IL156813A0 - Imidazolyl derivatives and pharmaceutical compositions containing the same - Google Patents

Imidazolyl derivatives and pharmaceutical compositions containing the same

Info

Publication number: IL156813A0
Authority: IL; Israel
Prior art keywords: same; pharmaceutical compositions; compositions containing; imidazolyl derivatives; imidazolyl
Prior art date: 2001-01-26

Application number

IL15681302A

Other languages

English (en)

Original Assignee

Bristol Myers Squibb Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-01-26

Filing date

2002-01-11

Publication date

2004-02-08

2002-01-11 Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co

2004-02-08 Publication of IL156813A0 publication Critical patent/IL156813A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/06—Antiabortive agents; Labour repressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Psychiatry (AREA)
Addiction (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Orthopedic Medicine & Surgery (AREA)
Diabetes (AREA)
Pregnancy & Childbirth (AREA)
Gynecology & Obstetrics (AREA)
Hospice & Palliative Care (AREA)
Obesity (AREA)
Hematology (AREA)
Child & Adolescent Psychology (AREA)
Anesthesiology (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Nutrition Science (AREA)

IL15681302A 2001-01-26 2002-01-11 Imidazolyl derivatives and pharmaceutical compositions containing the same IL156813A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US26457001P	2001-01-26	2001-01-26
PCT/US2002/000841 WO2002058704A1 (en)	2001-01-26	2002-01-11	Imidazolyl derivatives as corticotropin releasing factor inhibitors

Publications (1)

Publication Number	Publication Date
IL156813A0 true IL156813A0 (en)	2004-02-08

Family

ID=23006646

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL15681302A IL156813A0 (en)	2001-01-26	2002-01-11	Imidazolyl derivatives and pharmaceutical compositions containing the same

Country Status (22)

Country	Link
US (5)	US6888004B2 (es)
EP (1)	EP1359916A4 (es)
JP (1)	JP2004531475A (es)
KR (1)	KR20040034594A (es)
CN (1)	CN1499972A (es)
BG (1)	BG107999A (es)
BR (1)	BR0206698A (es)
CA (1)	CA2434558A1 (es)
CZ (1)	CZ20032044A3 (es)
EE (1)	EE200300342A (es)
HR (1)	HRP20030675A2 (es)
HU (1)	HUP0303721A2 (es)
IL (1)	IL156813A0 (es)
IS (1)	IS6889A (es)
MX (1)	MXPA03006484A (es)
NO (1)	NO20033350L (es)
PE (1)	PE20020844A1 (es)
PL (1)	PL368555A1 (es)
RU (1)	RU2003126188A (es)
SK (1)	SK9222003A3 (es)
WO (1)	WO2002058704A1 (es)
ZA (1)	ZA200305531B (es)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BR0206698A (pt) *	2001-01-26	2004-04-20	Bristol Myers Squibb Co	Derivados de imidazolila como inibidores de fator de liberação de corticotropina.
TWI312347B (en)	2001-02-08	2009-07-21	Eisai R&D Man Co Ltd	Bicyclic nitrogen-containing condensed ring compounds
KR100881647B1 (ko)	2001-04-27	2009-02-04	에자이 알앤드디 매니지먼트 가부시키가이샤	피라졸로[1,5-ａ]피리딘 화합물 및 그 의약
US7176216B2 (en)	2002-10-22	2007-02-13	Eisai Co., Ltd.	7-phenylpyrazolopyridine compounds
PT1555265E (pt)	2002-10-22	2009-05-12	Eisai R&D Man Co Ltd	Compostos de 7-fenil pirazolopiridina
WO2006065793A2 (en) *	2004-12-13	2006-06-22	Indevus Pharmaceuticals, Inc.	TREATMENT OF INTERSTITIAL CYSTITIS USING (6aR,10aR)-Δ8-TETRAHYDROCANNABINOL-11-OIC ACIDS
WO2007090087A2 (en) *	2006-01-27	2007-08-09	Research Development Foundation	Use of corticotropin releasing factor receptor-2 inhibitors for treating insulin-related diseases
EP2522351B1 (en)	2007-06-13	2017-09-06	Research Development Foundation	Treatment and prevention of tauopathies and amyloid beta amyloidosis by modulating CRF receptor signaling
EP2225238B1 (en) *	2007-11-29	2014-09-03	Boehringer Ingelheim International GmbH	Derivatives of 6,7-dihydro-5h-imidazoý1,2- ¨imidazole-3- carboxylic acid amides
ES2396126T3 (es)	2008-04-15	2013-02-19	Eisai R&D Management Co., Ltd.	Compuesto de 3-fenilpirazol[5,1-b]tiazol
US7994203B2 (en) *	2008-08-06	2011-08-09	Novartis Ag	Organic compounds
AR078521A1 (es)	2009-10-08	2011-11-16	Eisai R&D Man Co Ltd	Compuesto pirazolotiazol
JP2013518085A (ja) *	2010-02-01	2013-05-20	ノバルティスアーゲー	ＣＲＦ−１受容体アンタゴニストとしてのピラゾロ［５，１ｂ］オキサゾール誘導体
US9806270B2 (en)	2011-03-25	2017-10-31	Udc Ireland Limited	4H-imidazo[1,2-a]imidazoles for electronic applications
JP6072760B2 (ja) *	2011-03-25	2017-02-01	ユー・ディー・シーアイルランドリミテッド	エレクトロニクス用途のための４Ｈ−イミダゾ［１，２−ａ］イミダゾール
CN108440531B (zh)	2011-11-10	2021-11-02	Udc 爱尔兰有限责任公司	用于电子应用的4H-咪唑并[1,2-a]咪唑
TWI644888B (zh)	2012-02-07	2018-12-21	拜耳智慧財產有限公司	用於製備經取代之鄰胺苯甲酸衍生物之方法
IN2014DN10229A (es)	2012-05-25	2015-08-07	Nutech Ventures
JP6231561B2 (ja)	2012-07-10	2017-11-15	ユー・ディー・シーアイルランドリミテッド	電子用途のためのベンズイミダゾ［１，２−ａ］ベンズイミダゾール誘導体
CN104718213B (zh) *	2012-07-18	2018-02-27	圣母大学	5,5‑杂芳族抗感染化合物
US20140206667A1 (en)	2012-11-14	2014-07-24	Michela Gallagher	Methods and compositions for treating schizophrenia
CN105384691B (zh) *	2015-10-26	2018-06-29	深圳大学	一种谷氨酰胺酰基环化酶抑制剂的制备方法及应用
US11214550B2 (en)	2017-07-24	2022-01-04	University Of South Florida	Bis-cyclic guanidines as antibacterial agents
WO2019169113A1 (en) *	2018-03-02	2019-09-06	Ponce Medical School Foundation, Inc.	Compositions and methods for the treatment of endometriosis

