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FI913137L - Menetelmä uusien terapeuttisesti käyttökelpoisten 4"-deoksi-4"-epi-metyyliaminoavermekitiinisuolojen valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten 4"-deoksi-4"-epi-metyyliaminoavermekitiinisuolojen valmistamiseksi Download PDF

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Publication number
FI913137L
FI913137L FI913137A FI913137A FI913137L FI 913137 L FI913137 L FI 913137L FI 913137 A FI913137 A FI 913137A FI 913137 A FI913137 A FI 913137A FI 913137 L FI913137 L FI 913137L
Authority
FI
Finland
Prior art keywords
methylaminoavermectin
epi
deoxy
salts
therapeutically useful
Prior art date
Application number
FI913137A
Other languages
English (en)
Swedish (sv)
Other versions
FI97890C (fi
FI913137A0 (fi
FI97890B (fi
Inventor
Raymond Cvetovich
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of FI913137A0 publication Critical patent/FI913137A0/fi
Publication of FI913137L publication Critical patent/FI913137L/fi
Application granted granted Critical
Publication of FI97890B publication Critical patent/FI97890B/fi
Publication of FI97890C publication Critical patent/FI97890C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Silicon Polymers (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Fodder In General (AREA)
  • Steroid Compounds (AREA)
FI913137A 1990-06-28 1991-06-27 Menetelmä uusien terapeuttisesti käyttökelpoisten 4"-deoksi-4"-epi-metyyliaminoavermekitiinisuolojen valmistamiseksi FI97890C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54522990A 1990-06-28 1990-06-28
US54522990 1990-06-28

Publications (4)

Publication Number Publication Date
FI913137A0 FI913137A0 (fi) 1991-06-27
FI913137L true FI913137L (fi) 1991-12-29
FI97890B FI97890B (fi) 1996-11-29
FI97890C FI97890C (fi) 1997-03-10

Family

ID=24175383

Family Applications (1)

Application Number Title Priority Date Filing Date
FI913137A FI97890C (fi) 1990-06-28 1991-06-27 Menetelmä uusien terapeuttisesti käyttökelpoisten 4"-deoksi-4"-epi-metyyliaminoavermekitiinisuolojen valmistamiseksi

Country Status (21)

Country Link
US (1) US5288710A (fi)
EP (1) EP0465121B1 (fi)
JP (1) JPH0822870B2 (fi)
KR (1) KR100224292B1 (fi)
AT (1) ATE134377T1 (fi)
AU (1) AU641777B2 (fi)
CA (1) CA2045864C (fi)
CY (1) CY1949A (fi)
DE (1) DE69117223T2 (fi)
DK (1) DK0465121T3 (fi)
ES (1) ES2084110T3 (fi)
FI (1) FI97890C (fi)
GR (1) GR3019067T3 (fi)
HK (1) HK157096A (fi)
IE (1) IE71175B1 (fi)
IL (1) IL98599A (fi)
LV (1) LV5740B4 (fi)
NO (2) NO178339C (fi)
NZ (1) NZ238705A (fi)
PT (1) PT98117B (fi)
ZA (1) ZA914961B (fi)

