[go: up one dir, main page]

FR2668153B1 - NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM. - Google Patents

NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.

Info

Publication number
FR2668153B1
FR2668153B1 FR9013047A FR9013047A FR2668153B1 FR 2668153 B1 FR2668153 B1 FR 2668153B1 FR 9013047 A FR9013047 A FR 9013047A FR 9013047 A FR9013047 A FR 9013047A FR 2668153 B1 FR2668153 B1 FR 2668153B1
Authority
FR
France
Prior art keywords
novel
preparation
medicaments containing
ribonucleoside compounds
ribonucleoside
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9013047A
Other languages
French (fr)
Other versions
FR2668153A1 (en
Inventor
Lino Ronco Gino
Bougrine Tber
Pierre Villa
Joseph
Guy Ville
Andre
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Pasteur SA
Original Assignee
Pasteur Merieux Serum et Vaccines SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pasteur Merieux Serum et Vaccines SA filed Critical Pasteur Merieux Serum et Vaccines SA
Priority to FR9013047A priority Critical patent/FR2668153B1/en
Priority to PCT/FR1991/000831 priority patent/WO1992006993A1/en
Priority to EP19910919546 priority patent/EP0506935A1/en
Publication of FR2668153A1 publication Critical patent/FR2668153A1/en
Application granted granted Critical
Publication of FR2668153B1 publication Critical patent/FR2668153B1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9013047A 1990-10-22 1990-10-22 NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM. Expired - Fee Related FR2668153B1 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FR9013047A FR2668153B1 (en) 1990-10-22 1990-10-22 NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.
PCT/FR1991/000831 WO1992006993A1 (en) 1990-10-22 1991-10-22 Novel ribonucleoside compounds, process for their preparation and drugs containing said compounds
EP19910919546 EP0506935A1 (en) 1990-10-22 1991-10-22 Novel ribonucleoside compounds, process for their preparation and drugs containing said compounds

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9013047A FR2668153B1 (en) 1990-10-22 1990-10-22 NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.

Publications (2)

Publication Number Publication Date
FR2668153A1 FR2668153A1 (en) 1992-04-24
FR2668153B1 true FR2668153B1 (en) 1995-03-31

Family

ID=9401445

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9013047A Expired - Fee Related FR2668153B1 (en) 1990-10-22 1990-10-22 NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.

Country Status (3)

Country Link
EP (1) EP0506935A1 (en)
FR (1) FR2668153B1 (en)
WO (1) WO1992006993A1 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ234534A (en) * 1989-07-17 1994-12-22 Univ Birmingham Pyrimidine 4'-thionucleoside derivatives and their preparation; intermediates therefor
US5591722A (en) * 1989-09-15 1997-01-07 Southern Research Institute 2'-deoxy-4'-thioribonucleosides and their antiviral activity
US5478928A (en) * 1990-04-20 1995-12-26 Southern Research Institute 2',3'-dideoxy-4'-thioribonucleosides and synthetic precursors thereof
US5521163A (en) * 1990-07-13 1996-05-28 University Of Birmingham Antiviral pyrimidine nucleosides and methods for using same
GB9218810D0 (en) * 1992-09-04 1992-10-21 Univ Birmingham Antiviral pyrimidine nucleosides
WO1996001834A1 (en) * 1994-07-12 1996-01-25 Yamasa Corporation 2'-deoxy-2'-(substituted or unsubstituted methylidene)-4'-thionucleoside
AU2018205994B2 (en) * 2017-01-06 2021-09-09 F. Hoffmann-La Roche Ag Process for the preparation of 3-substituted 5-amino-6H-thiazolo[4,5-d]pyrimidine-2,7-dione compounds

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK166805B1 (en) * 1985-03-16 1993-07-19 Wellcome Found THE THREO ISOMER OF 3'-AZIDO-3'-DEOXYTHYMIDINE FOR USING THE TREATMENT OR PROPHYLAXY OF HUMAN RETROVIRUS INFECTIONS, USING THE COMPOUND FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION OF A MEDICINAL PRODUCT AND NAVE MEDICINE
HU196607B (en) * 1985-05-15 1988-12-28 Wellcome Found Process for producing dideoxy-nucleosides and pharmaceutics comprising such compounds
ATE190064T1 (en) * 1985-09-17 2000-03-15 Wellcome Found COMBINATION THERAPEUTIC NUCLEOSIDES WITH OTHER THERAPEUTICALLY EFFECTIVE COMPONENTS.
DD279407A1 (en) * 1986-07-24 1990-06-06 Akad Wissenschaften Ddr METHOD FOR PRODUCING AN AGENT AGAINST AIDS
EP0311107A3 (en) * 1987-10-08 1990-04-18 Stichting REGA V.Z.W. Anti-hiv active 3'-fluoro-purine-2',3'-dideoxyribosides
GB8726136D0 (en) * 1987-11-07 1987-12-09 Wellcome Found Therapeutic nucleosides
HU204843B (en) * 1988-09-27 1992-02-28 Merrell Dow Pharma Process for producing 2'-halogen-methylidene adenosine derivatives and pharmaceutical compositions comprising same
ZA898567B (en) * 1988-11-15 1990-08-29 Merrell Dow Pharma Novel 2'-halomethylidene,2'-ethenylidene and 2'-ethynyl cytidine,uridine and guanosine derivatives
IE74701B1 (en) * 1989-10-04 1997-07-30 Univ Birmingham Further antiviral pyrimidine nucleosides

