FR14C0039I1 - Formulation d'aripiprazole injectable sterile a liberation controlee et procede - Google Patents

Formulation d'aripiprazole injectable sterile a liberation controlee et procede

Info

Publication number: FR14C0039I1
Authority: FR; France
Prior art keywords: controlled release; sterile injectable; aripiprazole formulation; release sterile; injectable aripiprazole
Prior art date: 2003-10-23
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Active

Application number

FR14C0039C

Other languages

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Otsuka Pharmaceutical Co Ltd

Original Assignee

Otsuka Pharmaceutical Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-10-23

Filing date

2014-05-13

Publication date

2014-06-27

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34549292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR14C0039(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2014-05-13 Application filed by Otsuka Pharmaceutical Co Ltd filed Critical Otsuka Pharmaceutical Co Ltd

2014-06-27 Publication of FR14C0039I1 publication Critical patent/FR14C0039I1/fr

Status Active legal-status Critical Current

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Inorganic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Dermatology (AREA)
Neurosurgery (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Oil, Petroleum & Natural Gas (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)

FR14C0039C 2003-10-23 2014-05-13 Formulation d'aripiprazole injectable sterile a liberation controlee et procede Active FR14C0039I1 (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US51361803P	2003-10-23	2003-10-23
PCT/US2004/034367 WO2005041937A2 (en)	2003-10-23	2004-10-18	Controlled release sterile injectable aripiprazole formulation and method

Publications (1)

Publication Number	Publication Date
FR14C0039I1 true FR14C0039I1 (fr)	2014-06-27

Family

ID=34549292

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FR14C0039C Active FR14C0039I1 (fr)	2003-10-23	2014-05-13	Formulation d'aripiprazole injectable sterile a liberation controlee et procede

Country Status (32)

Country	Link
US (12)	US7807680B2 (da)
EP (1)	EP1675573B2 (da)
JP (2)	JP4836797B2 (da)
KR (1)	KR100931784B1 (da)
CN (1)	CN1870980B (da)
AR (2)	AR046141A1 (da)
AT (1)	ATE411797T2 (da)
AU (1)	AU2004285448C1 (da)
BR (1)	BRPI0415531B8 (da)
CA (1)	CA2543242C (da)
CO (1)	CO5690539A2 (da)
CY (2)	CY1109040T1 (da)
DE (1)	DE602004017342D1 (da)
DK (1)	DK1675573T4 (da)
EC (2)	ECSP066512A (da)
ES (1)	ES2315721T5 (da)
FR (1)	FR14C0039I1 (da)
GE (1)	GEP20115205B (da)
IL (1)	IL175072A (da)
LU (1)	LU92427I2 (da)
MX (1)	MXPA06004489A (da)
MY (1)	MY146093A (da)
NO (2)	NO334919B1 (da)
NZ (1)	NZ546063A (da)
PE (1)	PE20050811A1 (da)
PL (1)	PL1675573T4 (da)
PT (1)	PT1675573E (da)
SI (1)	SI1675573T2 (da)
TW (2)	TWI383810B (da)
UA (1)	UA82561C2 (da)
WO (1)	WO2005041937A2 (da)
ZA (1)	ZA200602347B (da)

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2004
- 2004-10-18 PL PL04795514T patent/PL1675573T4/pl unknown
- 2004-10-18 SI SI200430966T patent/SI1675573T2/sl unknown
- 2004-10-18 JP JP2006536693A patent/JP4836797B2/ja not_active Expired - Lifetime
- 2004-10-18 MX MXPA06004489A patent/MXPA06004489A/es active IP Right Grant
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- 2004-10-18 ZA ZA200602347A patent/ZA200602347B/en unknown
- 2004-10-18 DE DE602004017342T patent/DE602004017342D1/de not_active Expired - Lifetime
- 2004-10-18 AT AT04795514T patent/ATE411797T2/de active
- 2004-10-18 UA UAA200604046A patent/UA82561C2/uk unknown
- 2004-10-18 PT PT04795514T patent/PT1675573E/pt unknown
- 2004-10-18 AU AU2004285448A patent/AU2004285448C1/en active Active
- 2004-10-18 EP EP04795514A patent/EP1675573B2/en not_active Expired - Lifetime
- 2004-10-18 ES ES04795514T patent/ES2315721T5/es not_active Expired - Lifetime
- 2004-10-18 DK DK04795514.1T patent/DK1675573T4/da active
- 2004-10-18 NZ NZ546063A patent/NZ546063A/en not_active IP Right Cessation
- 2004-10-18 BR BRPI0415531A patent/BRPI0415531B8/pt active IP Right Grant
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- 2004-10-18 CN CN2004800308144A patent/CN1870980B/zh not_active Expired - Lifetime
- 2004-10-18 CA CA2543242A patent/CA2543242C/en not_active Expired - Lifetime
- 2004-10-18 WO PCT/US2004/034367 patent/WO2005041937A2/en not_active Ceased
- 2004-10-19 US US10/968,482 patent/US7807680B2/en not_active Expired - Lifetime
- 2004-10-20 TW TW093131836A patent/TWI383810B/zh not_active IP Right Cessation
- 2004-10-20 TW TW100136057A patent/TWI421101B/zh not_active IP Right Cessation
- 2004-10-22 AR ARP040103849A patent/AR046141A1/es not_active Application Discontinuation
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2006
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2007
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- 2007-10-31 US US11/979,149 patent/US8030313B2/en active Active
- 2007-10-31 US US11/979,145 patent/US8722679B2/en active Active
- 2007-10-31 US US11/979,144 patent/US20080112985A1/en not_active Abandoned
2008
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- 2011-12-28 US US13/338,827 patent/US8952013B2/en active Active
2012
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2013
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2014
- 2014-04-11 LU LU92427C patent/LU92427I2/fr unknown
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2016
- 2016-10-21 AR ARP160103230A patent/AR106449A2/es not_active Application Discontinuation
2017
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2019
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2021
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Also Published As