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JP4701538B2 (ja) 2001-05-21 2011-06-15 住友化学株式会社 農業害虫防除剤組成物
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DE10203688A1 (de) 2002-01-31 2003-08-07 Bayer Cropscience Ag Synergistische insektizide Mischungen
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GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
CN101065352A (zh) 2004-09-23 2007-10-31 先灵-普劳有限公司 使用新的三氟甲磺酰苯胺肟醚衍生物控制动物中的寄生虫
DE602005017419D1 (de) * 2004-11-19 2009-12-10 Schering Plough Ltd Kontrolle von parasiten bei tieren mittels verwendung von parasitiziden 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitril-derivaten
US20060281695A1 (en) * 2005-06-09 2006-12-14 Schering-Plough Animal Health Corporation Control of parasites in animals by N-[(phenyloxy)phenyl]-1,1,1-trifluoromethanesulfonamide and N-[(phenylsulfanyl)phenyl]-1,1,1-trifluoromethanesulfonamide derivatives
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
TWI422328B (zh) 2006-06-19 2014-01-11 Univ California 結合有殺線蟲之種子塗覆物的生物控制劑
FR2906469B1 (fr) * 2006-09-28 2008-11-28 Galderma Sa Utilisation de composes de la famille des avermectines pour le traitement de desordres dermatologiques chez l'homme
US8084643B2 (en) * 2006-12-13 2011-12-27 Intervet Inc. Water-soluble prodrugs of florfenicol and its analogs
EP2102154A1 (en) * 2006-12-13 2009-09-23 Schering-Plough Ltd. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
DE102007002872A1 (de) 2007-01-15 2008-07-17 Alpha-Biocare Gmbh Verwendung von Avermectin-Derivaten zur Behandlung gegen Parasiten von Fischen
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
EP2957284B1 (en) 2007-06-27 2018-01-17 E. I. du Pont de Nemours and Company Animal pest control method
TWI556741B (zh) 2007-08-17 2016-11-11 英特威特國際股份有限公司 異唑啉組成物及其作為抗寄生蟲藥上的應用
TWI401023B (zh) 2008-02-06 2013-07-11 Du Pont 中離子農藥
JP2011529895A (ja) * 2008-07-30 2011-12-15 インターベツト・インターナシヨナル・ベー・ベー フロルフェニコール中間体として有用なオキサゾリン保護アミノジオール化合物を調製する方法
CN102355891A (zh) 2009-03-17 2012-02-15 英特威国际有限公司 大环内酯药物递送系统
CN102574815A (zh) 2009-08-05 2012-07-11 杜邦公司 介离子杀虫剂
KR20120050467A (ko) 2009-08-05 2012-05-18 이 아이 듀폰 디 네모아 앤드 캄파니 메소이온성 살충제
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
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HUE058291T2 (hu) 2010-12-27 2022-07-28 Intervet Int Bv Topikális lokalizált izoxazolin formuláció
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CN107344954B (zh) * 2017-08-07 2020-08-11 河北蓝泰化工科技有限公司 增效型甲氨基阿维菌素b1或b2的盐及制备方法和应用
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CN108864230B (zh) * 2018-07-26 2021-05-14 河北威远生物化工有限公司 一种有机磷基团取代的阿维菌素衍生物及其制备方法和应用

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Also Published As

Publication number Publication date
FI97890C (fi) 1997-03-10
FI913137A0 (fi) 1991-06-27
DE69117223T2 (de) 1996-09-12
KR920000781A (ko) 1992-01-29
LV5740A4 (lv) 1996-08-20
GR3019067T3 (en) 1996-05-31
NO178339C (no) 1996-03-06
ATE134377T1 (de) 1996-03-15
JPH05306294A (ja) 1993-11-19
CA2045864A1 (en) 1991-12-29
NO178339B (no) 1995-11-27
ZA914961B (en) 1992-07-29
IE71175B1 (en) 1997-01-29
NO2001007I2 (no) 2007-02-26
KR100224292B1 (ko) 1999-10-15
DK0465121T3 (da) 1996-03-18
DE69117223D1 (de) 1996-03-28
AU641777B2 (en) 1993-09-30
PT98117B (pt) 1998-12-31
NZ238705A (en) 1993-07-27
EP0465121A1 (en) 1992-01-08
IE912251A1 (en) 1992-01-01
HK157096A (en) 1996-08-23
NO912535D0 (no) 1991-06-27
EP0465121B1 (en) 1996-02-21
LV5740B4 (lv) 1997-12-20
IL98599A0 (en) 1992-07-15
CY1949A (en) 1991-06-27
ES2084110T3 (es) 1996-05-01
PT98117A (pt) 1993-10-29
NO912535L (no) 1991-12-30
FI97890B (fi) 1996-11-29
US5288710A (en) 1994-02-22
CA2045864C (en) 2001-11-27
IL98599A (en) 1995-06-29
AU7939291A (en) 1992-01-02
JPH0822870B2 (ja) 1996-03-06

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Owner name: MERCK & CO., INC.

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