Also Published As

Publication number Publication date
FR2668153A1 (en) 1992-04-24
WO1992006993A1 (en) 1992-04-30
EP0506935A1 (en) 1992-10-07

Similar Documents

Publication Publication Date Title
FR2676230B1 (en) NOVEL PYRROLO [1,4] -BENZODIAZEPINES DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.
FR2567131B1 (en) NOVEL GANGLIOSIDE DERIVATIVES, PROCESS FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME
FR2603584B1 (en) NOVEL BENZOHETEROCYCLIC COMPOUNDS USEFUL AS ANTIMICROBIAL AGENTS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM
FR2518095B1 (en) NOVEL L-OXA-, THIA- AND AZA-SPIROCYCLO-BENZENE-ACETAMIDES AND BENZAMIDES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITION CONTAINING THEM
PT78340A (en) PROCESS FOR THE PREPARATION OF NOVEL 3', 4 ', 5,7-FLAVONE TETRAHYDROXY DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
FR2556343B1 (en) NOVEL AMINOGUANIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM
BE885268A (en) NOVEL N-PROPIONYL-SARCOSINE-ANILIDES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM
MA20664A1 (en) HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION PROCESS AND FUNGICIDAL COMPOSITIONS CONTAINING THEM
MA21588A1 (en) N-PHERYL PYRAZOLE-4-YLE ETHER DERIVATIVES, COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION.
FR2668153B1 (en) NOVEL RIBONUCLEOSIDE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM.
FR2671551B1 (en) NOVEL ARYL TRIAZINIC STRUCTURE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME.
BE884620A (en) NOVEL HALOVINCAMONE DERIVATIVES, THEIR PREPARATION METHOD AND MEDICAMENTS CONTAINING THEM
BE862278A (en) NEW HETEROCYCLIC COMPOUNDS, THEIR PREPARATION PROCESS AND THE MEDICINAL PRODUCT CONTAINING THEM
FR2556721B1 (en) NOVEL AMINO-ACID O-MERCAPTOPROPANAMIDE DERIVATIVES, THEIR PREPARATION PROCESS, THEIR USE AS MEDICAMENTS AND THE COMPOSITIONS CONTAINING THEM
FR2558835B1 (en) HYDANTOIN DERIVATIVES, THEIR PRODUCTION PROCESS AND MEDICAMENT CONTAINING THEM
FR2733498B1 (en) NOVEL CYCLOHEXANIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FR2669633B1 (en) NOVEL BENZOSELENAZOLINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
BE889990A (en) NOVEL CYTOSTATIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM
FR2648132B1 (en) PIGMENTOGENIC COMPOUNDS, DIFFUSION VEHICLES THEREOF, COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION
FR2528044B1 (en) ISOQUINOLEIN DERIVATIVES, THEIR PREPARATION METHOD AND MEDICAMENTS CONTAINING THEM
FR2603587B1 (en) 2,3,4,5,6,7-HEXAHYDRO-2,7-METHANO-1,5-BENZOXAZONINE (OR -1,4-BENZOXAZONINE) DERIVATIVES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATE COMPOUNDS
FR2508040B1 (en) PROLINE DERIVATIVES, THEIR PREPARATION PROCESS AND THE MEDICAMENT CONTAINING THEM
FR2549053B1 (en) NOVEL PYRROLIDINE DERIVATIVES ACTIVE IN THE CENTRAL NERVOUS SYSTEM, THEIR PREPARATION METHOD, THE MEDICINAL PRODUCTS CONTAINING THEM
BE887833A (en) NOVEL STEROID-SPIRO-OXATHIAZOLIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM
FR2551440B1 (en) AMINOCYCLOPENTANES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Legal Events

Date Code Title Description
ST Notification of lapse