GB2039277B - Preparation of pharmacologically-active piperidylindoles - Google Patents

Preparation of pharmacologically-active piperidylindoles

Info

Publication number: GB2039277B
Authority: GB; United Kingdom
Prior art keywords: piperidylindoles; pharmacologically; active; preparation; active piperidylindoles
Prior art date: 1978-12-22
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

GB7944358A

Other versions

GB2039277A (en

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sanofi Aventis France

Original Assignee

Roussel Uclaf SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-12-22

Filing date

1979-12-24

Publication date

1983-03-02

1979-12-24 Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA

1980-08-06 Publication of GB2039277A publication Critical patent/GB2039277A/en

1983-03-02 Application granted granted Critical

1983-03-02 Publication of GB2039277B publication Critical patent/GB2039277B/en

Status Expired legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Catalysts (AREA)

GB7944358A 1978-12-22 1979-12-24 Preparation of pharmacologically-active piperidylindoles Expired GB2039277B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR7836167A FR2444678A2 (en)	1978-12-22	1978-12-22	NOVEL PROCESS FOR THE PREPARATION OF PIPERIDYL-INDOLE DERIVATIVES AND THEIR SALTS

Publications (2)

Publication Number	Publication Date
GB2039277A GB2039277A (en)	1980-08-06
GB2039277B true GB2039277B (en)	1983-03-02

Family

ID=9216467

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
GB7944358A Expired GB2039277B (en)	1978-12-22	1979-12-24	Preparation of pharmacologically-active piperidylindoles

Country Status (17)

Country	Link
US (1)	US4232031A (en)
JP (1)	JPS5587786A (en)
AT (1)	AT375361B (en)
AU (1)	AU529439B2 (en)
BE (1)	BE880818A (en)
CA (1)	CA1128946A (en)
CH (1)	CH642963A5 (en)
DE (1)	DE2951912A1 (en)
ES (1)	ES487175A1 (en)
FR (1)	FR2444678A2 (en)
GB (1)	GB2039277B (en)
HU (1)	HU181947B (en)
IE (1)	IE49343B1 (en)
IT (1)	IT1164031B (en)
NL (1)	NL7909136A (en)
SE (1)	SE440651B (en)
ZA (1)	ZA796386B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2420536A1 (en) *	1978-03-22	1979-10-19	Roussel Uclaf	NEW DERIVATIVES OF 1,3-DIHYDRO 3- / 1- / 2- (2,3-DIHYDRO 1,4-BENZODIOXIN-2-YL) 2-HYDROXYETHYL / PIPERIDIN-4-YL / 2H-INDOL-2-ONE, PROCESS FOR THEIR PREPARATION AND APPLICATION AS MEDICINAL PRODUCTS
SE8004129L (en) *	1979-07-13	1981-01-14	Roussel Uclaf	NEW TETRAHYDROPYRIDIN-4-YL-INDOLD DERIVATIVES AND SALTS THEREOF, PREPARATION AND USE THEREOF AS A MEDICINAL PRODUCT AND COMPOSITIONS CONTAINING THESE COMPOUNDS
FR2460947A1 (en) *	1979-07-13	1981-01-30	Roussel Uclaf	NOVEL N-SUBSTITUTED TETRAHYDROPYRIDINYL-INDOLE DERIVATIVES, THEIR SALTS, PREPARATION METHOD, MEDICAMENT APPLICATION AND COMPOSITIONS COMPRISING SAME
IE58370B1 (en) *	1985-04-10	1993-09-08	Lundbeck & Co As H	Indole derivatives
WO1990007926A1 (en) *	1989-01-20	1990-07-26	Pfizer Inc.	3-(1,2,5,6-tetrahydropyridyl)-pyrrolopyridines
US5846982A (en) *	1996-06-14	1998-12-08	Eli Lilly And Company	Inhibition of serotonin reuptake
WO2004069828A1 (en) *	2003-02-04	2004-08-19	Mitsubishi Pharma Corporation	Piperidine compound and medicinal use thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2872453A (en) *		1959-02-03		Indole derivatives
FR2193584B1 (en) *	1972-07-28	1975-08-08	Roussel Uclaf
DE2322470A1 (en) *	1973-05-04	1974-11-21	Boehringer Sohn Ingelheim	NEW INDOLYL-PIPERIDINO- (OR 1,2,5,6TETRAHYDRO-PYRIDYL-) BUTYROPHENONE AND METHOD FOR THEIR PRODUCTION
FR2258843B1 (en) *	1974-01-30	1977-09-09	Roussel Uclaf
IL48508A (en) *	1974-12-09	1979-10-31	Roussel Uclaf	Pharmaceutical compositions comprising piperidylindole derivatives
JPS5283766A (en) *	1976-01-01	1977-07-12	Roussel Uclaf	Piperidyl indole derivative and its salts and medicine comprising same
FR2349331A1 (en) *	1976-04-30	1977-11-25	Roussel Uclaf	NEW DERIVATIVES OF 2,3 DIHYDRO A / 4- (3-INDOLYL) 1-PIPERIDINYL / METHYL 1,4-BENZODIOXIN-2-METHANOL, A PROCESS FOR THEIR PREPARATION AND APPLICATION AS MEDICINAL PRODUCTS
FR2362628A1 (en) *	1976-08-26	1978-03-24	Roussel Uclaf	NEW DERIVATIVES OF PIPERIDYL-INDOLE AND THEIR SALTS, METHOD OF PREPARATION AND APPLICATION AS MEDICINAL PRODUCTS

