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FR11C0037I1 - - Google Patents

Info

Publication number
FR11C0037I1
FR11C0037I1 FR11C0037C FR11C0037I1 FR 11C0037 I1 FR11C0037 I1 FR 11C0037I1 FR 11C0037 C FR11C0037 C FR 11C0037C FR 11C0037 I1 FR11C0037 I1 FR 11C0037I1
Authority
FR
France
Prior art keywords
derivatives
peperidino
mycaminosyltylonolide
pasteurellosis
disubstituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
Other languages
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of FR11C0037I1 publication Critical patent/FR11C0037I1/fr
Application granted granted Critical
Publication of FR11C0037I2 publication Critical patent/FR11C0037I2/en
Active legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Dental Preparations (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)
  • External Artificial Organs (AREA)
  • Materials For Medical Uses (AREA)

Abstract

20,23-disubstituted mycaminosyltylonolide derivatives and use of the same in the field of the prophylaxis and treatment of pasteurellosis are disclosed. The di-substituents are peperidino optionally substituted with one or two methyl groups. The derivatives have selective antibacterial activity against Pasteurella.
FR11C0037C 1999-08-30 2011-09-09 MACROLID ANTIBIOTICS AND THE TREATMENT OF PASTEURELLOSIS Active FR11C0037I2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP24328699 1999-08-30
PCT/JP2000/005721 WO2001016148A1 (en) 1999-08-30 2000-08-24 Macrolide antibiotics and treatment of pasteurellosis

Publications (2)

Publication Number Publication Date
FR11C0037I1 true FR11C0037I1 (en) 2011-10-14
FR11C0037I2 FR11C0037I2 (en) 2012-06-22

Family

ID=17101600

Family Applications (1)

Application Number Title Priority Date Filing Date
FR11C0037C Active FR11C0037I2 (en) 1999-08-30 2011-09-09 MACROLID ANTIBIOTICS AND THE TREATMENT OF PASTEURELLOSIS

Country Status (13)

Country Link
US (1) US6514946B1 (en)
EP (1) EP1216256B1 (en)
JP (1) JP4573411B2 (en)
AT (1) ATE261450T1 (en)
AU (1) AU763732B2 (en)
BE (1) BE2011C037I2 (en)
CA (1) CA2391834C (en)
DE (2) DE60008895T2 (en)
DK (1) DK1216256T3 (en)
ES (1) ES2213597T3 (en)
FR (1) FR11C0037I2 (en)
PT (1) PT1216256E (en)
WO (1) WO2001016148A1 (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006206952B2 (en) 2005-01-24 2011-08-18 Microbial Chemistry Research Foundation Anti-penicillin resistant pneumococci agent and novel 16-membered ring macrolide derivative
US9148795B2 (en) * 2005-12-22 2015-09-29 Qualcomm Incorporated Methods and apparatus for flexible reporting of control information
RU2450014C2 (en) * 2006-07-28 2012-05-10 Интервет Интернэшнл Б.В. Method of macrolide synthesis
CA2657483C (en) * 2006-07-28 2012-10-09 Intervet International B.V. Macrolide synthesis process
CN101506220B (en) * 2006-07-28 2012-10-17 英特威国际有限公司 Synthetic method of macrolide
EP2019112A1 (en) * 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
CN102863487B (en) * 2012-10-08 2014-11-05 齐鲁动物保健品有限公司 Process for preparing 20,23-bi-piperidyl-5-O-carbon mould amine glycosyl-tylosin lactone
PT2999707T (en) * 2013-05-23 2018-05-23 Kitasato Inst Tylosin derivatives and method for preparation thereof
CN103554203A (en) * 2013-08-17 2014-02-05 齐鲁动物保健品有限公司 Amorphous crystal of tylonolide, and preparation method thereof
CN108864228B (en) * 2014-01-22 2021-02-02 镇江威特药业有限责任公司 Sixteen-membered ring triamine lactone derivative and application thereof
CN103923141B (en) * 2014-04-21 2016-04-27 西南大学 A kind of synthetic method of relying on tilmicosin
CN104478974B (en) * 2014-11-28 2016-08-17 武汉回盛生物科技有限公司 A kind of 20, the synthetic method of 23-dipiperidino-5-O-mycamino syl-tylono lide
CN104447919B (en) * 2014-11-28 2017-03-08 武汉回盛生物科技股份有限公司 A kind of process for purification of 20,23 dipiperidino, 5 O mycaminose Ji Taile lactone bulk drug
CN104497082B (en) * 2015-01-13 2017-12-12 中国兽医药品监察所 A kind of synthetic method of tylonolide
CN104558076A (en) * 2015-02-10 2015-04-29 上海皓元化学科技有限公司 Preparation method of tildipirosin and intermediate compounds of tildipirosin
US10287275B2 (en) * 2015-04-16 2019-05-14 Victor Pharma Co., Ltd. Zhenjiang 16-member triamilide derivatives and uses thereof
CN105440093A (en) * 2015-11-17 2016-03-30 宁夏泰瑞制药股份有限公司 Synthetic method of tildipirosin
CN105919933A (en) * 2016-06-13 2016-09-07 上海同仁药业股份有限公司 Tildipirosin injection and preparation method thereof
CN106420600A (en) * 2016-09-21 2017-02-22 中国水产科学研究院珠江水产研究所 In situ gel for tilmicosin injection and preparation method thereof
CN108264530A (en) * 2016-12-30 2018-07-10 湖北回盛生物科技有限公司 20,23- dihalo -5-O- mycamino syl-tylono lides and its synthetic method and application
CN108264529A (en) * 2016-12-30 2018-07-10 湖北回盛生物科技有限公司 A kind of synthetic method of bis- piperidines -5-O- mycamino syl-tylono lides of 20,23-
JP2023551551A (en) * 2020-12-03 2023-12-08 インターベット インターナショナル ベー． フェー． How to treat hoof rot
CN116731096B (en) * 2023-06-10 2025-03-04 中国兽医药品监察所 20-Aldehyde-23-piperidyl-5-O-carbomycaminose-tylosin lactone and its synthesis process and use

