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GB0215775D0 - Pharmaceutical compounds - Google Patents

Pharmaceutical compounds

Info

Publication number
GB0215775D0
GB0215775D0 GB0215775A GB0215775A GB0215775D0 GB 0215775 D0 GB0215775 D0 GB 0215775D0 GB 0215775 A GB0215775 A GB 0215775A GB 0215775 A GB0215775 A GB 0215775A GB 0215775 D0 GB0215775 D0 GB 0215775D0
Authority
GB
United Kingdom
Prior art keywords
pharmaceutical compounds
pharmaceutical
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GB0215775A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astex Technology Ltd
Original Assignee
Astex Technology Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astex Technology Ltd filed Critical Astex Technology Ltd
Priority to GB0215775A priority Critical patent/GB0215775D0/en
Publication of GB0215775D0 publication Critical patent/GB0215775D0/en
Priority to PCT/GB2003/002905 priority patent/WO2004004730A2/fr
Priority to AU2003242860A priority patent/AU2003242860A1/en
Ceased legal-status Critical Current

Links

GB0215775A 2002-07-06 2002-07-06 Pharmaceutical compounds Ceased GB0215775D0 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
GB0215775A GB0215775D0 (en) 2002-07-06 2002-07-06 Pharmaceutical compounds
PCT/GB2003/002905 WO2004004730A2 (fr) 2002-07-06 2003-07-04 Composes pharmaceutiques
AU2003242860A AU2003242860A1 (en) 2002-07-06 2003-07-04 2-aminopyrazine derivatives as inhibitors of cyclin dependent kinases for the treatment of proliferative disorders

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB0215775A GB0215775D0 (en) 2002-07-06 2002-07-06 Pharmaceutical compounds

Publications (1)

Publication Number Publication Date
GB0215775D0 true GB0215775D0 (en) 2002-08-14

Family

ID=9940040

Family Applications (1)

Application Number Title Priority Date Filing Date
GB0215775A Ceased GB0215775D0 (en) 2002-07-06 2002-07-06 Pharmaceutical compounds

Country Status (3)

