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GB1011311A - Antiparasitic compositions and use thereof - Google Patents

Antiparasitic compositions and use thereof

Info

Publication number
GB1011311A
GB1011311A GB26608/63A GB2660863A GB1011311A GB 1011311 A GB1011311 A GB 1011311A GB 26608/63 A GB26608/63 A GB 26608/63A GB 2660863 A GB2660863 A GB 2660863A GB 1011311 A GB1011311 A GB 1011311A
Authority
GB
United Kingdom
Prior art keywords
chloro
hydroxy
formula
salt
phenoxide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB26608/63A
Inventor
Charles Sidney Franklin
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Parke Davis and Co LLC
Original Assignee
Parke Davis and Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Parke Davis and Co LLC filed Critical Parke Davis and Co LLC
Priority to GB26608/63A priority Critical patent/GB1011311A/en
Priority to US375638A priority patent/US3253986A/en
Publication of GB1011311A publication Critical patent/GB1011311A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/475Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Imidazo - [1,2-a : 3,4-a1] - diquinolin - 15 -ium salts of formula <FORM:1011311/C2/1> where R and R1 are hydrogen or methyl and X is a physiologically acceptable anion are prepared by condensing a quinoline compound of formula <FORM:1011311/C2/2> with a quinaldine of formula <FORM:1011311/C2/3> where R and R1 are as above, in the presence of an inert organic solvent containing iodine. The resulting iodide may be converted to any desired salt by treating an aqueous or aqueous alcoholic solution of the iode with a strong base ion exchange resin in the hydroxyl form (e.g. that sold under the Trade Mark Amberlite IRA-410) and treating the hydroxide directly with the acid. Alternatively, the acetate salt is formed from the hydroxide and the desired salt formed by metathesis using the sodium or potassium salt of an acid having the desired anion. Specified anions are the chloride, bromide, iodide, nitrate, bisulphite, hemisulphate, perchlorate, acetate, palmitate, stearate, hemipamoate, picrate, 1-decanesulphonate, 4-chloro - 2 - (5 - chlorosalicyl) phenoxide, 3-hydroxy - 2 - naphthoate, dodecylsulphate, cyclohexanesulphamate, 2,4,5 - trichlorophenoxide, 2,21 - thiobis - (4,6 - dichlorophenoxide), deoxycholate, 7 - chloro - 4 - hydroxy - 3 - quinolinecarboxylate 2,6 - dihydroxyisonicotinate, 1 - bromo - 2 - naphthoxide, hemiadipate, p-toluenesulphonate, hemi - (5,51 - thiodisalicylate), 3,5 - dichlorosalicylate, taurocholate, dioctylsulphosuccinate, 2,6 - di - iodo - 4 - nitrophenoxide, 1 - hexanesulphonate, 4 - chlorobenzenesulphonate, decanoate and phenolphthaleinate.ALSO:An anthelmintic composition also having antibacterial, antiamebic and antitrichomonal activity, in dosage unit form, comprises, as active ingredient, imidazo [1, 2-a : 3, 4-a1] diquinolin-15-ium salt having the formula <FORM:1011311/A5-A6/1> wherein R and R1 each independently represent hydrogen or methyl and X is a physiologically acceptable anion. Specified anions are the chloride, bromide, iodide, nitrate, bisulphite, hemisulphate, perchlorate, acetate, palmitate, stearate, hemipamoate, picrate, 1-decanesulphonate, 4-chloro-2-(5-chlorosalicyl) phenoxide, 3-hydroxy, 2-naphthoate, dodecylsulphate, cyclohexanesulphamate, 2, 4, 5-trichloro-phenoxide, 2, 21-thiobis (4, 6-dichlorophenoxide), deoxycholate, 7-chloro-4-hydroxy -3-quinolinecarboxlate, 2, 6-dihydroxyisonicotinate, 1-bromo-2-naphthoxide, hemiadipate, p-toluenesulphonate, hemi-(5, 51-thiodisalicylate), 3, 5-dichlorosalicylate, taurocholate, dioctylsulphosuccinate, 2, 6-di-iodo-4-nitrophenoxide, 1-hexanesulphonate, H-chlorobenzene sulphonate, decanoate and phenolphthaleinate. The composition may be used orally e.g. in the form of an aqueous suspension or solution containing suspending agents or solubilizers, preservatives and flavouring agents; or in the form of tablets or capsules in which the active ingredient is dissolved in a vegetable oil. The active ingredient may be dissolved in water containing sorbitan monostearate and polyethylene glycol. In the case of animals, the active material may be mixed with the animal feed.
GB26608/63A 1963-07-04 1963-07-04 Antiparasitic compositions and use thereof Expired GB1011311A (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
GB26608/63A GB1011311A (en) 1963-07-04 1963-07-04 Antiparasitic compositions and use thereof
US375638A US3253986A (en) 1963-07-04 1964-06-16 Antiparasitic compositions and use thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB26608/63A GB1011311A (en) 1963-07-04 1963-07-04 Antiparasitic compositions and use thereof

Publications (1)

Publication Number Publication Date
GB1011311A true GB1011311A (en) 1965-11-24

Family

ID=10246299

Family Applications (1)

Application Number Title Priority Date Filing Date
GB26608/63A Expired GB1011311A (en) 1963-07-04 1963-07-04 Antiparasitic compositions and use thereof

Country Status (2)

Country Link
US (1) US3253986A (en)
GB (1) GB1011311A (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB988483A (en) * 1963-02-11 1965-04-07 Soc D Etudes Prod Chimique Quinoline derivative and preparation thereof
US3541100A (en) * 1967-12-14 1970-11-17 American Cyanamid Co Benzheteroazolo(2,3-a)isoquinolium salts
GB1278272A (en) * 1969-02-19 1972-06-21 Pfizer Ltd Substituted hexahydro-imidazoquinolines
US4207320A (en) * 1978-08-28 1980-06-10 Warner-Lambert Company Amino-substituted imidazo[1,2-a:3,4-a']diquinolin-15-ium salts compositions and method of use
CA2644613A1 (en) * 2006-03-07 2007-09-13 Endacea, Inc. Compositions and methods for treating respiratory disorders
JP5558875B2 (en) * 2009-03-19 2014-07-23 日本曹達株式会社 Novel inclusion complex, epoxy resin composition and epoxy resin composition for semiconductor encapsulation

Also Published As

Publication number Publication date
US3253986A (en) 1966-05-31

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