FR2574793B1 - Composes derives d'indole, compositions pharmaceutiques les contenant et procede pour leur preparation - Google Patents
Composes derives d'indole, compositions pharmaceutiques les contenant et procede pour leur preparationInfo
- Publication number
- FR2574793B1 FR2574793B1 FR8518416A FR8518416A FR2574793B1 FR 2574793 B1 FR2574793 B1 FR 2574793B1 FR 8518416 A FR8518416 A FR 8518416A FR 8518416 A FR8518416 A FR 8518416A FR 2574793 B1 FR2574793 B1 FR 2574793B1
- Authority
- FR
- France
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- indole derivatives
- indole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- SIKJAQJRHWYJAI-UHFFFAOYSA-N Indole Chemical class C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 title 1
- 229940054051 antipsychotic indole derivative Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB848431426A GB8431426D0 (en) | 1984-12-13 | 1984-12-13 | Chemical compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2574793A1 FR2574793A1 (fr) | 1986-06-20 |
| FR2574793B1 true FR2574793B1 (fr) | 1988-10-14 |
Family
ID=10571103
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR8518416A Expired FR2574793B1 (fr) | 1984-12-13 | 1985-12-12 | Composes derives d'indole, compositions pharmaceutiques les contenant et procede pour leur preparation |
Country Status (11)
| Country | Link |
|---|---|
| JP (1) | JPS61151172A (fr) |
| AU (1) | AU579687B2 (fr) |
| BE (1) | BE903846A (fr) |
| CH (1) | CH667454A5 (fr) |
| DE (1) | DE3543982A1 (fr) |
| FR (1) | FR2574793B1 (fr) |
| GB (2) | GB8431426D0 (fr) |
| IT (1) | IT1182089B (fr) |
| NL (1) | NL8503424A (fr) |
| SE (1) | SE8505887L (fr) |
| ZA (1) | ZA859520B (fr) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8530507D0 (en) * | 1985-12-11 | 1986-01-22 | Glaxo Group Plc | Chemical compounds |
| GB8607824D0 (en) * | 1986-03-27 | 1986-04-30 | Glaxo Group Ltd | Chemical compounds |
| GB8614287D0 (en) * | 1986-06-12 | 1986-07-16 | Glaxo Group Ltd | Chemical compounds |
| US4894386A (en) * | 1987-04-15 | 1990-01-16 | Ici Americas Inc. | Aliphatic carboxamides |
| GB8719167D0 (en) * | 1987-08-13 | 1987-09-23 | Glaxo Group Ltd | Chemical compounds |
| US5225431A (en) * | 1987-10-23 | 1993-07-06 | Burroughs Wellcome Co. | Therapeutic substituted indole compounds and compositions thereof |
| EP0636623B1 (fr) * | 1990-06-07 | 2001-08-16 | AstraZeneca AB | Dérivés d'indole comme 5-HT1-like agonistes |
| GB9209882D0 (en) * | 1992-05-07 | 1992-06-24 | Glaxo Lab Sa | Compositions |
| GB9211277D0 (en) | 1992-05-28 | 1992-07-15 | Glaxo Group Inc | Pharmaceutical compositions |
| GB9216009D0 (en) * | 1992-07-28 | 1992-09-09 | Almirall Lab | New indol derivatives |
| ES2056025B1 (es) * | 1992-10-08 | 1995-05-01 | Almirall Lab | Nuevos derivados de indol. |
| FR2707639B1 (fr) * | 1993-06-30 | 1995-10-13 | Pf Medicament | Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. |
| US7189753B1 (en) | 1997-11-06 | 2007-03-13 | Cady Roger K | Preemptive prophylaxis of migraine |
| WO2004056769A2 (fr) | 2002-12-20 | 2004-07-08 | Ciba Specialty Chemicals Holding Inc. | Synthèse d'amines et intermédiaires pour cette synthèse |
| WO2005118551A2 (fr) | 2004-05-28 | 2005-12-15 | Ligand Pharmaceuticals Inc. | Composes modulant l'activite de la thrombopoietine et methodes associees |
| ATE486859T1 (de) * | 2004-10-25 | 2010-11-15 | Ligand Pharm Inc | Verbindungen modulierende thrombopoietinaktivität und verfahren |
| EP2141148B1 (fr) | 2007-03-29 | 2013-07-03 | Daiichi Sankyo Company, Limited | Dérivé d'indole ayant une activité inhibitrice de cpla2, utilisation de celui-ci et procédé de production de celui-ci |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA795239B (en) * | 1978-10-12 | 1980-11-26 | Glaxo Group Ltd | Heterocyclic compounds |
| GB2082175B (en) * | 1980-08-12 | 1984-05-02 | Glaxo Group Ltd | Heterocyclic compounds |
| SE8505715L (sv) * | 1984-12-04 | 1986-06-05 | Glaxo Group Ltd | Indolderivat |
| GB8530507D0 (en) * | 1985-12-11 | 1986-01-22 | Glaxo Group Plc | Chemical compounds |
-
1984
- 1984-12-13 GB GB848431426A patent/GB8431426D0/en active Pending
-
1985
- 1985-12-12 BE BE0/216004A patent/BE903846A/fr not_active IP Right Cessation
- 1985-12-12 IT IT48921/85A patent/IT1182089B/it active
- 1985-12-12 AU AU51151/85A patent/AU579687B2/en not_active Ceased
- 1985-12-12 ZA ZA859520A patent/ZA859520B/xx unknown
- 1985-12-12 JP JP60278124A patent/JPS61151172A/ja active Pending
- 1985-12-12 FR FR8518416A patent/FR2574793B1/fr not_active Expired
- 1985-12-12 CH CH5301/85A patent/CH667454A5/fr not_active IP Right Cessation
- 1985-12-12 DE DE19853543982 patent/DE3543982A1/de not_active Withdrawn
- 1985-12-12 SE SE8505887A patent/SE8505887L/xx not_active Application Discontinuation
- 1985-12-12 GB GB08530591A patent/GB2168347B/en not_active Expired
- 1985-12-12 NL NL8503424A patent/NL8503424A/nl not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| FR2574793A1 (fr) | 1986-06-20 |
| GB2168347A (en) | 1986-06-18 |
| IT8548921A0 (it) | 1985-12-12 |
| AU5115185A (en) | 1986-06-19 |
| GB8431426D0 (en) | 1985-01-23 |
| SE8505887L (sv) | 1986-06-14 |
| IT1182089B (it) | 1987-09-30 |
| CH667454A5 (fr) | 1988-10-14 |
| BE903846A (fr) | 1986-06-12 |
| ZA859520B (en) | 1986-08-27 |
| DE3543982A1 (de) | 1986-06-19 |
| GB8530591D0 (en) | 1986-01-22 |
| JPS61151172A (ja) | 1986-07-09 |
| NL8503424A (nl) | 1986-07-01 |
| AU579687B2 (en) | 1988-12-01 |
| SE8505887D0 (sv) | 1985-12-12 |
| GB2168347B (en) | 1988-02-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |