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GT201200289A - 3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas - Google Patents

3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas

Info

Publication number
GT201200289A
GT201200289A GT201200289A GT201200289A GT201200289A GT 201200289 A GT201200289 A GT 201200289A GT 201200289 A GT201200289 A GT 201200289A GT 201200289 A GT201200289 A GT 201200289A GT 201200289 A GT201200289 A GT 201200289A
Authority
GT
Guatemala
Prior art keywords
fungicides
substituted
dihydropirimidine
onas
imino
Prior art date
Application number
GT201200289A
Other languages
English (en)
Inventor
Boebel Timothy
Lorsbach Beth
Martin Timothy
Owen W John
Sullenberger Michael
Webster Jeffery
Yao Chenglin
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT201200289A publication Critical patent/GT201200289A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

LA PRESENTE INVENCIÓN ESTÁ RELACIONADA CON EL CAMPO DE N3-SUSTITUIDO-N1-SULFONIL-5-FLÚORPIRIMIDINONA Y SUS DERIVADOS Y EL USO DE ESTOS COMPUESTOS COMO FUNGICIDAS.
GT201200289A 2010-04-26 2012-10-25 3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas GT201200289A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32785510P 2010-04-26 2010-04-26

Publications (1)

Publication Number Publication Date
GT201200289A true GT201200289A (es) 2014-04-08

Family

ID=44816310

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201200289A GT201200289A (es) 2010-04-26 2012-10-25 3-sustituido-5-fluoro-4-imino-3,4-dihidropirimidina-2-(1h)-onas como fungicidas

Country Status (33)

Country Link
US (1) US8263603B2 (es)
EP (1) EP2563129B1 (es)
JP (1) JP5784705B2 (es)
KR (1) KR101793766B1 (es)
CN (1) CN102946730B (es)
AU (1) AU2011245544B2 (es)
BR (1) BR112012027439B1 (es)
CA (1) CA2797226C (es)
CL (1) CL2012002979A1 (es)
CO (1) CO6592042A2 (es)
CR (1) CR20120584A (es)
CY (1) CY1117956T1 (es)
DK (1) DK2563129T3 (es)
EC (1) ECSP12012302A (es)
ES (1) ES2588742T3 (es)
GT (1) GT201200289A (es)
HN (1) HN2012002272A (es)
HR (1) HRP20161107T1 (es)
HU (1) HUE029489T2 (es)
IL (1) IL222646A (es)
LT (1) LT2563129T (es)
ME (1) ME02530B (es)
MX (1) MX2012012530A (es)
NZ (1) NZ603151A (es)
PH (1) PH12012502138B1 (es)
PL (1) PL2563129T3 (es)
PT (1) PT2563129T (es)
RS (1) RS55239B1 (es)
RU (1) RU2562840C2 (es)
SI (1) SI2563129T1 (es)
SM (1) SMT201600298B (es)
UA (1) UA108101C2 (es)
WO (1) WO2011137002A1 (es)

