IL166685A0 - Methods for treating carbonic anhydrase mediated disorders - Google Patents
Methods for treating carbonic anhydrase mediated disordersInfo
- Publication number
- IL166685A0 IL166685A0 IL16668505A IL16668505A IL166685A0 IL 166685 A0 IL166685 A0 IL 166685A0 IL 16668505 A IL16668505 A IL 16668505A IL 16668505 A IL16668505 A IL 16668505A IL 166685 A0 IL166685 A0 IL 166685A0
- Authority
- IL
- Israel
- Prior art keywords
- methods
- carbonic anhydrase
- mediated disorders
- treating
- anhydrase mediated
- Prior art date
Links
- 102000003846 Carbonic anhydrases Human genes 0.000 title 1
- 108090000209 Carbonic anhydrases Proteins 0.000 title 1
- 230000001404 mediated effect Effects 0.000 title 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
- A61K31/10—Sulfides; Sulfoxides; Sulfones
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A61K31/4164—1,3-Diazoles
- A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Hematology (AREA)
- Ophthalmology & Optometry (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Pulmonology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Reproductive Health (AREA)
- Hospice & Palliative Care (AREA)
- Pregnancy & Childbirth (AREA)
- Vascular Medicine (AREA)
- Oncology (AREA)
- Transplantation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/213,793 US20030100594A1 (en) | 2001-08-10 | 2002-08-07 | Carbonic anhydrase inhibitor |
| PCT/US2003/004494 WO2004014352A2 (fr) | 2002-08-07 | 2003-02-14 | Methodes de traitement de troubles dont la mediation est assuree par l'anhydrase carbonique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL166685A0 true IL166685A0 (en) | 2006-01-15 |
Family
ID=31714232
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16668505A IL166685A0 (en) | 2002-08-07 | 2005-02-03 | Methods for treating carbonic anhydrase mediated disorders |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US20030100594A1 (fr) |
| EP (2) | EP1526895A2 (fr) |
| JP (2) | JP2005539023A (fr) |
| KR (1) | KR20050056189A (fr) |
| CN (1) | CN1681557A (fr) |
| AU (2) | AU2003225571A1 (fr) |
| BR (2) | BR0313282A (fr) |
| CA (2) | CA2495502A1 (fr) |
| IL (1) | IL166685A0 (fr) |
| MX (2) | MXPA05001497A (fr) |
| PL (1) | PL374994A1 (fr) |
| WO (2) | WO2004014430A1 (fr) |
Families Citing this family (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10035227A1 (de) * | 2000-07-20 | 2002-01-31 | Solvay Pharm Gmbh | Verfahren zum Auffinden von Verbindungen, welche zur Behandlung und/oder Prophylaxe von Fettleibigkeit geeignet sind |
| US6946243B2 (en) * | 2000-07-20 | 2005-09-20 | Solvay Pharmaceuticals Gmbh | Method of identifying compounds suitable for treatment and/or prophylaxis of obesity |
| US20100135980A1 (en) * | 2000-10-16 | 2010-06-03 | Rodriguez Victorio C | Therapeutic and prophylactic uses of cell specific carbonic anhydrase enzymes in treating aging, disorders of aging, cancer, as growth factors, and as an alternative to stem cell therapy |
| US20030220376A1 (en) * | 2001-08-10 | 2003-11-27 | Pharmacia Corporation | Methods for treating carbonic anhydrase mediated disorders |
| KR101084871B1 (ko) * | 2003-05-22 | 2011-11-21 | 네르비아노 메디칼 사이언시스 에스.알.엘. | 피라졸로-퀴나졸린 유도체, 그의 제조 방법 및 상기유도체의 키나제 저해제로서의 용도 |
| WO2005079781A1 (fr) * | 2004-02-25 | 2005-09-01 | La Trobe University | Methode therapeutique et/ou prophylactique |
| WO2005094815A1 (fr) * | 2004-03-30 | 2005-10-13 | Amorepacific Corporation | Double inhibition de la cyclooxygenase 2 et de l'anhydrase carbonique |
| US8722097B2 (en) | 2004-04-30 | 2014-05-13 | Allergan, Inc. | Oil-in-water method for making polymeric implants containing a hypotensive lipid |
| US8673341B2 (en) | 2004-04-30 | 2014-03-18 | Allergan, Inc. | Intraocular pressure reduction with intracameral bimatoprost implants |
| US9498457B2 (en) | 2004-04-30 | 2016-11-22 | Allergan, Inc. | Hypotensive prostamide-containing biodegradable intraocular implants and related implants |