Publication number	Publication date
DK1675573T3 (da)	2009-01-05
ECSP12006512A (es)	2012-02-29
ECSP066512A (es)	2006-10-10
PT1675573E (pt)	2008-12-30
TW201204413A (en)	2012-02-01
WO2005041937A3 (en)	2006-04-06
US9763935B2 (en)	2017-09-19
US20140018369A1 (en)	2014-01-16
RU2342927C2 (ru)	2009-01-10
AR046141A1 (es)	2005-11-23
GEP20115205B (en)	2011-04-26
BRPI0415531B8 (pt)	2021-05-25
SI1675573T2 (sl)	2012-08-31
UA82561C2 (uk)	2008-04-25
KR100931784B1 (ko)	2009-12-14
NO2014027I2 (no)	2014-10-27
US8030313B2 (en)	2011-10-04
US20080107745A1 (en)	2008-05-08
US20080112986A1 (en)	2008-05-15
ES2315721T3 (es)	2009-04-01
TW200524638A (en)	2005-08-01
NZ546063A (en)	2009-05-31
CY1109040T1 (el)	2014-07-02
US7807680B2 (en)	2010-10-05
BRPI0415531B1 (pt)	2019-07-30
ES2315721T5 (es)	2012-08-24
NO334919B1 (no)	2014-07-14
US20200061057A1 (en)	2020-02-27
ZA200602347B (en)	2007-09-26
TWI383810B (zh)	2013-02-01
CN1870980B (zh)	2010-06-23
CN1870980A (zh)	2006-11-29
ES2315721T9 (es)	2015-11-05
IL175072A0 (en)	2006-08-20
JP2007509148A (ja)	2007-04-12
JP5372032B2 (ja)	2013-12-18
NO20062319L (no)	2006-07-21
CA2543242C (en)	2015-04-14
DK1675573T4 (da)	2012-08-06
ATE411797T2 (de)	2008-11-15
PE20050811A1 (es)	2005-09-25
AU2004285448A1 (en)	2005-05-12
US20120100190A1 (en)	2012-04-26
EP1675573A2 (en)	2006-07-05
DE602004017342D1 (de)	2008-12-04
SI1675573T1 (sl)	2009-02-28
US8952013B2 (en)	2015-02-10
LU92427I2 (fr)	2014-06-11
JP2011102316A (ja)	2011-05-26
EP1675573B1 (en)	2008-10-22
CY2014021I2 (el)	2017-03-15
US20080221121A1 (en)	2008-09-11
US20210338663A1 (en)	2021-11-04
MY146093A (en)	2012-06-29
CO5690539A2 (es)	2006-10-31
BRPI0415531A (pt)	2006-12-26
RU2006109111A (ru)	2007-09-27
US20150024056A1 (en)	2015-01-22
AU2004285448C1 (en)	2021-08-19
NO2014027I1 (no)	2014-11-10
PL1675573T3 (pl)	2009-04-30
CY2014021I1 (el)	2014-07-02
MXPA06004489A (es)	2006-06-20
HK1095266A1 (zh)	2007-05-04
TWI421101B (zh)	2014-01-01
KR20060118450A (ko)	2006-11-23
PL1675573T5 (pl)	2012-10-31
IL175072A (en)	2015-06-30
US20240261280A1 (en)	2024-08-08
PL1675573T4 (pl)	2016-04-29
LU92427I9 (da)	2019-01-17
CA2543242A1 (en)	2005-05-12
US20170348308A1 (en)	2017-12-07
AR106449A2 (es)	2018-01-17
US20080112985A1 (en)	2008-05-15
WO2005041937A2 (en)	2005-05-12
EP1675573B2 (en)	2012-06-13
JP4836797B2 (ja)	2011-12-14
US20050148597A1 (en)	2005-07-07
AU2004285448B2 (en)	2009-06-11
US8722679B2 (en)	2014-05-13

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