FR2747678B1 - Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique - Google Patents
Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutiqueInfo
- Publication number
- FR2747678B1 FR2747678B1 FR9605002A FR9605002A FR2747678B1 FR 2747678 B1 FR2747678 B1 FR 2747678B1 FR 9605002 A FR9605002 A FR 9605002A FR 9605002 A FR9605002 A FR 9605002A FR 2747678 B1 FR2747678 B1 FR 2747678B1
- Authority
- FR
- France
- Prior art keywords
- imidazobenzoxazine
- processes
- preparation
- therapeutic uses
- compounds derived
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 150000001875 compounds Chemical class 0.000 title 1
- UCCWJUWUHMVASJ-UHFFFAOYSA-N imidazo[4,5-h][1,2]benzoxazine Chemical compound C1=CC2=CC=NOC2=C2C1=NC=N2 UCCWJUWUHMVASJ-UHFFFAOYSA-N 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9605002A FR2747678B1 (fr) | 1996-04-22 | 1996-04-22 | Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9605002A FR2747678B1 (fr) | 1996-04-22 | 1996-04-22 | Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2747678A1 FR2747678A1 (fr) | 1997-10-24 |
| FR2747678B1 true FR2747678B1 (fr) | 1998-05-22 |
Family
ID=9491427
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR9605002A Expired - Fee Related FR2747678B1 (fr) | 1996-04-22 | 1996-04-22 | Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique |
Country Status (1)
| Country | Link |
|---|---|
| FR (1) | FR2747678B1 (fr) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2771093B1 (fr) | 1997-11-19 | 2000-01-21 | Synthelabo | Derives d'imidazole, leur preparation et leur application en therapeutique |
| US7771842B2 (en) | 2003-06-25 | 2010-08-10 | Nissan Chemical Industries, Ltd. | 1,4-benzodioxane sulfonic acid compound and use thereof as electron-acceptor material |
| CA2609562A1 (fr) | 2005-06-14 | 2006-12-28 | Schering Corporation | Inhibiteurs heterocycliques et macrocycliques de l'aspartyl protease |
| MX366703B (es) | 2013-03-15 | 2019-07-22 | Incyte Holdings Corp | Heterociclos tricíclicos como inhibidores de la proteína bet. |
| EP3019502B1 (fr) | 2013-07-08 | 2017-05-17 | Incyte Holdings Corporation | Hétérocycles tricycliques en tant qu'inhibiteurs de protéines bet |
| WO2015081189A1 (fr) | 2013-11-26 | 2015-06-04 | Incyte Corporation | Hétérocycles bicycliques servant d'inhibiteurs des protéines bet |
| US9399640B2 (en) | 2013-11-26 | 2016-07-26 | Incyte Corporation | Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors |
| WO2015095492A1 (fr) | 2013-12-19 | 2015-06-25 | Incyte Corporation | Hétérocycles tricycliques en tant qu'inhibiteurs des protéines bet |
| KR102702503B1 (ko) | 2014-04-23 | 2024-09-05 | 인사이트 홀딩스 코포레이션 | BET 단백질의 저해제로서의 1H-피롤로[2,3-c]피리딘-7(6H)-온 및 피라졸로[3,4-c]피리딘-7(6H)-온 |
| WO2016044130A1 (fr) * | 2014-09-15 | 2016-03-24 | Incyte Corporation | Hétérocycles tricycliques utilisés en tant qu'inhibiteurs des protéines bet |
| US20170121347A1 (en) | 2015-10-29 | 2017-05-04 | Incyte Corporation | Amorphous solid form of a bet protein inhibitor |
| PH12021551886A1 (en) | 2016-06-20 | 2023-07-17 | Incyte Corp | Crystalline solid forms of a bet inhibitor |
| EP3813827A4 (fr) * | 2018-06-28 | 2022-04-13 | Jiangsu Hengrui Medicine Co., Ltd. | Composés hétérocycliques tricycliques fusionnés et leurs utilisations thérapeutiques |
| JP2022511540A (ja) * | 2018-12-14 | 2022-01-31 | ジエンス ヘンルイ メデイシンカンパニー リミテッド | Stingアゴニストとしての三環式化合物、ならびにその調製方法および医薬用途 |
| EP3938340B1 (fr) * | 2019-03-11 | 2025-07-09 | Collaborative Medicinal Development, LLC | Dérivés aromatiques hétérobicycliques et hétéroaromatiques pour le traitement de troubles liés à la ferroptose |
