MN02574A
IN2014MN02574A IN2574MUN2014A IN2014MN02574A IN 2014MN02574 A IN2014MN02574 A IN 2014MN02574A IN 2574MUN2014 A IN2574MUN2014 A IN 2574MUN2014A IN 2014MN02574 A IN2014MN02574 A IN 2014MN02574A
Authority
IN
India
Prior art keywords
compounds
subscript
compositions
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meaning
Prior art date
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English (en)
Inventor
Jean Christophe Andrez
Sultan Chowdhury
Shannon Decker
Christoph Martin Dehnhardt
Thilo Focken
Michael Edward Grimwood
Ivan William Hemeon
Qi Jia
Jun Li
Daniel F Ortwine
Brian Safina
Tao Sheng
Shaoyi Sun
Daniel P Sutherlin
Michael Scott Wilson
Alla Yurevna Zenova
Original Assignee
Genentech Inc
Xenon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Genentech Inc, Xenon Pharmaceuticals Inc filed Critical Genentech Inc
Publication of IN2014MN02574A publication Critical patent/IN2014MN02574A/en

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
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    • A61K31/18—Sulfonamides
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
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    • C—CHEMISTRY; METALLURGY
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    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
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CO7160015A2 (es) 2015-01-15
US20160297754A1 (en) 2016-10-13
SG11201408284VA (en) 2015-02-27
EP2855428A1 (fr) 2015-04-08
IL235846A0 (en) 2015-02-01
EA026393B1 (ru) 2017-04-28
US20130317001A1 (en) 2013-11-28
EA201492166A1 (ru) 2015-09-30
WO2013177224A1 (fr) 2013-11-28
AU2013266398A1 (en) 2015-01-22
JP6038297B2 (ja) 2016-12-07
CA2874621A1 (fr) 2013-11-28
HK1206711A1 (en) 2016-01-15
US8933236B2 (en) 2015-01-13
ZA201409334B (en) 2016-09-28
CR20140578A (es) 2015-04-30
JP2015518863A (ja) 2015-07-06
KR20150032534A (ko) 2015-03-26
PE20150400A1 (es) 2015-03-27
US20150224071A1 (en) 2015-08-13
CN104718188A (zh) 2015-06-17
US20130317000A1 (en) 2013-11-28
MX2014014234A (es) 2015-05-07
CL2014003181A1 (es) 2015-07-10
BR112014029161A2 (pt) 2017-06-27
PH12014502597A1 (en) 2015-02-02
AR091112A1 (es) 2015-01-14
US20170002017A1 (en) 2017-01-05
KR101719893B1 (ko) 2017-03-24
HK1209100A1 (en) 2016-03-24
US8952169B2 (en) 2015-02-10
US9771376B2 (en) 2017-09-26
CN104718188B (zh) 2018-08-21
TW201400446A (zh) 2014-01-01

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