1978
- 1978-12-22 FR FR7836167A patent/FR2444678A2/en active Granted
1979
- 1979-11-13 SE SE7909367A patent/SE440651B/en not_active IP Right Cessation
- 1979-11-26 ZA ZA00796386A patent/ZA796386B/en unknown
- 1979-11-27 HU HU79RO1048A patent/HU181947B/en not_active IP Right Cessation
- 1979-12-06 US US06/100,909 patent/US4232031A/en not_active Expired - Lifetime
- 1979-12-18 JP JP16364679A patent/JPS5587786A/en active Granted
- 1979-12-19 NL NL7909136A patent/NL7909136A/en not_active Application Discontinuation
- 1979-12-20 CA CA342,441A patent/CA1128946A/en not_active Expired
- 1979-12-21 AU AU54152/79A patent/AU529439B2/en not_active Ceased
- 1979-12-21 BE BE0/198712A patent/BE880818A/en not_active IP Right Cessation
- 1979-12-21 IE IE2508/79A patent/IE49343B1/en unknown
- 1979-12-21 AT AT0809679A patent/AT375361B/en not_active IP Right Cessation
- 1979-12-21 CH CH1142679A patent/CH642963A5/en not_active IP Right Cessation
- 1979-12-21 IT IT51166/79A patent/IT1164031B/en active
- 1979-12-21 DE DE19792951912 patent/DE2951912A1/en active Granted
- 1979-12-21 ES ES487175A patent/ES487175A1/en not_active Expired
- 1979-12-24 GB GB7944358A patent/GB2039277B/en not_active Expired

Also Published As

Publication number	Publication date
AU5415279A (en)	1980-06-26
US4232031A (en)	1980-11-04
IT1164031B (en)	1987-04-08
SE440651B (en)	1985-08-12
NL7909136A (en)	1980-06-24
HU181947B (en)	1983-11-28
BE880818A (en)	1980-06-23
CH642963A5 (en)	1984-05-15
CA1128946A (en)	1982-08-03
FR2444678A2 (en)	1980-07-18
DE2951912C2 (en)	1989-05-11
AU529439B2 (en)	1983-06-09
ATA809679A (en)	1983-12-15
IT7951166A0 (en)	1979-12-21
JPS6345387B2 (en)	1988-09-09
AT375361B (en)	1984-07-25
IE792508L (en)	1980-06-22
DE2951912A1 (en)	1980-07-10
FR2444678B2 (en)	1982-09-17
GB2039277A (en)	1980-08-06
JPS5587786A (en)	1980-07-02
ES487175A1 (en)	1980-09-16
SE7909367L (en)	1980-06-23
IE49343B1 (en)	1985-09-18
ZA796386B (en)	1980-10-29

Publication	Publication Date	Title
GB2042507B (en)	1982-12-08	Preparation of fluoronitrobenzenes
GB2016449B (en)	1982-09-15	Preparation of cis-alkylcyclohexanols
PH15168A (en)	1982-08-31	Preparation of cis-hexahydrodibenzopyranones
IL58106A0 (en)	1979-12-30	The preparation of 4-fluoro-3-phenoxy-toluene
GB2034336B (en)	1983-03-30	Preparation of ethylene-butene
IL57350A0 (en)	1979-09-30	Preparation of acetanilides
GB2033910B (en)	1983-03-30	Preparation of ethylene-butene
GB2039277B (en)	1983-03-02	Preparation of pharmacologically-active piperidylindoles
IL56636A0 (en)	1979-05-31	Preparation of hydoxyphenyl ethers
DE2960517D1 (en)	1981-10-29	Preparation of 4-methyl-5-hydroxymethyl-imidazole
IL58778A (en)	1982-11-30	Preparation of 21-acylthiopregnenes
GB2037769B (en)	1983-05-05	Preparation of methyl-nonyl-acetaldehyde
GB2017106B (en)	1982-07-07	Preparation of sulphonium plymers
IL57507A0 (en)	1979-10-31	The preparation of 2-oximinophenylaceto-nitrile
GB2034713B (en)	1983-01-06	Preparation of amenophenol ether
IL58732A0 (en)	1980-02-29	Preparation of 3-phenoxy-benzaldehydes
GB2022091B (en)	1982-11-03	Preparation of isocyanates
IL57352A0 (en)	1979-09-30	Preparation of 2-isopropylamino-pyrimidine
JPS54133582A (en)	1979-10-17	Preparation of polymerpolyol
GB2038826B (en)	1983-03-23	Preparation of 2-methylenealdehydes
IL57423A (en)	1982-02-28	Furonaphthyridine compounds and their preparation
JPS54119532A (en)	1979-09-17	Preparation of dihydroquinacrydone
IL58268A0 (en)	1979-12-30	The preparation of nn-dimethylaminoacetonitrile
GB2023111B (en)	1982-12-22	Preparation of shaped bodies
JPS5541201A (en)	1980-03-24	Preparation of honeycomb

Legal Events

Date	Code	Title	Description
1992-08-19	PCNP	Patent ceased through non-payment of renewal fee