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FI935134A0 - Substituerade 3-aminokinuklidiner - Google Patents

Substituerade 3-aminokinuklidiner

Info

Publication number
FI935134A0
FI935134A0 FI935134A FI935134A FI935134A0 FI 935134 A0 FI935134 A0 FI 935134A0 FI 935134 A FI935134 A FI 935134A FI 935134 A FI935134 A FI 935134A FI 935134 A0 FI935134 A0 FI 935134A0
Authority
FI
Finland
Prior art keywords
compounds
aminoquinuclidine
substituent
disorders
antagonists
Prior art date
Application number
FI935134A
Other languages
English (en)
Finnish (fi)
Other versions
FI935134L (fi
FI935134A7 (fi
Inventor
Fumitaka Ito
Toshihide Kokura
Masami Nakane
Kunio Satake
Hiroaki Wakabayashi
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI935134L publication Critical patent/FI935134L/fi
Publication of FI935134A0 publication Critical patent/FI935134A0/fi
Publication of FI935134A7 publication Critical patent/FI935134A7/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Medicinal Preparation (AREA)
FI935134A 1991-05-22 1992-05-19 Substituoidut 3-aminokinuklidiinit FI935134A7 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP14682691 1991-05-22
PCT/US1992/004002 WO1992020676A1 (en) 1991-05-22 1992-05-19 Substituted 3-aminoquinuclidines

Publications (3)

Publication Number Publication Date
FI935134L FI935134L (fi) 1993-11-19
FI935134A0 true FI935134A0 (fi) 1993-11-19
FI935134A7 FI935134A7 (fi) 1993-11-19

Family

ID=15416402

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935134A FI935134A7 (fi) 1991-05-22 1992-05-19 Substituoidut 3-aminokinuklidiinit

Country Status (25)

Country Link
EP (1) EP0585328B1 (es)
KR (1) KR100246065B1 (es)
CN (1) CN1041827C (es)
AT (1) ATE211743T1 (es)
AU (1) AU658898B2 (es)
BR (1) BR9206044A (es)
CA (1) CA2109415C (es)
CZ (1) CZ247993A3 (es)
DE (2) DE69232334T2 (es)
DK (1) DK0585328T3 (es)
EG (1) EG20218A (es)
ES (1) ES2168260T3 (es)
FI (1) FI935134A7 (es)
HU (1) HUT65771A (es)
IE (1) IE921662A1 (es)
IL (1) IL101960A (es)
MX (1) MX9202449A (es)
NO (1) NO305173B1 (es)
NZ (2) NZ242880A (es)
PL (4) PL170513B1 (es)
PT (1) PT100514B (es)
RU (1) RU2092486C1 (es)
UA (1) UA26401C2 (es)
WO (1) WO1992020676A1 (es)
ZA (1) ZA923773B (es)

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JP2656702B2 (ja) * 1992-03-23 1997-09-24 ファイザー製薬株式会社 ペプチド性キヌクリジン
ATE208376T1 (de) * 1992-08-19 2001-11-15 Pfizer Substituierte benzylamin-stickstoff enthaltende nichtaromatische heterocyclen
JP2656699B2 (ja) * 1992-10-21 1997-09-24 ファイザー製薬株式会社 置換ベンジルアミノキヌクリジン
US5837711A (en) * 1992-10-28 1998-11-17 Pfizer Inc. Substituted quinuclidines as substance P antagonists
JP2656700B2 (ja) * 1992-10-28 1997-09-24 ファイザー製薬株式会社 置換キヌクリジン誘導体
JP2722279B2 (ja) * 1992-12-10 1998-03-04 ファイザー・インク． アミノメチレンで置換した非芳香族複素環式化合物及びサブスタンスｐのアンタゴニストとしての使用
IL109646A0 (en) * 1993-05-19 1994-08-26 Pfizer Heteroatom substituted alkyl benzylamino-quinuclidines
JP2822274B2 (ja) * 1993-05-19 1998-11-11 ファイザー製薬株式会社 Ｐ物質拮抗剤としてのヘテロ原子置換アルキルベンジルアミノキヌクリジン類
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ATE171945T1 (de) 1993-07-15 1998-10-15 Pfizer Benzyloxychinuclidine als substanz p antagonisten
DK0719253T3 (da) * 1993-09-17 2004-07-26 Pfizer 3-amino-5-carboxy-substituerede piperidiner og 3-amino-4-carboxy-substituerede pyrrolidiner som tachykininantagonister
US6083943A (en) * 1993-09-17 2000-07-04 Pfizer Inc Substituted azaheterocyclecarboxylic acid
EP0653208A3 (en) * 1993-11-17 1995-10-11 Pfizer Substance P antagonists for the treatment or prevention of sunburn.
EP0659409A3 (en) * 1993-11-23 1995-08-09 Pfizer Substance P antagonists for the inhibition of angiogenesis.
EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
PE8798A1 (es) * 1995-07-17 1998-03-02 Pfizer Procedimiento de separacion de los enantiomeros del 1-azabiciclo[2.2.2] octan-3-amina, 2-(difenilmetil) -n- [[2-metoxi-5-(1-metiletil) fenil] metil]
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FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
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Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX18467A (es) * 1988-11-23 1993-07-01 Pfizer Agentes terapeuticos de quinuclidinas

Also Published As

Publication number Publication date
ES2168260T3 (es) 2002-06-16
DE69232334T2 (de) 2002-11-14
EP0585328A1 (en) 1994-03-09
NO305173B1 (no) 1999-04-12
RU2092486C1 (ru) 1997-10-10
EG20218A (en) 1997-11-30
PT100514A (pt) 1993-09-30
WO1992020676A1 (en) 1992-11-26
NO934195L (no) 1993-11-19
NO934195D0 (no) 1993-11-19
CA2109415A1 (en) 1992-11-23
FI935134L (fi) 1993-11-19
IL101960A0 (en) 1994-04-12
BR9206044A (pt) 1995-03-01
ZA923773B (en) 1993-11-22
KR100246065B1 (en) 2000-04-01
PL172069B1 (pl) 1997-07-31
DK0585328T3 (da) 2002-02-11
ATE211743T1 (de) 2002-01-15
PL170525B1 (en) 1996-12-31
CZ247993A3 (en) 1994-07-13
EP0585328B1 (en) 2002-01-09
NZ272941A (en) 1997-05-26
DE9290057U1 (de) 1994-01-05
PT100514B (pt) 1999-06-30
CA2109415C (en) 1998-12-29
UA26401C2 (uk) 1999-08-30
PL171921B1 (pl) 1997-06-30
CN1068571A (zh) 1993-02-03
HUT65771A (en) 1994-07-28
AU658898B2 (en) 1995-05-04
NZ242880A (en) 1995-10-26
PL170513B1 (en) 1996-12-31
HU9303307D0 (en) 1994-03-28
IL101960A (en) 1999-03-12
CN1041827C (zh) 1999-01-27
DE69232334D1 (de) 2002-02-14
AU1927592A (en) 1992-12-30
FI935134A7 (fi) 1993-11-19
IE921662A1 (en) 1992-12-02
MX9202449A (es) 1993-03-01

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