[go: up one dir, main page]

FR2747678B1 - Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique - Google Patents

Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique

Info

Publication number
FR2747678B1
FR2747678B1 FR9605002A FR9605002A FR2747678B1 FR 2747678 B1 FR2747678 B1 FR 2747678B1 FR 9605002 A FR9605002 A FR 9605002A FR 9605002 A FR9605002 A FR 9605002A FR 2747678 B1 FR2747678 B1 FR 2747678B1
Authority
FR
France
Prior art keywords
imidazobenzoxazine
processes
preparation
therapeutic uses
compounds derived
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9605002A
Other languages
English (en)
Other versions
FR2747678A1 (fr
Inventor
Luc Even
Gerard Defosse
Samir Jegham
Philippe Bovy
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR9605002A priority Critical patent/FR2747678B1/fr
Publication of FR2747678A1 publication Critical patent/FR2747678A1/fr
Application granted granted Critical
Publication of FR2747678B1 publication Critical patent/FR2747678B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FR9605002A 1996-04-22 1996-04-22 Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique Expired - Fee Related FR2747678B1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR9605002A FR2747678B1 (fr) 1996-04-22 1996-04-22 Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9605002A FR2747678B1 (fr) 1996-04-22 1996-04-22 Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique

Publications (2)

Publication Number Publication Date
FR2747678A1 FR2747678A1 (fr) 1997-10-24
FR2747678B1 true FR2747678B1 (fr) 1998-05-22

Family

ID=9491427

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9605002A Expired - Fee Related FR2747678B1 (fr) 1996-04-22 1996-04-22 Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique

Country Status (1)

Country Link
FR (1) FR2747678B1 (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2771093B1 (fr) 1997-11-19 2000-01-21 Synthelabo Derives d'imidazole, leur preparation et leur application en therapeutique
US7771842B2 (en) 2003-06-25 2010-08-10 Nissan Chemical Industries, Ltd. 1,4-benzodioxane sulfonic acid compound and use thereof as electron-acceptor material
CA2609562A1 (fr) 2005-06-14 2006-12-28 Schering Corporation Inhibiteurs heterocycliques et macrocycliques de l'aspartyl protease
MX366703B (es) 2013-03-15 2019-07-22 Incyte Holdings Corp Heterociclos tricíclicos como inhibidores de la proteína bet.
EP3019502B1 (fr) 2013-07-08 2017-05-17 Incyte Holdings Corporation Hétérocycles tricycliques en tant qu'inhibiteurs de protéines bet
WO2015081189A1 (fr) 2013-11-26 2015-06-04 Incyte Corporation Hétérocycles bicycliques servant d'inhibiteurs des protéines bet
US9399640B2 (en) 2013-11-26 2016-07-26 Incyte Corporation Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors
WO2015095492A1 (fr) 2013-12-19 2015-06-25 Incyte Corporation Hétérocycles tricycliques en tant qu'inhibiteurs des protéines bet
KR102702503B1 (ko) 2014-04-23 2024-09-05 인사이트 홀딩스 코포레이션 BET 단백질의 저해제로서의 1H-피롤로[2,3-c]피리딘-7(6H)-온 및 피라졸로[3,4-c]피리딘-7(6H)-온
WO2016044130A1 (fr) * 2014-09-15 2016-03-24 Incyte Corporation Hétérocycles tricycliques utilisés en tant qu'inhibiteurs des protéines bet
US20170121347A1 (en) 2015-10-29 2017-05-04 Incyte Corporation Amorphous solid form of a bet protein inhibitor
PH12021551886A1 (en) 2016-06-20 2023-07-17 Incyte Corp Crystalline solid forms of a bet inhibitor
EP3813827A4 (fr) * 2018-06-28 2022-04-13 Jiangsu Hengrui Medicine Co., Ltd. Composés hétérocycliques tricycliques fusionnés et leurs utilisations thérapeutiques
JP2022511540A (ja) * 2018-12-14 2022-01-31 ジエンス ヘンルイ メデイシンカンパニー リミテッド Stingアゴニストとしての三環式化合物、ならびにその調製方法および医薬用途
EP3938340B1 (fr) * 2019-03-11 2025-07-09 Collaborative Medicinal Development, LLC Dérivés aromatiques hétérobicycliques et hétéroaromatiques pour le traitement de troubles liés à la ferroptose
US11833155B2 (en) 2020-06-03 2023-12-05 Incyte Corporation Combination therapy for treatment of myeloproliferative neoplasms