Family Cites Families (30)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3865836A (en) *	1972-12-08	1975-02-11	Janssen Pharmaceutica Nv	Bicyclic imidazoles
DE2827617A1 (de) *	1978-06-23	1980-01-10	Boehringer Sohn Ingelheim	Neue imidazo eckige klammer auf 1,2- alpha eckige klammer zu imidazole, deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung
IL69417A (en) *	1982-08-27	1987-12-20	Roussel Uclaf	2-acyl imidazo(1,2-a)pyrimidines,their preparation and pharmaceutical compositions containing them
US4551530A (en) *	1984-11-19	1985-11-05	American Cyanamid Company	Pyridyl imidazo[1,2-a]pyrimidines
DK155524C (da) *	1987-03-18	1989-09-11	Ferrosan As	Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
JPH05107705A (ja) *	1991-10-17	1993-04-30	Konica Corp	新規な写真用カプラー
ATE172975T1 (de) *	1992-05-19	1998-11-15	Adir	Benzimidezolderivate mit antidiabetischer und anti-plättchenklumpungswirkung
EP0607076A1 (fr) *	1993-01-15	1994-07-20	Synthelabo	Dérivés de 9h-imidazo 1,2-a benzimidazole-3-acétamide à activité GABA
FR2722501B1 (fr) *	1994-07-13	1996-08-09	Synthelabo	Derives de 9h-imidazo(1,2-a)benzimidazole-3-acetamide, leur preparation et leur application en therapeutique
DE69628804T2 (de)	1995-12-08	2003-12-18	Pfizer Inc., New York	Substitutierte heterozyclische Derivate als CRF Antagonisten
KR100421626B1 (ko) *	1996-02-07	2004-05-20	뉴로크린 바이오사이언시즈 인코퍼레이티드	Crf수용체에대한길항제로서의피라졸로피리미딘
US6022978A (en)	1996-06-11	2000-02-08	Pfizer Inc.	Benzimidazole derivatives
AU4398597A (en) *	1996-10-03	1998-04-24	Nissan Chemical Industries Ltd.	Heterocycle-fused pyrimidinone derivatives and herbicides
AU6279598A (en)	1997-02-18	1998-09-08	Neurocrine Biosciences, Inc.	Biazacyclic CRF antagonists
EE04280B1 (et)	1997-07-03	2004-04-15	Dupont Pharmaceuticals Company	Imidasopürimidiinid ja imidasopüridiinid neuroloogiliste häirete käitlemiseks
WO1999010350A1 (en)	1997-08-22	1999-03-04	Du Pont Pharmaceuticals Company	NITROGEN SUBSTITUTED IMIDAZO[4,5-c]PYRAZOLES AS CORTICOTROPIN RELEASING HORMONE ANTAGONISTS
BR9803368A (pt)	1997-09-05	2001-04-24	Sumitomo Chemical Co	Derivados de perimidona e herbecidas contendo os mesmos
WO1999024038A1 (en) *	1997-11-07	1999-05-20	Johns Hopkins University	Methods for treatment of disorders of cardiac contractility
WO1999033831A1 (en) *	1997-12-26	1999-07-08	Takeda Chemical Industries, Ltd.	Nitrogen-containing heterocyclic compounds, their production and use
US6509338B1 (en)	1998-06-22	2003-01-21	Bristol-Myers Squibb Company	Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists
US6124463A (en)	1998-07-02	2000-09-26	Dupont Pharmaceuticals	Benzimidazoles as corticotropin release factor antagonists
US6365589B1 (en)	1998-07-02	2002-04-02	Bristol-Myers Squibb Pharma Company	Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
US6271380B1 (en)	1998-12-30	2001-08-07	Dupont Pharmaceuticals Company	1H-imidazo[4,5-d]pyridazin-7-ones, 3H-imidazo-[4,5-c]pyridin-4-ones and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands
WO2000059907A2 (en)	1999-04-06	2000-10-12	Du Pont Pharmaceuticals Company	Pyrazolotriazines as crf antagonists
WO2000059908A2 (en)	1999-04-06	2000-10-12	Du Pont Pharmaceuticals Company	Pyrazolopyrimidines as crf antagonists
US6492408B1 (en) *	1999-07-21	2002-12-10	Boehringer Ingelheim Pharmaceuticals, Inc.	Small molecules useful in the treatment of inflammatory disease
MXPA03000914A (es) *	2000-08-09	2003-10-06	Boehringer Ingelheim Pharma	Sintesis de (r)-3-(4 -bromobencil) -1-(3, 5-diclorofenil) -5-yodo-3 -metil-1-h -imidazo[1, 2-a]imidazol -2-ona.
US6696441B1 (en) *	2000-08-11	2004-02-24	The Regents Of The University Of California	Inhibition of p53-induced stress response
AU2001296255B2 (en) *	2000-09-21	2005-07-28	Bristol-Myers Squibb Company	Substituted azole derivatives as inhibitors of corticotropin releasing factor
BR0206698A (pt) *	2001-01-26	2004-04-20	Bristol Myers Squibb Co	Derivados de imidazolila como inibidores de fator de liberação de corticotropina.

