FI911285A7 - Antipsykoottisia bisyklisiä 4-/4-(3-bentsisotiatsolyyli)-1-piperatsiny yli/butyylisiltaimidejä - Google Patents

Antipsykoottisia bisyklisiä 4-/4-(3-bentsisotiatsolyyli)-1-piperatsiny yli/butyylisiltaimidejä Download PDF

Info

Publication number: FI911285A7
Authority: FI; Finland
Prior art keywords: sylimides; benzisothiazolyl; antipsychotic; piperazinyl; bicyclic
Prior art date: 1988-09-16

Application number

FI911285A

Other languages

English (en)

Swedish (sv)

Other versions

FI911285A0 (fi

Inventor

Iii John A Lowe

Gene Michael Bright

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-09-16

Filing date

1988-09-16

Publication date

1991-03-15

1988-09-16 Application filed by Pfizer filed Critical Pfizer

1991-03-15 Publication of FI911285A0 publication Critical patent/FI911285A0/fi

1991-03-15 Publication of FI911285A7 publication Critical patent/FI911285A7/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Biomedical Technology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Psychiatry (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

FI911285A 1988-09-16 1988-09-16 Antipsykoottisia bisyklisiä 4-/4-(3-bentsisotiatsolyyli)-1-piperatsiny yli/butyylisiltaimidejä FI911285A7 (fi)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US1988/003230 WO1990002552A1 (en)	1988-09-16	1988-09-16	Antipsychotic 4-[4-(3-benzisothiazolyl)-1-piperazinyl]butyl bridged bicyclic imides

Publications (2)

Publication Number	Publication Date
FI911285A0 FI911285A0 (fi)	1991-03-15
FI911285A7 true FI911285A7 (fi)	1991-03-15

Family

ID=22208913

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI911285A FI911285A7 (fi)	1988-09-16	1988-09-16	Antipsykoottisia bisyklisiä 4-/4-(3-bentsisotiatsolyyli)-1-piperatsiny yli/butyylisiltaimidejä

Country Status (20)

Country	Link
US (1)	US5077295A (fi)
EP (1)	EP0364091B1 (fi)
JP (1)	JPH0631231B2 (fi)
KR (1)	KR930002568B1 (fi)
AT (1)	ATE92063T1 (fi)
AU (1)	AU607354B2 (fi)
CA (1)	CA1339314C (fi)
DE (1)	DE68907845T2 (fi)
DK (1)	DK175200B1 (fi)
ES (1)	ES2058542T3 (fi)
FI (1)	FI911285A7 (fi)
HU (1)	HUT61760A (fi)
IE (1)	IE61413B1 (fi)
IL (1)	IL91552A (fi)
MY (1)	MY104207A (fi)
NO (1)	NO911042L (fi)
NZ (1)	NZ230672A (fi)
PT (1)	PT91703B (fi)
WO (1)	WO1990002552A1 (fi)
ZA (1)	ZA897049B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5235283A (en) *	1991-02-07	1993-08-10	Siemens Aktiengesellschaft	Gradient coil system for a nuclear magnetic resonance tomography apparatus which reduces acoustic noise
PT790236E (pt) *	1996-02-13	2004-04-30	Pfizer	Pro-farmacos de 5-(2-(4-(1,2-benzisotiazol-3-il)-1-piperazinil)-etil-6-cloro-1,3-di-hidro-2h-indol-2-ona
US6084097A (en) *	1997-10-20	2000-07-04	Council Of Scientific & Industrial Research	Methods for preparing 1-[4-arylpiperazin-1-yl]-3-[2-oxopyrrolidin/piperidin-1-yl] propanes
EP3610890A1 (en)	2012-11-14	2020-02-19	The Johns Hopkins University	Methods and compositions for treating schizophrenia