Country Link
AU (1) AU2003242860A1 (fr)
GB (1) GB0215775D0 (fr)
WO (1) WO2004004730A2 (fr)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2486187C (fr) 2002-05-23 2013-02-19 Cytopia Pty Ltd. Inhibiteurs de la kinase
WO2005058876A1 (fr) * 2003-12-16 2005-06-30 Gpc Biotech Ag Derives de la pyrazine utilises en tant que composes efficaces contre les maladies infectieuses
AU2005230847B2 (en) * 2004-03-31 2012-11-08 Exelixis, Inc. Anaplastic lymphoma kinase modulators and methods of use
ATE458730T1 (de) 2004-04-13 2010-03-15 Icagen Inc Polycyclische pyrazine als kaliumionenkanal- modulatoren
WO2006044826A2 (fr) * 2004-10-20 2006-04-27 Compass Pharmaceuticals Llc Compositions et leur utilisation en tant qu'agents antitumoraux
GB0719644D0 (en) * 2007-10-05 2007-11-14 Cancer Rec Tech Ltd Therapeutic compounds and their use
DE102008022788A1 (de) * 2008-05-08 2009-11-12 Süd-Chemie AG 2,6-Pyrazinverbrückte Carbenkomplexe
EP2417123A2 (fr) * 2009-04-06 2012-02-15 Agios Pharmaceuticals, Inc. Compositions thérapeutiques et procédés d'utilisation associés
DK2427441T3 (en) 2009-05-04 2017-03-20 Agios Pharmaceuticals Inc PKM2 Activators for use in the treatment of cancer
CA2944788C (fr) 2009-06-29 2023-08-22 Agios Pharmaceuticals, Inc. Composes, et compositions associees, qui modulent la pyruvate kinase m2, et methodes de fabrication associees
EP2448581B1 (fr) 2009-06-29 2016-12-07 Agios Pharmaceuticals, Inc. Compositions thérapeutiques et procédés d'utilisation associés
JP5837091B2 (ja) 2010-12-17 2015-12-24 アジオス ファーマシューティカルズ, インコーポレイテッド ピルビン酸キナーゼm2(pkm2)調節剤としての新規n−(4−(アゼチジン−1−カルボニル)フェニル)−(ヘテロ−)アリールスルホンアミド誘導体
JP6092118B2 (ja) 2010-12-21 2017-03-08 アジオス ファーマシューティカルズ, インコーポレイテッド ニ環式pkm2活性化剤
TWI549947B (zh) 2010-12-29 2016-09-21 阿吉歐斯製藥公司 治療化合物及組成物
KR101873543B1 (ko) 2011-05-03 2018-07-02 아지오스 파마슈티컬스 아이엔씨. 치료에 사용하기 위한 피루베이트 키나아제 활성제
WO2012151440A1 (fr) 2011-05-03 2012-11-08 Agios Pharmaceuticals, Inc. Procédés d'utilisation d'activateurs de pyruvate kinase
ES2634014T3 (es) 2013-01-30 2017-09-26 Bayer Pharma Aktiengesellschaft Isotiazoles sustituidos con amino
WO2014139144A1 (fr) 2013-03-15 2014-09-18 Agios Pharmaceuticals, Inc. Composés et compositions thérapeutiques
CN105985322A (zh) * 2015-03-03 2016-10-05 苏州翔实医药发展有限公司 氨基吡嗪化合物及其用途
DK3307271T3 (da) 2015-06-11 2023-10-09 Agios Pharmaceuticals Inc Fremgangsmåder til anvendelse af pyruvatkinase-aktivatorer
CN112142716B (zh) * 2020-10-29 2021-08-31 山东新时代药业有限公司 一种5元杂芳基取代的吡嗪衍生物及其应用
WO2024050374A2 (fr) * 2022-09-02 2024-03-07 Miralogx Llc Composés anti-inflammatoires, compositions pharmaceutiques et méthodes de traitement de l'hémochromatose et d'autres troubles

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0254259A3 (fr) * 1986-07-21 1989-11-23 Otsuka Pharmaceutical Factory, Inc. Dérivés de p-aminophénols
GR900100380A (el) * 1989-05-20 1991-10-10 Fisons Plc Μέ?οδος παρασκευής αντι-φλεγμονωδών παραγώγων αμινοφενόλης.
US6506747B1 (en) * 1998-06-05 2003-01-14 Boehringer Ingelheim Pharmaceuticals, Inc. Substituted 1-(4-aminophenyl)pyrazoles and their use as anti-inflammatory agents
SE9903894D0 (sv) * 1999-10-28 1999-10-28 New Pharma Research Ab Novel compounds
SE9904108D0 (sv) * 1999-11-15 1999-11-15 New Pharma Research Ab Nya föreningar
PT1330452E (pt) * 2000-09-20 2009-01-22 Ortho Mcneil Pharm Inc Derivados de pirazina como moduladores de tirosina-cinases
PL361690A1 (en) * 2000-11-20 2004-10-04 Biovitrum Ab Piperazinylpyrazine compounds as agonist or antagonist of serotonin 5ht-2 receptor
WO2002060492A1 (fr) * 2001-01-30 2002-08-08 Cytopia Pty Ltd Procedes d'inhibition de kinases
AU2002342051B2 (en) * 2001-10-12 2009-06-11 Irm Llc Kinase inhibitor scaffolds and methods for their preparation
GB0124939D0 (en) * 2001-10-17 2001-12-05 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
AU2003242860A1 (en) 2004-01-23
WO2004004730A2 (fr) 2004-01-15
AU2003242860A8 (en) 2004-01-23
WO2004004730A3 (fr) 2004-04-29

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Legal Events

Date Code Title Description
AT Applications terminated before publication under section 16(1)