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UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону
US9321734B2 (en) * 2012-12-28 2016-04-26 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives
HK1214518A1 (zh) * 2012-12-28 2016-07-29 Adama Makhteshim Ltd. 1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3，4-二氢嘧啶-2(1h)-酮衍生物
US9622474B2 (en) * 2012-12-28 2017-04-18 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylate derivatives
AU2013370494B2 (en) * 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
EA030056B1 (ru) * 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
CN106068268A (zh) * 2013-12-31 2016-11-02 阿达玛马克西姆股份有限公司 5‑氟‑4‑亚氨基‑3‑（烷基/取代烷基）‑1‑（芳基磺酰基）‑3,4‑二氢嘧啶‑2（1h）‑酮及其制备方法
MA41272A (fr) * 2014-12-23 2017-10-31 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences
JP6862939B2 (ja) * 2016-03-11 2021-04-21 住友化学株式会社 植物病害防除組成物及び植物病害防除方法
US11051513B2 (en) 2017-01-26 2021-07-06 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
JP7134946B2 (ja) 2017-04-10 2022-09-12 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
JP7168556B2 (ja) 2017-04-10 2022-11-09 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
TWI771402B (zh) 2017-04-11 2022-07-21 日商三井化學Agro股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
WO2018225829A1 (ja) 2017-06-08 2018-12-13 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
MA49639A (fr) 2017-07-17 2020-05-27 Adama Makhteshim Ltd Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
CR20210270A (es) * 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
IL321760A (en) 2019-07-22 2025-08-01 Adama Makhteshim Ltd Fungicidal combinations, mixtures and compositions and uses thereof
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound
EP4118073A1 (en) * 2020-03-09 2023-01-18 Adama Makhteshim Ltd. Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one
CN116113623A (zh) * 2020-05-04 2023-05-12 阿达玛马克西姆有限公司 包含5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的混合物及组合物，及其使用方法
EP4178358A1 (en) 2020-07-08 2023-05-17 Adama Makhteshim Ltd. Fungicidal mixtures
CA3206570A1 (en) 2021-01-27 2022-08-04 Alexandra ROSENMUND 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases
CA3216622A1 (en) 2021-05-04 2022-11-10 Stefano Luca Giaffreda Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
IL311455A (en) * 2021-09-15 2024-05-01 Adama Makhteshim Ltd Method for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-H1-pyrimidin-2-one
CN118555910A (zh) * 2022-01-12 2024-08-27 安道麦马克西姆有限公司 包含含有邻苯二甲酰亚胺杀真菌剂的组合的杀真菌混合物
AU2023227455A1 (en) 2022-03-03 2024-09-19 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2023275068A1 (en) 2022-05-26 2024-11-28 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2024189563A1 (en) 2023-03-14 2024-09-19 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
IL308593A (en) 2023-11-15 2025-06-01 Adama Makhteshim Ltd Reducing environmental impact of fungicidal enhancement
WO2025114931A1 (en) 2023-11-28 2025-06-05 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

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HRP970239B1 (en) * 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US20090163567A1 (en) * 2005-11-22 2009-06-25 Ishihara Sangyo Kaisha, Ltd Germicide composition for agricultural and gardening applications and method for controlling plant disease
PT2252594E (pt) * 2008-01-22 2015-11-30 Dow Agrosciences Llc Derivados de 5-fluoro-pirimidina como fungicidas
UA107651C2 (en) * 2008-08-01 2015-02-10 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону

Also Published As

Publication number Publication date
UA108101C2 (xx) 2015-03-25
HUE029489T2 (en) 2017-02-28
PT2563129T (pt) 2016-09-05
BR112012027439A2 (pt) 2015-09-15
CA2797226C (en) 2019-02-26
PL2563129T3 (pl) 2017-08-31
CN102946730A (zh) 2013-02-27
RU2012150293A (ru) 2014-06-10
CL2012002979A1 (es) 2013-01-25
EP2563129A1 (en) 2013-03-06
EP2563129B1 (en) 2016-06-01
JP5784705B2 (ja) 2015-09-24
IL222646A0 (en) 2012-12-31
KR20130093000A (ko) 2013-08-21
PH12012502138A1 (en) 2013-02-04
ECSP12012302A (es) 2012-12-28
CA2797226A1 (en) 2011-11-03
AU2011245544A1 (en) 2012-11-15
ES2588742T3 (es) 2016-11-04
US20110263627A1 (en) 2011-10-27
LT2563129T (lt) 2016-10-25
WO2011137002A1 (en) 2011-11-03
SMT201600298B (it) 2016-11-10
CY1117956T1 (el) 2017-05-17
KR101793766B1 (ko) 2017-11-03
US8263603B2 (en) 2012-09-11
BR112012027439A8 (pt) 2017-07-11
SI2563129T1 (sl) 2016-12-30
MX2012012530A (es) 2012-12-17
NZ603151A (en) 2013-10-25
RU2562840C2 (ru) 2015-09-10
IL222646A (en) 2017-01-31
HN2012002272A (es) 2015-04-27
DK2563129T3 (en) 2016-09-12
AU2011245544B2 (en) 2015-04-16
HRP20161107T1 (hr) 2016-12-30
CN102946730B (zh) 2015-02-04
CR20120584A (es) 2013-01-03
BR112012027439B1 (pt) 2018-01-16
ME02530B (me) 2017-02-20
CO6592042A2 (es) 2013-01-02
RS55239B1 (sr) 2017-02-28
EP2563129A4 (en) 2013-08-07
PH12012502138B1 (en) 2019-09-25
HK1182594A1 (en) 2013-12-06
JP2013525434A (ja) 2013-06-20

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