FR2789078B3 - PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents
PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEMInfo
- Publication number
- FR2789078B3 FR2789078B3 FR9901201A FR9901201A FR2789078B3 FR 2789078 B3 FR2789078 B3 FR 2789078B3 FR 9901201 A FR9901201 A FR 9901201A FR 9901201 A FR9901201 A FR 9901201A FR 2789078 B3 FR2789078 B3 FR 2789078B3
- Authority
- FR
- France
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- acid derivatives
- pyrazolecarboxylic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- KOPFEFZSAMLEHK-UHFFFAOYSA-N 1h-pyrazole-5-carboxylic acid Chemical class OC(=O)C=1C=CNN=1 KOPFEFZSAMLEHK-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/72—Hydrazones
- C07C251/74—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C251/78—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
- C07C251/80—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton the carbon skeleton containing rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (44)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9901201A FR2789078B3 (en) | 1999-02-01 | 1999-02-01 | PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| FR9910166A FR2789079B3 (en) | 1999-02-01 | 1999-08-02 | PYRAZOLECARBOXYLIC ACID DERIVATIVE, ITS PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
| DK00901661T DK1150961T3 (en) | 1999-02-01 | 2000-01-28 | Pyrazole carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them |
| US09/890,242 US6432984B1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| KR10-2001-7009572A KR100425405B1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic Acid Derivatives, Their Preparation, Pharmaceutical Compositions Containing Them |
| CZ20012697A CZ297667B6 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivative process for its preparation and pharmaceutical preparations in which the derivative is comprised |
| EP00901661A EP1150961B1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| CNB008054681A CN1146544C (en) | 1999-02-01 | 2000-01-28 | Pyrazoelcarboxylic acid derivatives, their preparation, pharmaceutical compositions containing |
| UA2001074905A UA66900C2 (en) | 1999-02-01 | 2000-01-28 | Pyrazole carbonic acid derivatives, a method for the preparation thereof, a pharmaceutical composition containing them |
| RU2001121186/04A RU2216542C2 (en) | 1999-02-01 | 2000-01-28 | Derivatives of pyrazole carboxylic acid, their preparing, pharmaceutical composition containing thereof |
| AT00901661T ATE252562T1 (en) | 1999-02-01 | 2000-01-28 | PYRAZOLECARBONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
| IL14419800A IL144198A0 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| ES00901661T ES2208267T3 (en) | 1999-02-01 | 2000-01-28 | NEVUO DERIVED FROM PIRAZOL, ITS SALTS AND SOLVATES, PROCEDURE FOR THE PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. |
| SI200030284T SI1150961T1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| IDW00200101603A ID29534A (en) | 1999-02-01 | 2000-01-28 | PIRAZOLKARBOKSILAT ACID DERIVES, THEIR PRODUCTION, THE PHARMACY COMPOSITION THAT CONTAINS IT |
| HR20010564A HRP20010564B1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| HK02100712.5A HK1039329B (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| NZ512886A NZ512886A (en) | 1999-02-01 | 2000-01-28 | N-Piperidino-5-(4-bromophenyl)-1-(2,4-dichlorophenyl)-4-ethylpyrazole-3-carboxamide |
| YUP-539/01A RS50209B (en) | 1999-02-01 | 2000-01-28 | PYRAZOLOCARBOXYLIC ACIDS, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS WITH THE CONTENT OF THE SAME |
| EEP200100399A EE04343B1 (en) | 1999-02-01 | 2000-01-28 | Pyrazole carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them |
| AU22989/00A AU754771B2 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| BR0007895-6A BR0007895A (en) | 1999-02-01 | 2000-01-28 | Pyrazolcarboxylic acid derivatives, their preparation and pharmaceutical compositions |
| PL350030A PL198422B1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| MEP-2008-114A ME00052B (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| PT00901661T PT1150961E (en) | 1999-02-01 | 2000-01-28 | PIRAZOLECARBOXYLIC ACID DERIVATIVES PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM |
| JP2000597279A JP3794925B2 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their production, pharmaceutical compositions containing them |
| HU0201278A HUP0201278A3 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboamide derivative, its preparation, pharmaceutical compositions containing it and its intermediates |
| ARP000100386A AR020558A1 (en) | 1999-02-01 | 2000-01-28 | A PIRAZOLCARBOXILICO ACID DERIVATIVE, ITS USE, A PROCEDURE FOR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING IT AND USEFUL COMPOUNDS AS INTERMEDIARIES TO PREPARE IT |
| CA002358885A CA2358885C (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| TR2001/02054T TR200102054T2 (en) | 1999-02-01 | 2000-01-28 | Pyrazolcarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them. |
| PCT/FR2000/000194 WO2000046209A1 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| SK1087-2001A SK284203B6 (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| PE2000000066A PE20001493A1 (en) | 1999-02-01 | 2000-01-28 | DERIVATIVES OF PIRAZOLCARBOXILICO ACID, A PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM |
| DE60006070T DE60006070T2 (en) | 1999-02-01 | 2000-01-28 | PYRAZOL CARBOXYLIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEREOF |
| MEP-114/08A MEP11408A (en) | 1999-02-01 | 2000-01-28 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing same |
| CO00005429A CO5160257A1 (en) | 1999-02-01 | 2000-01-31 | N-PIPERIDINO-5- (4-BROMOFENIL) -1- (2,4-DICLOROPHENIL) -4-ETILPIRAZOL-3-CARBOXAMIDE, ITS SALTS, ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT |
| TW089101649A TW581764B (en) | 1999-02-01 | 2000-01-31 | Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them |
| IL144198A IL144198A (en) | 1999-02-01 | 2001-07-08 | Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them |
| ZA200105739A ZA200105739B (en) | 1999-02-01 | 2001-07-12 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them. |
| IS6002A IS2448B (en) | 1999-02-01 | 2001-07-13 | Pyrazolecarboxylic acid derivatives, their preparation, pharmaceutical compositions containing them |
| BG105749A BG65193B1 (en) | 1999-02-01 | 2001-07-27 | Pyrazolecarboxylic acid derivative, preparation thereof and pharmaceutical compositions containing it |
| NO20013736A NO319824B1 (en) | 1999-02-01 | 2001-07-30 | Pyrazole carboxylic acid derivatives, their preparation and use and pharmaceutical compositions containing the same, as well as intermediate compounds. |
| US10/165,140 US6645985B2 (en) | 1999-02-01 | 2002-06-07 | Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them, and method of treating |
| US10/455,220 US20040039024A1 (en) | 1999-02-01 | 2003-06-05 | Pyrazolecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9901201A FR2789078B3 (en) | 1999-02-01 | 1999-02-01 | PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2789078A1 FR2789078A1 (en) | 2000-08-04 |
| FR2789078B3 true FR2789078B3 (en) | 2001-03-02 |
Family
ID=9541521
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR9901201A Expired - Lifetime FR2789078B3 (en) | 1999-02-01 | 1999-02-01 | PYRAZOLECARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Country Status (2)
| Country | Link |
|---|---|
| FR (1) | FR2789078B3 (en) |
| ZA (1) | ZA200105739B (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005533748A (en) | 2002-03-08 | 2005-11-10 | シグナル ファーマシューティカルズ,インコーポレイテッド | Combination therapies to treat, prevent, or manage proliferative disorders and cancer |
| BR0313041A (en) * | 2002-07-29 | 2005-06-21 | Hoffmann La Roche | Compounds; pharmaceutical compositions; method for the treatment and / or prophylaxis of diseases that are associated with cb1 receptor modulation; and use of compounds |
-
1999
- 1999-02-01 FR FR9901201A patent/FR2789078B3/en not_active Expired - Lifetime
-
2001
- 2001-07-12 ZA ZA200105739A patent/ZA200105739B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2789078A1 (en) | 2000-08-04 |
| ZA200105739B (en) | 2002-01-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TP | Transmission of property | ||
| CD | Change of name or company name |