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4454314A (en) 1982-08-02 1984-06-12 Pfizer Inc. Antibacterial mycaminosyl tylonolide and related macrolide derivatives
JPS5951299A (en) * 1982-09-17 1984-03-24 Microbial Chem Res Found 23-deoxy-20-dihydro-mycaminosyltylonolide derivative
JPS59225199A (en) * 1983-02-10 1984-12-18 Microbial Chem Res Found 20,23-dideoxy-23-alkyleneimino-20-substituted amino mycaminosylleronolide
ZA841277B (en) * 1983-02-28 1985-09-25 Lilly Co Eli C-20-and c-23-modified macrolide derivatives
IL71032A0 (en) * 1983-02-28 1984-05-31 Lilly Co Eli C-20 and c-23-modified macrolide derivatives
US4629786A (en) 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
JPS59181299A (en) * 1983-03-31 1984-10-15 Microbial Chem Res Found 20,23-dideoxy-20,23-bis-substituted amino-mycaminosylleronolide
JPS59227897A (en) * 1983-06-10 1984-12-21 Microbial Chem Res Found 20,23-dideoxy-23-alkyleneimino-20-substituted-mycaminosylleronolide
US4604380A (en) * 1985-01-18 1986-08-05 Eli Lilly And Company C-23-substituted mycaminosyltylonolide compounds, pharmaceutical compositions and methods of use
TW226373B (en) * 1992-07-15 1994-07-11 Pfizer

Also Published As

Publication number Publication date
CA2391834C (en) 2008-08-05
JP2001139592A (en) 2001-05-22
EP1216256A1 (en) 2002-06-26
JP4573411B2 (en) 2010-11-04
DE122011100013I1 (en) 2011-09-15
DK1216256T3 (en) 2004-06-21
ATE261450T1 (en) 2004-03-15
PT1216256E (en) 2004-07-30
AU763732B2 (en) 2003-07-31
US6514946B1 (en) 2003-02-04
AU6729400A (en) 2001-03-26
DE60008895T2 (en) 2005-01-20
BE2011C037I2 (en) 2019-10-16
CA2391834A1 (en) 2001-03-08
ES2213597T3 (en) 2004-09-01
WO2001016148A1 (en) 2001-03-08
FR11C0037I2 (en) 2012-06-22
EP1216256B1 (en) 2004-03-10
DE60008895D1 (en) 2004-04-15

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