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FI981956A0 - 2-(4-hydroksipiperidino)-1-alkanolijohdannaisia verettömyyden vastaisia aineina - Google Patents

2-(4-hydroksipiperidino)-1-alkanolijohdannaisia verettömyyden vastaisia aineina

Info

Publication number
FI981956A0
FI981956A0 FI981956A FI981956A FI981956A0 FI 981956 A0 FI981956 A0 FI 981956A0 FI 981956 A FI981956 A FI 981956A FI 981956 A FI981956 A FI 981956A FI 981956 A0 FI981956 A0 FI 981956A0
Authority
FI
Finland
Prior art keywords
hydroxypiperidino
ischemic agents
alkanol derivatives
alkanol
derivatives
Prior art date
Application number
FI981956A
Other languages
English (en)
Swedish (sv)
Other versions
FI981956L (fi
FI981956A7 (fi
Inventor
Jr Willard Mckowan Welch
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI981956L publication Critical patent/FI981956L/fi
Publication of FI981956A7 publication Critical patent/FI981956A7/fi
Publication of FI981956A0 publication Critical patent/FI981956A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI981956A 1991-07-17 1992-06-19 2-(4-hydroksipiperidino)-1-alkanolijohdannaisia verettömyyden vastaisia aineina FI981956A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73157791A 1991-07-17 1991-07-17
PCT/US1992/004973 WO1993002052A1 (en) 1991-07-17 1992-06-19 2-(4-hydroxypiperidino)-1-alkanol derivatives as antiischemic agents

Publications (3)

Publication Number Publication Date
FI981956L FI981956L (fi) 1998-09-11
FI981956A7 FI981956A7 (fi) 1998-09-11
FI981956A0 true FI981956A0 (fi) 1998-09-11

Family

ID=24940103

Family Applications (2)

Application Number Title Priority Date Filing Date
FI940192A FI940192A7 (fi) 1991-07-17 1992-06-19 2-(4-hydroksipiperidino)-1-alkonolijohdannaisia verettömyyden vastaisi na aineina
FI981956A FI981956A0 (fi) 1991-07-17 1992-06-19 2-(4-hydroksipiperidino)-1-alkanolijohdannaisia verettömyyden vastaisia aineina

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI940192A FI940192A7 (fi) 1991-07-17 1992-06-19 2-(4-hydroksipiperidino)-1-alkonolijohdannaisia verettömyyden vastaisi na aineina

Country Status (22)

Country Link
EP (1) EP0594729A1 (fi)
JP (1) JP2571904B2 (fi)
KR (1) KR0165003B1 (fi)
CN (1) CN1043759C (fi)
AU (1) AU655840B2 (fi)
BR (1) BR9206272A (fi)
CA (1) CA2113568A1 (fi)
CZ (1) CZ284133B6 (fi)
EG (1) EG20048A (fi)
FI (2) FI940192A7 (fi)
HU (1) HUT70528A (fi)
IE (1) IE922311A1 (fi)
IL (1) IL102473A (fi)
MX (1) MX9204190A (fi)
NO (1) NO180445C (fi)
NZ (1) NZ243580A (fi)
PL (1) PL169884B1 (fi)
PT (1) PT100689B (fi)
RU (1) RU2065859C1 (fi)
TW (1) TW201732B (fi)
WO (1) WO1993002052A1 (fi)
ZA (1) ZA925306B (fi)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5436255A (en) * 1992-07-23 1995-07-25 Pfizer Inc. Method of treating diseases susceptable to treatment by blocking NMDA-receptors
DE69309297T2 (de) * 1992-10-30 1997-07-03 Pfizer Neuroprotektive 3,4-dihydro-2(1h)-chinolone
US5498610A (en) * 1992-11-06 1996-03-12 Pfizer Inc. Neuroprotective indolone and related derivatives
US6978166B2 (en) 1994-10-07 2005-12-20 Saint Louis University System for use in displaying images of a body part
ZA9610741B (en) 1995-12-22 1997-06-24 Warner Lambert Co 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610745B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610738B (en) 1995-12-22 1997-06-24 Warner Lambert Co Subtype selective nmda receptor ligands and the use thereof
ZA9610736B (en) * 1995-12-22 1997-06-27 Warner Lambert Co 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists
CA2220649C (en) * 1996-12-03 2007-02-13 F. Hoffmann-La Roche Ag 4-hydroxy-piperidine derivatives
EP1182193A4 (en) * 1999-04-09 2002-09-11 Mochida Pharm Co Ltd REMEDIES FOR NEUROGENIC PAIN
TWI254043B (en) * 1999-06-08 2006-05-01 Hoffmann La Roche Ethanesulfonyl-piperidine derivatives having good affinity to N-methyl-D-aspartate (NMDA) receptor
US6476041B1 (en) 1999-10-29 2002-11-05 Merck & Co., Inc. 1,4 substituted piperidinyl NMDA/NR2B antagonists
US6369076B1 (en) 1999-10-29 2002-04-09 Merck & Co. Inc. 5-benzyl-octahydroindole and 6-benzyl-decahydroquinoline NMDA/NR2B antagonists
US6362196B1 (en) 1999-10-29 2002-03-26 Merck & Co., Inc. Method to treat pain utilizing benzimidazole NMDA/NR2B antagonists
US6495561B2 (en) 1999-10-29 2002-12-17 Merck & Co., Inc. 2-cyclohexyl imidazopyridine NMDA/NR2B antagonists
US6380205B1 (en) 1999-10-29 2002-04-30 Merck & Co., Inc. 2-cyclohexyl quinazoline NMDA/NR2B antagonists
US6291499B1 (en) 1999-10-29 2001-09-18 Merck & Co., Inc. 2-cyclohexyl benzimidazole NMDA/NR2B antagonists
US6489477B1 (en) 1999-10-29 2002-12-03 Merck & Co., Inc. 2-aza-bicyclo[2.2.2]octane NMDA/NR2B antigonists
US6432976B1 (en) 1999-10-29 2002-08-13 Merck & Co., Inc. 8-aza-bicyclo[3.2.1]octane NMDA/NR2B antagonists
US6316474B1 (en) 1999-10-29 2001-11-13 Merck & Co., Inc. 2-benzyl and 2-heteroaryl benzimidazole NMDA/NR2B antagonists
DE60210944T3 (de) 2001-02-23 2015-07-23 Merck Sharp & Dohme Corp. N-substituierte nichtaryl-heterocyclische nmda/nr2b antagonisten
JP2005511478A (ja) 2001-04-03 2005-04-28 メルク エンド カムパニー インコーポレーテッド N−置換非アリール複素環アミジル系nmda/nr2b拮抗薬
AU2003302416A1 (en) 2002-11-25 2004-06-18 Mochida Pharmaceutical Co., Ltd. Therapeutic agent for respiratory disease containing 4-hydroxypiperidine derivative as active ingredient
JP2007508288A (ja) * 2003-10-08 2007-04-05 ファイザー株式会社 縮合ラクタム化合物
TWI409289B (zh) 2010-09-02 2013-09-21 Taiwan Union Technology Corp 由氮氧雜環化合物所製得之聚合物之穩態溶液及其製法與用途
KR20230026449A (ko) * 2020-06-23 2023-02-24 바이오하벤 테라퓨틱스 리미티드 (1s)-1-페닐-2-피리딘-2-일레탄아민의 국소 제형

