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FR2761073B1 - PYRAZINO [1,2-A] INDOLE-1-ONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION - Google Patents

PYRAZINO [1,2-A] INDOLE-1-ONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Info

Publication number
FR2761073B1
FR2761073B1 FR9703390A FR9703390A FR2761073B1 FR 2761073 B1 FR2761073 B1 FR 2761073B1 FR 9703390 A FR9703390 A FR 9703390A FR 9703390 A FR9703390 A FR 9703390A FR 2761073 B1 FR2761073 B1 FR 2761073B1
Authority
FR
France
Prior art keywords
pyrazino
indole
derivatives
preparation
therapeutic application
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9703390A
Other languages
French (fr)
Other versions
FR2761073A1 (en
Inventor
Gary Mccort
Christian Hoornaert
Olivier Duclos
Eric Guilpain
Caroline Cadilhac
Genevieve Dellac
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR9703390A priority Critical patent/FR2761073B1/en
Publication of FR2761073A1 publication Critical patent/FR2761073A1/en
Application granted granted Critical
Publication of FR2761073B1 publication Critical patent/FR2761073B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9703390A 1997-03-20 1997-03-20 PYRAZINO [1,2-A] INDOLE-1-ONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION Expired - Fee Related FR2761073B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR9703390A FR2761073B1 (en) 1997-03-20 1997-03-20 PYRAZINO [1,2-A] INDOLE-1-ONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9703390A FR2761073B1 (en) 1997-03-20 1997-03-20 PYRAZINO [1,2-A] INDOLE-1-ONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Publications (2)

Publication Number Publication Date
FR2761073A1 FR2761073A1 (en) 1998-09-25
FR2761073B1 true FR2761073B1 (en) 1999-04-23

Family

ID=9505002

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9703390A Expired - Fee Related FR2761073B1 (en) 1997-03-20 1997-03-20 PYRAZINO [1,2-A] INDOLE-1-ONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION

Country Status (1)

Country Link
FR (1) FR2761073B1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104203950B (en) 2012-03-16 2016-08-24 生命医药公司 Liver X receptor modulators
HUE029402T2 (en) 2012-03-16 2017-02-28 Vitae Pharmaceuticals Inc Liver x receptor modulators
JP6757312B2 (en) * 2014-03-27 2020-09-16 ヴァンダービルト ユニバーシティー Substituted indole MCL-1 inhibitor

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2027898A6 (en) * 1991-01-24 1992-06-16 Espanola Prod Quimicos 2-Methoxyphenylpiperazine derivatives.
EP0572863A1 (en) * 1992-06-05 1993-12-08 F. Hoffmann-La Roche Ag CNS pyrazinoindoles

Also Published As

Publication number Publication date
FR2761073A1 (en) 1998-09-25

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Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse

Effective date: 20051130