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2710915B1 (fr) * 1993-10-04 1995-11-24 Synthelabo Dérivés de pipéridine, leur préparation et leur utilisation en thérapeutique.

Also Published As

Publication number Publication date
FR2747678A1 (fr) 1997-10-24

Similar Documents

Publication Publication Date Title
FR2768733B1 (fr) Nouveaux composes 4,4-dihydroxypyrazolin-5-ones ; leurs procedes de preparation et utilisations cosmetiques
EP0912549A4 (fr) Composes et procedes d'obtention de preparations pharmacologiquement actives et leurs utilisations
FR2747678B1 (fr) Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique
FR2751966B1 (fr) Nouveaux derives 1,2-diarylindoles, leurs procedes de preparation, et leurs utilisations en therapeutique
EP1013660A4 (fr) Derives de la 2-fluorofucosyl-n-aroylglucosamine, leurs intermediaires, et leurs procedes d'obtention
IL117807A0 (en) 1,3-dihydro-1-(phenylalkyl)-2h-imidazol-2-one derivatives their preparation and use
FR2753449B1 (fr) Nouveaux derives 3,4-diaryloxazolone, leurs procedes de preparation, et leurs utilisations en therapeutique
DE69618634D1 (de) 1,4-benzodioxin-derivate
FR2769311B1 (fr) Nouveaux derives 3,4-diarylthiazolin-2-one ou -2-thione, leurs procedes de preparation et leurs utilisations en therapeutique
EE9800076A (et) Kombineeritud mullakultiveerimismasin
FR2682679B1 (fr) Nouveaux derives d'alkylpolyosides, leurs procedes de preparation et applications comme agents de surface.
BR9609884A (pt) N-aril- 1,2,4-triazolin-5-onas
FR2751964B1 (fr) Nouveaux derives diarylmethylene carbocycliques, leurs procedes de preparation, et leurs utilisations en therapeutique
FR2689508B1 (fr) Derives de l'imidazole, leur procede de preparation et leur application en therapeutique.
ZA962755B (en) 1,3-dihydro-1-(phenylalkenyl)-2H-imidazol-2-one derivatives.
FR2747123B1 (fr) Nouveaux derives diarylmethylidene tetrahydrofurane, leurs procedes de preparation, et leurs utilisations en therapeutique
FR2771093B1 (fr) Derives d'imidazole, leur preparation et leur application en therapeutique
IL117806A0 (en) 1,3-Dihydro-2h-imidazol-2-one derivatives their preparation and pharmaceutical compositions containing them
FR2751647B1 (fr) Derives de benzimidazole, leurs preparations et leurs applications en therapeutique
FR2775477B1 (fr) Nouveaux derives diarylmethylene heterocycliques, leurs procedes de preparation et leurs utilisations en therapeutique
DE69622415D1 (de) 12H-Dibenzo[d,g][1,3]dioxocin Derivate
FR2772378B1 (fr) Derives d'imidazole, leur preparation et leur application en therapeutique
FR2754256B1 (fr) Nouveaux derives 1,2-diarylmethylenes, leurs procedes de preparation, et leurs utilisations en therapeutique
DE69636837D1 (de) 1,2,4-benzotriazinoxid-formulierungen
MA22143A1 (fr) Derives de 1,5 benzothiazepinone, leurs preparations et leur application

Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse

Effective date: 20051230