GT200600332A - Inhibidores de 6-alquiliden-penem beta-lactamasa triciclicos y combinación de antibióticos de b-lactama: un antibiotico de amplio espectro - Google Patents
Inhibidores de 6-alquiliden-penem beta-lactamasa triciclicos y combinación de antibióticos de b-lactama: un antibiotico de amplio espectroInfo
- Publication number
- GT200600332A GT200600332A GT200600332A GT200600332A GT200600332A GT 200600332 A GT200600332 A GT 200600332A GT 200600332 A GT200600332 A GT 200600332A GT 200600332 A GT200600332 A GT 200600332A GT 200600332 A GT200600332 A GT 200600332A
- Authority
- GT
- Guatemala
- Prior art keywords
- lactama
- lactamasa
- alquiliden
- penem
- tricycles
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/424—Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
- A61K31/431—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems containing further heterocyclic rings, e.g. ticarcillin, azlocillin, oxacillin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
LA PRESENTE INVENCIÓN PROPORCIONA UN ANTIBIÓTICO DE B-LACTAMA TAL COMO CEFEPIME Y UN COMPUESTO DE LA FÓRMULA I, COMPOSICIONES FARMACÉUTICAS Y EL USO DEL MISMO PARA EL TRATAMIENTO DE INFECCIÓN O ENFERMEDAD BACTERIANA EN UN PACIENTE QUE NECESITE DEL MISMO.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US70280805P | 2005-07-27 | 2005-07-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT200600332A true GT200600332A (es) | 2007-03-14 |
Family
ID=37809337
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT200600332A GT200600332A (es) | 2005-07-27 | 2006-07-26 | Inhibidores de 6-alquiliden-penem beta-lactamasa triciclicos y combinación de antibióticos de b-lactama: un antibiotico de amplio espectro |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20070027130A1 (es) |
| EP (1) | EP1909786A2 (es) |
| JP (1) | JP2009502932A (es) |
| CN (1) | CN101257902A (es) |
| AR (1) | AR055097A1 (es) |
| AU (1) | AU2006285308A1 (es) |
| BR (1) | BRPI0613928A2 (es) |
| CA (1) | CA2616468A1 (es) |
| GT (1) | GT200600332A (es) |
| MX (1) | MX2008001083A (es) |
| PE (1) | PE20070342A1 (es) |
| TW (1) | TW200738235A (es) |
| WO (1) | WO2007027323A2 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR039475A1 (es) * | 2002-05-01 | 2005-02-23 | Wyeth Corp | 6-alquiliden-penems triciclicos como inhibidores de beta-lactamasa |
| CN101798315B (zh) * | 2008-10-06 | 2012-07-04 | 山东轩竹医药科技有限公司 | 含有环丙烷并氮杂环的头孢菌素衍生物 |
| US20110288063A1 (en) * | 2010-05-19 | 2011-11-24 | Naeja Pharmaceutical Inc. | Novel fused bridged bicyclic heteroaryl substituted 6-alkylidene penems as potent beta-lactamase inhibitors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4206067A (en) * | 1978-10-02 | 1980-06-03 | Chevron Research Company | Thermally stabilized erosion-inhibited functional fluids containing perhalometal compounds and an organic base |
| DE3176517D1 (en) * | 1980-04-24 | 1987-12-17 | Beecham Group Plc | Beta-lactam compounds, their preparation and use |
| US4891369A (en) * | 1986-12-03 | 1990-01-02 | Taiho Pharmaceutical Company, Limited | 2β-Substituted-methylpenicillanic acid derivatives, and salts and esters thereof |
| JP3865770B2 (ja) * | 1994-04-25 | 2007-01-10 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | ベータ−ラクタム抗生物質と組み合わせてベータ−ラクタマーゼ阻害性ペネムを含有する医薬製剤および細菌感染の治療におけるそれらの使用 |
| US5464616A (en) * | 1994-08-04 | 1995-11-07 | Synphar Laboratories, Ind. | 6β-substituted penicillanic acids as beta-lactamase inhibitors |
| CA2346813A1 (en) * | 1998-10-15 | 2000-04-20 | Sarawak Medichem Pharmaceuticals Incorporated | Method and composition for treating and preventing tuberculosis |
| GB9928290D0 (en) * | 1999-12-01 | 2000-01-26 | Univ Belfast | Process for preparing ambient temperature ionic liquids |
| AR039475A1 (es) * | 2002-05-01 | 2005-02-23 | Wyeth Corp | 6-alquiliden-penems triciclicos como inhibidores de beta-lactamasa |
| US20040132708A1 (en) * | 2002-05-01 | 2004-07-08 | Wyeth | Process for preparing 6-alkylidene penem derivatives |
| AR039476A1 (es) * | 2002-05-01 | 2005-02-23 | Wyeth Corp | Proceso para preparar derivados de 6-alquiliden penem |
| AR039774A1 (es) * | 2002-05-01 | 2005-03-02 | Wyeth Corp | 6-alquiliden-penems biciclicos como inhibidores de beta-lactamasas |
| AR046041A1 (es) * | 2003-10-03 | 2005-11-23 | Aventis Pharma Inc | Procedimiento para la preparacion de compuestos heterociclicos n-amino sustituidos |
-
2006
- 2006-07-26 JP JP2008524076A patent/JP2009502932A/ja not_active Withdrawn
- 2006-07-26 CA CA002616468A patent/CA2616468A1/en not_active Abandoned
- 2006-07-26 AU AU2006285308A patent/AU2006285308A1/en not_active Abandoned
- 2006-07-26 BR BRPI0613928-0A patent/BRPI0613928A2/pt not_active Application Discontinuation
- 2006-07-26 US US11/493,331 patent/US20070027130A1/en not_active Abandoned
- 2006-07-26 PE PE2006000908A patent/PE20070342A1/es not_active Application Discontinuation
- 2006-07-26 MX MX2008001083A patent/MX2008001083A/es unknown
- 2006-07-26 WO PCT/US2006/028883 patent/WO2007027323A2/en not_active Ceased
- 2006-07-26 GT GT200600332A patent/GT200600332A/es unknown
- 2006-07-26 CN CNA2006800322600A patent/CN101257902A/zh active Pending
- 2006-07-26 EP EP06824782A patent/EP1909786A2/en not_active Withdrawn
- 2006-07-26 TW TW095127308A patent/TW200738235A/zh unknown
- 2006-07-27 AR ARP060103241A patent/AR055097A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2009502932A (ja) | 2009-01-29 |
| BRPI0613928A2 (pt) | 2011-02-15 |
| TW200738235A (en) | 2007-10-16 |
| WO2007027323A3 (en) | 2007-05-31 |
| WO2007027323A2 (en) | 2007-03-08 |
| US20070027130A1 (en) | 2007-02-01 |
| CA2616468A1 (en) | 2007-03-08 |
| MX2008001083A (es) | 2008-03-19 |
| PE20070342A1 (es) | 2007-05-08 |
| EP1909786A2 (en) | 2008-04-16 |
| AR055097A1 (es) | 2007-08-08 |
| AU2006285308A1 (en) | 2007-03-08 |
| CN101257902A (zh) | 2008-09-03 |
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