[go: up one dir, main page]

FR2896690B1 - Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique - Google Patents

Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique

Info

Publication number
FR2896690B1
FR2896690B1 FR0600811A FR0600811A FR2896690B1 FR 2896690 B1 FR2896690 B1 FR 2896690B1 FR 0600811 A FR0600811 A FR 0600811A FR 0600811 A FR0600811 A FR 0600811A FR 2896690 B1 FR2896690 B1 FR 2896690B1
Authority
FR
France
Prior art keywords
mequitazine
enantiomer
preparation
medicinal product
limiting
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0600811A
Other languages
English (en)
Other versions
FR2896690A1 (fr
Inventor
Alain Latil
Versailles Jacky Tisne
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre Medicament SA
Original Assignee
Pierre Fabre Medicament SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pierre Fabre Medicament SA filed Critical Pierre Fabre Medicament SA
Priority to FR0600811A priority Critical patent/FR2896690B1/fr
Priority to PCT/EP2007/050828 priority patent/WO2007085652A1/fr
Publication of FR2896690A1 publication Critical patent/FR2896690A1/fr
Application granted granted Critical
Publication of FR2896690B1 publication Critical patent/FR2896690B1/fr
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR0600811A 2006-01-30 2006-01-30 Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique Expired - Fee Related FR2896690B1 (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
FR0600811A FR2896690B1 (fr) 2006-01-30 2006-01-30 Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique
PCT/EP2007/050828 WO2007085652A1 (fr) 2006-01-30 2007-01-29 Utilisation de l'enantiomere (s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0600811A FR2896690B1 (fr) 2006-01-30 2006-01-30 Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique

Publications (2)

Publication Number Publication Date
FR2896690A1 FR2896690A1 (fr) 2007-08-03
FR2896690B1 true FR2896690B1 (fr) 2008-05-02

Family

ID=37027771

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0600811A Expired - Fee Related FR2896690B1 (fr) 2006-01-30 2006-01-30 Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique

Country Status (2)

Country Link
FR (1) FR2896690B1 (fr)
WO (1) WO2007085652A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2916142A1 (fr) * 2007-05-15 2008-11-21 Pierre Fabre Medicament Sa Forme pharmaceutique comprenant du (10-[(3s)-1-azabicyclo [2.2.2]oct-3-ylmethyl]-10h-phenothiazine se presentant sous une forme appropriee pour l'administration d'unde dose journaliere comprise entre 1 et 3 mg
FR2924344B1 (fr) * 2007-12-04 2010-04-16 Pf Medicament Utilisation de la mequitazine sous la forme de racemate ou d'enantiomeres pour la preparation d'un medicament destine au traitement ou a la prevention de pathologies impliquant les recepteurs histaminiques h4.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2522660A1 (fr) * 1982-03-05 1983-09-09 Pharmuka Lab Isomere levogyre de la mequitazine, son procede de preparation et medicaments le contenant
FR2772029B1 (fr) * 1997-12-08 2000-02-25 Pf Medicament Procede de preparation de la mequitazine et nouvel intermediaire de synthese

Also Published As

Publication number Publication date
WO2007085652A1 (fr) 2007-08-02
FR2896690A1 (fr) 2007-08-03

Similar Documents

Publication Publication Date Title
EP1909772A4 (fr) Formulation pour l'administration transdermique de medicaments
EP1789075A4 (fr) Substances ameliorant l'absorption destinees a l'administration de medicaments
EP1971372A4 (fr) Compositions de supports a noyau hydrophobe pour l'administration d'agents therapeutiques, et procedes de preparation et d'utilisation
EP2152195A4 (fr) Peptide pharmaceutique pour administration orale
ZA200704163B (en) Oral medicament for the modified release of at least one active principle, in a multimicrocapsule form
BRPI0810646A2 (pt) " compostos farmacêuticos ".
IL198301A (en) Aryl amides are stored in thiazole and oxazole, a pharmaceutical preparation containing them and their use in the preparation of drugs
EP2164322A4 (fr) Composition agrochimique et procédé de préparation et d'utilisation de celle-ci
EP2520305A4 (fr) Composition médicinale comprenant un extrait de `, procédé de préparation et d'utilisation de celle-ci
FR2959416B1 (fr) Utilisation d'anticorps anti-cd71 pour la preparation d'un medicament
ECSP045493A (es) Nuevas composiciones farmacéuticas que contienen flibanserina polimorfo a
DE502007005902D1 (de) -methyl-19-nor-20- spirox-4-en-3-one), sowie diese enthaltende pharmazeutische präparate
TWI366457B (en) Use of a beta2-adrenoceptor agonist for the preparation of a dermatological medicament
EP2292242A4 (fr) Dérivé de scutellarine, procédé d'élaboration, composition pharmaceutique, et utilisation correspondante
FR2930150B1 (fr) Utilisation de la dronedarone pour la preparation d'un medicament destine a reguler le taux de potassium dans le sang
EP2147922A4 (fr) Dérivé hétérocyclique condensé, composition pharmaceutique comprenant le dérivé et utilisation de la composition pour des objectifs médicaux
FR2898272B1 (fr) Utilisation de derives du 3,5-seco-4-nor-cholestrane pour l'obtention d'un medicament cytoprotecteur
FR2896690B1 (fr) Utilisation de l'enantiomere(s) de la mequitazine pour la preparation d'un medicament, tout en limitant la toxicite genomique
FR2920776B1 (fr) Utilisation de derives de purine pour la fabrication d'un medicament
FR2924019B1 (fr) Dispositif de preparation d'un produit pharmaceutique ou medicamenteux injectable
ZA201005398B (en) 15,16-methylene-17-(1'-propenyl)-17,3'-oxidoestra-4-en-3-one derivative,use thereof,and medicament containing said derivative
IL205975A (en) Pharmaceutical preparation suitable for rectal administration, disposable packaging and a method for increasing its stability
FR2909879B1 (fr) Utilisation d'un heptapeptide a activite anxiolytique pour la preparation de medicaments et de complements alimentaires
FR2924345B1 (fr) Utilisation de la mequitazine sous la forme de racemate ou d'enantiomeres pour la preparation d'un medicament destine au traitement ou a la prevention de pathologies impliquant les recepteurs histaminiques h4.
FR2904318B1 (fr) Derives de pyrimidinone et leur utilisation comme medicament

Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20150930