2002
- 2002-01-11 BR BR0206698-0A patent/BR0206698A/pt not_active IP Right Cessation
- 2002-01-11 WO PCT/US2002/000841 patent/WO2002058704A1/en not_active Ceased
- 2002-01-11 PL PL02368555A patent/PL368555A1/xx unknown
- 2002-01-11 EP EP02705754A patent/EP1359916A4/en not_active Withdrawn
- 2002-01-11 IL IL15681302A patent/IL156813A0/xx unknown
- 2002-01-11 US US10/044,183 patent/US6888004B2/en not_active Expired - Lifetime
- 2002-01-11 CA CA002434558A patent/CA2434558A1/en not_active Abandoned
- 2002-01-11 CN CNA028071352A patent/CN1499972A/zh active Pending
- 2002-01-11 KR KR10-2003-7009883A patent/KR20040034594A/ko not_active Withdrawn
- 2002-01-11 JP JP2002559038A patent/JP2004531475A/ja active Pending
- 2002-01-11 HU HU0303721A patent/HUP0303721A2/hu unknown
- 2002-01-11 RU RU2003126188/04A patent/RU2003126188A/ru not_active Application Discontinuation
- 2002-01-11 HR HR20030675A patent/HRP20030675A2/hr not_active Application Discontinuation
- 2002-01-11 EE EEP200300342A patent/EE200300342A/xx unknown
- 2002-01-11 MX MXPA03006484A patent/MXPA03006484A/es unknown
- 2002-01-11 SK SK922-2003A patent/SK9222003A3/sk unknown
- 2002-01-11 CZ CZ20032044A patent/CZ20032044A3/cs unknown
- 2002-01-25 PE PE2002000063A patent/PE20020844A1/es not_active Application Discontinuation
2003
- 2003-07-17 BG BG107999A patent/BG107999A/xx unknown
- 2003-07-17 ZA ZA200305531A patent/ZA200305531B/en unknown
- 2003-07-24 IS IS6889A patent/IS6889A/is unknown
- 2003-07-25 NO NO20033350A patent/NO20033350L/no not_active Application Discontinuation
2004
- 2004-01-29 US US10/767,645 patent/US7211669B2/en not_active Expired - Lifetime
- 2004-02-04 US US10/771,766 patent/US7238699B2/en not_active Expired - Lifetime
- 2004-02-04 US US10/772,027 patent/US7244746B2/en not_active Expired - Lifetime
- 2004-02-04 US US10/771,661 patent/US7125990B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
SK9222003A3 (en)	2004-05-04
KR20040034594A (ko)	2004-04-28
US7238699B2 (en)	2007-07-03
US7211669B2 (en)	2007-05-01
US7244746B2 (en)	2007-07-17
PE20020844A1 (es)	2002-09-27
CA2434558A1 (en)	2002-08-01
US20020183375A1 (en)	2002-12-05
NO20033350D0 (no)	2003-07-25
HRP20030675A2 (en)	2004-08-31
PL368555A1 (en)	2005-04-04
ZA200305531B (en)	2004-07-27
BR0206698A (pt)	2004-04-20
MXPA03006484A (es)	2003-09-22
NO20033350L (no)	2003-09-22
BG107999A (en)	2004-08-31
US20040235924A1 (en)	2004-11-25
US7125990B2 (en)	2006-10-24
US6888004B2 (en)	2005-05-03
EP1359916A1 (en)	2003-11-12
US20040225130A1 (en)	2004-11-11
US20040254382A1 (en)	2004-12-16
US20040225001A1 (en)	2004-11-11
CZ20032044A3 (cs)	2003-12-17
JP2004531475A (ja)	2004-10-14
HUP0303721A2 (hu)	2004-03-01
WO2002058704A1 (en)	2002-08-01
CN1499972A (zh)	2004-05-26
IS6889A (is)	2003-07-24
EE200300342A (et)	2003-12-15
RU2003126188A (ru)	2005-03-27
EP1359916A4 (en)	2004-04-07

