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Publication of GT200300090ApublicationCriticalpatent/GT200300090A/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
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Acyclic And Carbocyclic Compounds In Medicinal Compositions
(AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A COMPUESTOS DE FORMULA GENERAL I EN DONDE R1,R2,R3,R4,R5,R6,R14, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS TIENEN ACTIVIDAD ADRENERGICA SELECTIVA SOBRE LOS RECEPTORES ALFA Y POR LO TANTO SON DE UTILIDAD EN UNA AMPLIA VARIEDAD DE CUADROS TALES COMO INCONTINENCIA URINARIA, CONGESTION NASAL, DISFUNCION SEXUAL ENTRE OTRAS DESCRITAS EN LA SOLICITUD.THE PRESENT INVENTION CONCERNS COMPOUNDS OF GENERAL FORMULA I WHERE R1, R2, R3, R4, R5, R6, R14, ARE FUNCTIONAL GROUPS DESCRIBED IN THE RECORD. THESE COMPOUNDS HAVE SELECTIVE ADRENERGIC ACTIVITY ON ALFA RECEPTORS AND THEREFORE ARE USEFUL IN A LARGE VARIETY OF TABLES AS URINARY INCONTINENCE, NASAL CONGESTION, SEXUAL DYSFUNCTION BETWEEN OTHER DESCRIBED IN THE APPLICATION.