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FR2789078B3 - PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents

PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Info

Publication number
FR2789078B3
FR2789078B3 FR9901201A FR9901201A FR2789078B3 FR 2789078 B3 FR2789078 B3 FR 2789078B3 FR 9901201 A FR9901201 A FR 9901201A FR 9901201 A FR9901201 A FR 9901201A FR 2789078 B3 FR2789078 B3 FR 2789078B3
Authority
FR
France
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
acid derivatives
pyrazolecarboxylic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
FR9901201A
Other languages
French (fr)
Other versions
FR2789078A1 (en
Inventor
Francis Barth
Frederic Larguier
Murielle Rinaldi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi SA
Original Assignee
Sanofi SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi SA filed Critical Sanofi SA
Priority to FR9901201A priority Critical patent/FR2789078B3/en
Priority to FR9910166A priority patent/FR2789079B3/en
Priority to DK00901661T priority patent/DK1150961T3/en
Priority to US09/890,242 priority patent/US6432984B1/en
Priority to KR10-2001-7009572A priority patent/KR100425405B1/en
Priority to CZ20012697A priority patent/CZ297667B6/en
Priority to EP00901661A priority patent/EP1150961B1/en
Priority to CNB008054681A priority patent/CN1146544C/en
Priority to UA2001074905A priority patent/UA66900C2/en
Priority to RU2001121186/04A priority patent/RU2216542C2/en
Priority to AT00901661T priority patent/ATE252562T1/en
Priority to IL14419800A priority patent/IL144198A0/en
Priority to ES00901661T priority patent/ES2208267T3/en
Priority to SI200030284T priority patent/SI1150961T1/en
Priority to IDW00200101603A priority patent/ID29534A/en
Priority to HR20010564A priority patent/HRP20010564B1/en
Priority to HK02100712.5A priority patent/HK1039329B/en
Priority to NZ512886A priority patent/NZ512886A/en
Priority to YUP-539/01A priority patent/RS50209B/en
Priority to EEP200100399A priority patent/EE04343B1/en
Priority to AU22989/00A priority patent/AU754771B2/en
Priority to BR0007895-6A priority patent/BR0007895A/en
Priority to PL350030A priority patent/PL198422B1/en
Priority to MEP-2008-114A priority patent/ME00052B/en
Priority to PT00901661T priority patent/PT1150961E/en
Priority to JP2000597279A priority patent/JP3794925B2/en
Priority to HU0201278A priority patent/HUP0201278A3/en
Priority to ARP000100386A priority patent/AR020558A1/en
Priority to CA002358885A priority patent/CA2358885C/en
Priority to TR2001/02054T priority patent/TR200102054T2/en
Priority to PCT/FR2000/000194 priority patent/WO2000046209A1/en
Priority to SK1087-2001A priority patent/SK284203B6/en
Priority to PE2000000066A priority patent/PE20001493A1/en
Priority to DE60006070T priority patent/DE60006070T2/en
Priority to MEP-114/08A priority patent/MEP11408A/en
Priority to CO00005429A priority patent/CO5160257A1/en
Priority to TW089101649A priority patent/TW581764B/en
Publication of FR2789078A1 publication Critical patent/FR2789078A1/en
Application granted granted Critical
Publication of FR2789078B3 publication Critical patent/FR2789078B3/en
Priority to IL144198A priority patent/IL144198A/en
Priority to ZA200105739A priority patent/ZA200105739B/en
Priority to IS6002A priority patent/IS2448B/en
Priority to BG105749A priority patent/BG65193B1/en
Priority to NO20013736A priority patent/NO319824B1/en
Priority to US10/165,140 priority patent/US6645985B2/en
Priority to US10/455,220 priority patent/US20040039024A1/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/72Hydrazones
    • C07C251/74Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C251/78Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
    • C07C251/80Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton the carbon skeleton containing rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9901201A 1999-02-01 1999-02-01 PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Expired - Lifetime FR2789078B3 (en)

Priority Applications (44)