Publication	Publication Date	Title
IL161616A0 (en)	2004-09-27	Indazolypyrrolotriazine derivatives and pharmaceutical compositions containing the same
IL158044A0 (en)	2004-03-28	Cyclopropylindole derivatives and pharmaceutical compositions containing the same
IL158300A0 (en)	2004-05-12	Bisarylimidazol derivatives and pharmaceutical compositions containing the same
IL158041A0 (en)	2004-03-28	Benzimidazole derivatives and pharmaceutical compositions containing the same
IL156369A0 (en)	2004-01-04	Pyrazole derivatives and pharmaceutical compositions containing the same
IL154786A0 (en)	2003-10-31	Pyrazole derivatives and pharmaceutical compositions containing the same
IL145757A0 (en)	2002-07-25	Pyrazole derivatives and pharmaceutical compositions containing the same
IL145756A0 (en)	2002-07-25	Pyrazole derivatives and pharmaceutical compositions containing the same
IL164209A0 (en)	2005-12-18	Pyrazole derivatives and pharmaceutical compositions containing the same
IL166620A0 (en)	2006-01-15	Pyrazole derivatives and pharmaceutical compositions containing the same
IL152451A0 (en)	2003-05-29	2-chloro-2-nitrophenylcarboxamide derivatives and pharmaceutical compositions containing the same
HUP0301178A3 (en)	2009-08-28	Glucopyranosyloxybenzylbenzene derivatives and pharmaceutical compositions containing the same
IL153123A0 (en)	2003-06-24	N-ureidoheterocycloalkyl-piperidine derivatives and pharmaceutical compositions containing the same
IL158076A0 (en)	2004-03-28	Benzamidine derivatives and pharmaceutical compositions containing the same
IL156812A0 (en)	2004-02-08	Phthalazinone-piperidino derivatives and pharmaceutical compositions containing the same
IL162548A0 (en)	2005-11-20	4-Oxoquinoline derivatives and pharmaceutical compositions containing the same
IL156813A0 (en)	2004-02-08	Imidazolyl derivatives and pharmaceutical compositions containing the same
IL157131A0 (en)	2004-02-08	Nitrogen containing heterocyclic derivatives and pharmaceutical compositions containing the same
IL158523A0 (en)	2004-05-12	Epothilone derivatives and pharmaceutical compositions containing the same
IL163117A (en)	2010-05-31	Indazole derivatives and pharmaceutical compositions containing the same
IL166482A0 (en)	2006-01-15	Dihydropyrazolopyridine derivatives and pharmaceutical compositions containing the same
AU2002306269A1 (en)	2003-05-15	N-arylphenylacetamide derivatives and pharmaceutical composition containing the same
IL157029A0 (en)	2004-02-08	Azaindoleoxoacetic piperazine derivatives and pharmaceutical compositions containing the same
IL158671A0 (en)	2004-05-12	Benzyloxy derivatives and pharmaceutical compositions containing the same
IL157740A0 (en)	2004-03-28	Heterocyclic derivatives and pharmaceutical compositions containing the same