| US11833155B2 (en) | 2020-06-03 | 2023-12-05 | Incyte Corporation | Combination therapy for treatment of myeloproliferative neoplasms |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2710915B1 (fr) * | 1993-10-04 | 1995-11-24 | Synthelabo | Dérivés de pipéridine, leur préparation et leur utilisation en thérapeutique. |
-
1996
- 1996-04-22 FR FR9605002A patent/FR2747678B1/fr not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| FR2747678A1 (fr) | 1997-10-24 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR2768733B1 (fr) | Nouveaux composes 4,4-dihydroxypyrazolin-5-ones ; leurs procedes de preparation et utilisations cosmetiques | |
| EP0912549A4 (fr) | Composes et procedes d'obtention de preparations pharmacologiquement actives et leurs utilisations | |
| FR2747678B1 (fr) | Composes derives d'imidazobenzoxazine, leurs procedes de preparation et leurs utilisations en therapeutique | |
| FR2751966B1 (fr) | Nouveaux derives 1,2-diarylindoles, leurs procedes de preparation, et leurs utilisations en therapeutique | |
| EP1013660A4 (fr) | Derives de la 2-fluorofucosyl-n-aroylglucosamine, leurs intermediaires, et leurs procedes d'obtention | |
| IL117807A0 (en) | 1,3-dihydro-1-(phenylalkyl)-2h-imidazol-2-one derivatives their preparation and use | |
| FR2753449B1 (fr) | Nouveaux derives 3,4-diaryloxazolone, leurs procedes de preparation, et leurs utilisations en therapeutique | |
| DE69618634D1 (de) | 1,4-benzodioxin-derivate | |
| FR2769311B1 (fr) | Nouveaux derives 3,4-diarylthiazolin-2-one ou -2-thione, leurs procedes de preparation et leurs utilisations en therapeutique | |
| EE9800076A (et) | Kombineeritud mullakultiveerimismasin | |
| FR2682679B1 (fr) | Nouveaux derives d'alkylpolyosides, leurs procedes de preparation et applications comme agents de surface. | |
| BR9609884A (pt) | N-aril- 1,2,4-triazolin-5-onas | |
| FR2751964B1 (fr) | Nouveaux derives diarylmethylene carbocycliques, leurs procedes de preparation, et leurs utilisations en therapeutique | |
| FR2689508B1 (fr) | Derives de l'imidazole, leur procede de preparation et leur application en therapeutique. | |
| ZA962755B (en) | 1,3-dihydro-1-(phenylalkenyl)-2H-imidazol-2-one derivatives. | |
| FR2747123B1 (fr) | Nouveaux derives diarylmethylidene tetrahydrofurane, leurs procedes de preparation, et leurs utilisations en therapeutique | |
| FR2771093B1 (fr) | Derives d'imidazole, leur preparation et leur application en therapeutique | |
| IL117806A0 (en) | 1,3-Dihydro-2h-imidazol-2-one derivatives their preparation and pharmaceutical compositions containing them | |
| FR2751647B1 (fr) | Derives de benzimidazole, leurs preparations et leurs applications en therapeutique | |
| FR2775477B1 (fr) | Nouveaux derives diarylmethylene heterocycliques, leurs procedes de preparation et leurs utilisations en therapeutique | |
| DE69622415D1 (de) | 12H-Dibenzo[d,g][1,3]dioxocin Derivate | |
| FR2772378B1 (fr) | Derives d'imidazole, leur preparation et leur application en therapeutique | |
| FR2754256B1 (fr) | Nouveaux derives 1,2-diarylmethylenes, leurs procedes de preparation, et leurs utilisations en therapeutique | |
| DE69636837D1 (de) | 1,2,4-benzotriazinoxid-formulierungen | |
| MA22143A1 (fr) | Derives de 1,5 benzothiazepinone, leurs preparations et leur application |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TP | Transmission of property | ||
| ST | Notification of lapse |
Effective date: 20051230 |