Application Number Priority Date Filing Date Title
FR9901201A FR2789078B3 (en) 1999-02-01 1999-02-01 PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FR9910166A FR2789079B3 (en) 1999-02-01 1999-08-02 PYRAZOLECARBOXYLIC ACID DERIVATIVE, ITS PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
DK00901661T DK1150961T3 (en) 1999-02-01 2000-01-28 Pyrazole carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
US09/890,242 US6432984B1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
KR10-2001-7009572A KR100425405B1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic Acid Derivatives, Their Preparation, Pharmaceutical Compositions Containing Them
CZ20012697A CZ297667B6 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivative process for its preparation and pharmaceutical preparations in which the derivative is comprised
EP00901661A EP1150961B1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
CNB008054681A CN1146544C (en) 1999-02-01 2000-01-28 Pyrazoelcarboxylic acid derivatives, their preparation, pharmaceutical compositions containing
UA2001074905A UA66900C2 (en) 1999-02-01 2000-01-28 Pyrazole carbonic acid derivatives, a method for the preparation thereof, a pharmaceutical composition containing them
RU2001121186/04A RU2216542C2 (en) 1999-02-01 2000-01-28 Derivatives of pyrazole carboxylic acid, their preparing, pharmaceutical composition containing thereof
AT00901661T ATE252562T1 (en) 1999-02-01 2000-01-28 PYRAZOLECARBONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
IL14419800A IL144198A0 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
ES00901661T ES2208267T3 (en) 1999-02-01 2000-01-28 NEVUO DERIVED FROM PIRAZOL, ITS SALTS AND SOLVATES, PROCEDURE FOR THE PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
SI200030284T SI1150961T1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
IDW00200101603A ID29534A (en) 1999-02-01 2000-01-28 PIRAZOLKARBOKSILAT ACID DERIVES, THEIR PRODUCTION, THE PHARMACY COMPOSITION THAT CONTAINS IT
HR20010564A HRP20010564B1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
HK02100712.5A HK1039329B (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
NZ512886A NZ512886A (en) 1999-02-01 2000-01-28 N-Piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxamide
YUP-539/01A RS50209B (en) 1999-02-01 2000-01-28 PYRAZOLOCARBOXYLIC ACIDS, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS WITH THE CONTENT OF THE SAME
EEP200100399A EE04343B1 (en) 1999-02-01 2000-01-28 Pyrazole carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
AU22989/00A AU754771B2 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
BR0007895-6A BR0007895A (en) 1999-02-01 2000-01-28 Pyrazolcarboxylic acid derivatives, their preparation and pharmaceutical compositions
PL350030A PL198422B1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
MEP-2008-114A ME00052B (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
PT00901661T PT1150961E (en) 1999-02-01 2000-01-28 PIRAZOLECARBOXYLIC ACID DERIVATIVES PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM
JP2000597279A JP3794925B2 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their production, pharmaceutical compositions containing them
HU0201278A HUP0201278A3 (en) 1999-02-01 2000-01-28 Pyrazolecarboamide derivative, its preparation, pharmaceutical compositions containing it and its intermediates
ARP000100386A AR020558A1 (en) 1999-02-01 2000-01-28 A PIRAZOLCARBOXILICO ACID DERIVATIVE, ITS USE, A PROCEDURE FOR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING IT AND USEFUL COMPOUNDS AS INTERMEDIARIES TO PREPARE IT
CA002358885A CA2358885C (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
TR2001/02054T TR200102054T2 (en) 1999-02-01 2000-01-28 Pyrazolcarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them.
PCT/FR2000/000194 WO2000046209A1 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
SK1087-2001A SK284203B6 (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
PE2000000066A PE20001493A1 (en) 1999-02-01 2000-01-28 DERIVATIVES OF PIRAZOLCARBOXILICO ACID, A PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM
DE60006070T DE60006070T2 (en) 1999-02-01 2000-01-28 PYRAZOL CARBOXYLIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEREOF
MEP-114/08A MEP11408A (en) 1999-02-01 2000-01-28 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing same
CO00005429A CO5160257A1 (en) 1999-02-01 2000-01-31 N-PIPERIDINO-5- (4-BROMOFENIL) -1- (2,4-DICLOROPHENIL) -4-ETILPIRAZOL-3-CARBOXAMIDE, ITS SALTS, ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT
TW089101649A TW581764B (en) 1999-02-01 2000-01-31 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
IL144198A IL144198A (en) 1999-02-01 2001-07-08 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
ZA200105739A ZA200105739B (en) 1999-02-01 2001-07-12 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them.
IS6002A IS2448B (en) 1999-02-01 2001-07-13 Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them
BG105749A BG65193B1 (en) 1999-02-01 2001-07-27 Pyrazolecarboxylic acid derivative, preparation thereof and pharmaceutical compositions containing it
NO20013736A NO319824B1 (en) 1999-02-01 2001-07-30 Pyrazole carboxylic acid derivatives, their preparation and use and pharmaceutical compositions containing the same, as well as intermediate compounds.
US10/165,140 US6645985B2 (en) 1999-02-01 2002-06-07 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them, and method of treating
US10/455,220 US20040039024A1 (en) 1999-02-01 2003-06-05 Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9901201A FR2789078B3 (en) 1999-02-01 1999-02-01 PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Publications (2)

Publication Number Publication Date
FR2789078A1 FR2789078A1 (en) 2000-08-04
FR2789078B3 true FR2789078B3 (en) 2001-03-02

Family

ID=9541521

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9901201A Expired - Lifetime FR2789078B3 (en) 1999-02-01 1999-02-01 PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Country Status (2)

Country Link
FR (1) FR2789078B3 (en)
ZA (1) ZA200105739B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005533748A (en) 2002-03-08 2005-11-10 シグナル ファーマシューティカルズ,インコーポレイテッド Combination therapies to treat, prevent, or manage proliferative disorders and cancer
BR0313041A (en) * 2002-07-29 2005-06-21 Hoffmann La Roche Compounds; pharmaceutical compositions; method for the treatment and / or prophylaxis of diseases that are associated with cb1 receptor modulation; and use of compounds

Also Published As

Publication number Publication date
FR2789078A1 (en) 2000-08-04
ZA200105739B (en) 2002-01-24

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