| US7799336B2 (en) | 2004-04-30 | 2010-09-21 | Allergan, Inc. | Hypotensive lipid-containing biodegradable intraocular implants and related methods |
| US7993634B2 (en) | 2004-04-30 | 2011-08-09 | Allergan, Inc. | Oil-in-oil emulsified polymeric implants containing a hypotensive lipid and related methods |
| MY147767A (en) | 2004-06-16 | 2013-01-31 | Janssen Pharmaceutica Nv | Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders |
| JP2008545650A (ja) | 2005-05-20 | 2008-12-18 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | スルファミド誘導体の製造方法 |
| JP4872076B2 (ja) * | 2005-09-15 | 2012-02-08 | 国立大学法人 長崎大学 | 硝子体可視化剤 |
| US20070155823A1 (en) * | 2005-12-19 | 2007-07-05 | Smith-Swintosky Virginia L | Use of benzo-fused heterocycle sulfamide derivatives as neuroprotective agents |
| US8497298B2 (en) | 2005-12-19 | 2013-07-30 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels |
| US8937096B2 (en) | 2005-12-19 | 2015-01-20 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder |
| US8691867B2 (en) | 2005-12-19 | 2014-04-08 | Janssen Pharmaceutica Nv | Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction |
| AU2007253814A1 (en) | 2006-05-19 | 2007-11-29 | Janssen Pharmaceutica N.V. | Co-therapy for the treatment of epilepsy |
| US8969415B2 (en) | 2006-12-01 | 2015-03-03 | Allergan, Inc. | Intraocular drug delivery systems |
| WO2008075148A2 (fr) * | 2006-12-15 | 2008-06-26 | Pfizer Products Inc. | Inhibiteurs tricycliques d'anhydrase carbonique |
| BRPI0906797A2 (pt) * | 2008-01-09 | 2015-07-14 | Molecular Insight Pharm Inc | Inibidores de anidrase carbônica ix |
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-
2002
- 2002-08-07 US US10/213,793 patent/US20030100594A1/en not_active Abandoned
-
2003
- 2003-02-14 BR BR0313282-0A patent/BR0313282A/pt not_active IP Right Cessation
- 2003-02-14 WO PCT/US2003/004469 patent/WO2004014430A1/fr not_active Ceased
- 2003-02-14 AU AU2003225571A patent/AU2003225571A1/en not_active Abandoned
- 2003-02-14 EP EP03709105A patent/EP1526895A2/fr not_active Withdrawn
- 2003-02-14 CA CA002495502A patent/CA2495502A1/fr not_active Abandoned
- 2003-02-14 CN CNA038218801A patent/CN1681557A/zh active Pending
- 2003-02-14 KR KR1020057002072A patent/KR20050056189A/ko not_active Ceased
- 2003-02-14 CA CA002495516A patent/CA2495516A1/fr not_active Abandoned
- 2003-02-14 WO PCT/US2003/004494 patent/WO2004014352A2/fr not_active Ceased
- 2003-02-14 JP JP2004527531A patent/JP2005539023A/ja not_active Withdrawn
- 2003-02-14 EP EP03784730A patent/EP1526869A1/fr not_active Withdrawn
- 2003-02-14 MX MXPA05001497A patent/MXPA05001497A/es not_active Application Discontinuation
- 2003-02-14 MX MXPA05001496A patent/MXPA05001496A/es not_active Application Discontinuation
- 2003-02-14 PL PL03374994A patent/PL374994A1/xx unknown
- 2003-02-14 BR BR0313299-4A patent/BR0313299A/pt not_active IP Right Cessation
- 2003-02-14 AU AU2003213062A patent/AU2003213062A1/en not_active Abandoned
- 2003-02-14 JP JP2004527530A patent/JP2005539022A/ja not_active Withdrawn
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2004
- 2004-04-19 US US10/827,075 patent/US20040198781A1/en not_active Abandoned
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2005
- 2005-02-03 IL IL16668505A patent/IL166685A0/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20040198781A1 (en) | 2004-10-07 |
| PL374994A1 (en) | 2005-11-14 |
| CA2495516A1 (fr) | 2004-02-19 |
| EP1526895A2 (fr) | 2005-05-04 |
| BR0313282A (pt) | 2005-10-18 |
| BR0313299A (pt) | 2005-06-14 |
| US20030100594A1 (en) | 2003-05-29 |
| EP1526869A1 (fr) | 2005-05-04 |
| MXPA05001497A (es) | 2005-05-27 |
| WO2004014352A2 (fr) | 2004-02-19 |
| JP2005539022A (ja) | 2005-12-22 |
| WO2004014430A1 (fr) | 2004-02-19 |
| JP2005539023A (ja) | 2005-12-22 |
| AU2003213062A1 (en) | 2004-02-25 |
| AU2003225571A1 (en) | 2004-02-25 |
| WO2004014352A3 (fr) | 2004-09-10 |
| CA2495502A1 (fr) | 2004-02-19 |
| KR20050056189A (ko) | 2005-06-14 |
| MXPA05001496A (es) | 2005-05-16 |
| CN1681557A (zh) | 2005-10-12 |
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