IN2013MU03508A - - Google Patents
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- Publication number
- IN2013MU03508A IN2013MU03508A IN3508MU2013A IN2013MU03508A IN 2013MU03508 A IN2013MU03508 A IN 2013MU03508A IN 3508MU2013 A IN3508MU2013 A IN 3508MU2013A IN 2013MU03508 A IN2013MU03508 A IN 2013MU03508A
- Authority
- IN
- India
- Prior art keywords
- linezolid
- present
- crystalline form
- relates
- crystallizing
- Prior art date
Links
- TYZROVQLWOKYKF-ZDUSSCGKSA-N linezolid Chemical compound O=C1O[C@@H](CNC(=O)C)CN1C(C=C1F)=CC=C1N1CCOCC1 TYZROVQLWOKYKF-ZDUSSCGKSA-N 0.000 abstract 4
- 229960003907 linezolid Drugs 0.000 abstract 4
- 238000000034 method Methods 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000007787 solid Substances 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/IB2014/065837 WO2015068121A1 (fr) | 2013-11-06 | 2014-11-06 | Procédé pour la préparation de la forme cristalline i de linézolide et ses compositions |
| IN3508MU2013 IN2013MU03508A (fr) | 2013-11-06 | 2014-11-06 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN3508MU2013 IN2013MU03508A (fr) | 2013-11-06 | 2014-11-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2013MU03508A true IN2013MU03508A (fr) | 2015-07-24 |
Family
ID=52144768
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN3508MU2013 IN2013MU03508A (fr) | 2013-11-06 | 2014-11-06 |
Country Status (2)
| Country | Link |
|---|---|
| IN (1) | IN2013MU03508A (fr) |
| WO (1) | WO2015068121A1 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105566242B (zh) * | 2016-01-12 | 2017-12-05 | 江苏豪森药业集团有限公司 | 利奈唑胺及其中间体的制备方法 |
| CN110483431A (zh) * | 2019-09-04 | 2019-11-22 | 桂林南药股份有限公司 | 利奈唑胺杂质化合物、其制备方法以及其应用 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY115155A (en) | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
| US5688792A (en) | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
| HUP0004388A3 (en) | 1997-11-07 | 2001-10-29 | Upjohn Co | Process for the preparation of oxazolidinones, intermediates and preparation thereof |
| US6444813B2 (en) | 2000-02-02 | 2002-09-03 | Pharmacia & Upjohn Company | Linezolid-crystal form II |
| DE09163348T1 (de) | 2003-10-16 | 2010-01-07 | Symed Labs Ltd., Hyderabad | Kristalline Form von Linezolid |
| WO2006110155A1 (fr) | 2004-06-29 | 2006-10-19 | Teva Pharmaceutical Industries Ltd | Formes solides du linezolide et leurs procedes de preparation |
| US7649096B2 (en) | 2005-07-15 | 2010-01-19 | Glenmark Pharmaceuticals Limited | Process for the preparation of a crystalline form of (S)-N [[3-(3-fluoro-4(4-morpholinyl) phenyl]-2-oxo-5-oxazolidinyl] methyl] acetamide |
| WO2007026369A1 (fr) | 2005-08-29 | 2007-03-08 | Symed Labs Limited | Nouvelle forme amorphe du linezolid |
| US20070197529A1 (en) | 2005-12-01 | 2007-08-23 | Viviana Braude | Isolated desfluoro-linezolid, preparation thereof and its use as a reference marker and standard |
| CN101774978B (zh) | 2009-01-13 | 2011-09-21 | 联化科技股份有限公司 | 一种利奈唑胺的制备方法及其中间体 |
| WO2011050826A1 (fr) | 2009-10-28 | 2011-05-05 | Synthon B.V. | Procédé de fabrication d'une forme cristalline de linézolide |
| CA2785620A1 (fr) | 2009-12-26 | 2011-06-30 | Alembic Pharmaceuticals Limited | Procede pour la preparation de linezolide |
| WO2012019632A1 (fr) | 2010-08-11 | 2012-02-16 | Synthon B.V. | Procédé pour fabriquer du linézolid |
| WO2012114354A1 (fr) | 2011-02-24 | 2012-08-30 | Lee Pharma Limited | Forme ii cristalline anhydre de linézolide |
| WO2012119653A1 (fr) | 2011-03-09 | 2012-09-13 | Synthon Bv | Procédé de préparation de la forme cristalline a du linézolid |
| WO2013072923A1 (fr) | 2011-09-19 | 2013-05-23 | Cadila Healthcare Limited | Procédé de préparation de linézolide cristallin |
| WO2013093751A1 (fr) | 2011-12-24 | 2013-06-27 | Alembic Pharmaceuticals Limited | Conditionnement pour le linézolide |
| WO2013120496A1 (fr) | 2012-02-14 | 2013-08-22 | Pharmathen S.A. | Procédé pour la préparation de linézolide sous forme cristalline et de sels de celui-ci |
| CN102850290A (zh) | 2012-10-10 | 2013-01-02 | 天津市炜杰科技有限公司 | 晶型i型利奈唑胺的制备方法 |
| WO2014101064A1 (fr) * | 2012-12-27 | 2014-07-03 | 上海创诺医药集团有限公司 | Procédé de préparation de la forme i cristalline de linézolide |
-
2014
- 2014-11-06 IN IN3508MU2013 patent/IN2013MU03508A/en unknown
- 2014-11-06 WO PCT/IB2014/065837 patent/WO2015068121A1/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2015068121A1 (fr) | 2015-05-14 |
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