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH17194A (en) * 1980-03-06 1984-06-19 Otsuka Pharma Co Ltd Novel carbostyril derivatives,and pharmaceutical composition containing the same
FR2546166B1 (fr) * 1983-05-19 1985-10-25 Synthelabo Enantiomeres du erythro (benzyl-4 piperidino)-2 (hydroxy-4 ou benzyloxy-4 phenyl)-1 propanol, leur preparation et leur application en therapeutique
FR2640266B2 (fr) * 1988-07-12 1992-07-10 Synthelabo Derives de (hydroxy-1 piperidinyl-2 alkyl) indolones-2, quinoleinones-2, benzo(b)azepinones-2 et benzimidazolones-2, leur preparation et leur application en therapeutique
ES2098248T3 (es) * 1989-05-17 1997-05-01 Pfizer Derivados de 2-piperidino-1-alcanoles como agentes antiisquemicos.
AU642994B2 (en) * 1990-05-10 1993-11-04 Pfizer Inc. Neuroprotective indolone and related derivatives

Also Published As

Publication number Publication date
PT100689B (pt) 1999-06-30
FI940192L (fi) 1994-01-14
IL102473A (en) 1997-07-13
NO940144L (no) 1994-01-14
WO1993002052A1 (en) 1993-02-04
PL169884B1 (pl) 1996-09-30
CN1043759C (zh) 1999-06-23
CZ284133B6 (cs) 1998-08-12
IE922311A1 (en) 1993-01-27
FI940192A0 (fi) 1994-01-14
CN1068566A (zh) 1993-02-03
FI981956L (fi) 1998-09-11
FI981956A7 (fi) 1998-09-11
PT100689A (pt) 1993-10-29
NO180445B (no) 1997-01-13
MX9204190A (es) 1993-01-01
HU9400136D0 (en) 1994-05-30
AU655840B2 (en) 1995-01-12
FI940192A7 (fi) 1994-01-14
ZA925306B (en) 1994-01-17
JPH06504293A (ja) 1994-05-19
TW201732B (fi) 1993-03-11
CZ400892A3 (en) 1994-03-16
NO940144D0 (no) 1994-01-14
CA2113568A1 (en) 1993-02-04
HUT70528A (en) 1995-10-30
AU2322592A (en) 1993-02-23
NZ243580A (en) 1994-10-26
NO180445C (no) 1997-04-23
EP0594729A1 (en) 1994-05-04
RU2065859C1 (ru) 1996-08-27
IL102473A0 (en) 1993-01-14
JP2571904B2 (ja) 1997-01-16
EG20048A (en) 1997-03-27
KR0165003B1 (en) 1999-01-15
BR9206272A (pt) 1995-04-11

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