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE759371A (fr) *	1969-11-24	1971-05-24	Bristol Myers Co	Azaspirodecanediones heterocycliques et procedes pour leur preparation
US4411901A (en) *	1981-12-23	1983-10-25	Mead Johnson & Company	Benzisothiazole and benzisoxazole piperazine derivatives
US4507303A (en) *	1981-12-22	1985-03-26	Sumitomo Chemical Company, Limited	Succinimide derivatives, compositions and method of use
US4452799A (en) *	1981-12-23	1984-06-05	Mead Johnson & Company	Benzisothiazole and benzisoxazole piperazine derivatives
US4423049A (en) *	1981-12-28	1983-12-27	Mead Johnson & Company	2-[4-[(4,4-Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyrimidines
JPS5995267A (ja) *	1982-11-25	1984-06-01	Eisai Co Ltd	カルボン酸イミド誘導体およびその製造方法
US4524206A (en) *	1983-09-12	1985-06-18	Mead Johnson & Company	1-Heteroaryl-4-(2,5-pyrrolidinedion-1-yl)alkyl)piperazine derivatives
US4562255A (en) *	1984-03-30	1985-12-31	American Home Products Corporation	Substituted bi-alicyclic imides
US4585773A (en) *	1984-07-11	1986-04-29	Bristol-Myers Company	Isoindolinyl-alkyl-piperazines
US4590196A (en) *	1984-08-23	1986-05-20	Bristol-Myers Company	Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
JPH0625181B2 (ja) *	1985-03-27	1994-04-06	住友製薬株式会社	新規なイミド誘導体
US4656173A (en) *	1985-04-24	1987-04-07	Bristol-Myers Company	Antipsychotic benzisothiazole S-oxide compound
HUT43600A (en) *	1985-06-22	1987-11-30	Sandoz Ag	Process for production of new thiazole derivatives and medical compound containing those
US4732984A (en) *	1985-10-17	1988-03-22	American Home Products Corporation	Piperazinoisothiazolones with psychotropic activity
JPS6310786A (ja) *	1986-07-01	1988-01-18	Sumitomo Pharmaceut Co Ltd	新規イミド誘導体およびその製造法
JPS6310760A (ja) *	1986-07-01	1988-01-18	Sumitomo Pharmaceut Co Ltd	イミド誘導体の新規製造法
DD263531A5 (de) *	1986-10-21	1989-01-04	��@��Kk��	Verfahren zur herstellung von verbrueckten bicyclischen imidverbindungen
US4748240A (en) *	1987-04-03	1988-05-31	American Home Products Corporation	Psychotropic bicyclic imides
US4883795A (en) *	1988-01-22	1989-11-28	Pfizer Inc.	Piperazinyl-heterocyclic compounds
JPH0310760A (ja) *	1989-06-09	1991-01-18	Nippon Spindle Mfg Co Ltd	結晶質脆性材料切断用ワイヤソー

1988
- 1988-09-16 WO PCT/US1988/003230 patent/WO1990002552A1/en not_active Ceased
- 1988-09-16 FI FI911285A patent/FI911285A7/fi not_active Application Discontinuation
- 1988-09-16 HU HU892131A patent/HUT61760A/hu unknown
- 1988-09-16 US US07/659,407 patent/US5077295A/en not_active Expired - Lifetime
1989
- 1989-08-22 EP EP89308479A patent/EP0364091B1/en not_active Expired - Lifetime
- 1989-08-22 AT AT89308479T patent/ATE92063T1/de not_active IP Right Cessation
- 1989-08-22 DE DE89308479T patent/DE68907845T2/de not_active Expired - Fee Related
- 1989-08-22 ES ES89308479T patent/ES2058542T3/es not_active Expired - Lifetime
- 1989-09-07 IL IL9155289A patent/IL91552A/en not_active IP Right Cessation
- 1989-09-12 KR KR1019890013262A patent/KR930002568B1/ko not_active Expired - Fee Related
- 1989-09-13 JP JP1238347A patent/JPH0631231B2/ja not_active Expired - Fee Related
- 1989-09-13 PT PT91703A patent/PT91703B/pt not_active IP Right Cessation
- 1989-09-14 MY MYPI89001253A patent/MY104207A/en unknown
- 1989-09-14 CA CA000611376A patent/CA1339314C/en not_active Expired - Fee Related
- 1989-09-15 NZ NZ230672A patent/NZ230672A/en unknown
- 1989-09-15 AU AU41506/89A patent/AU607354B2/en not_active Ceased
- 1989-09-15 DK DK198904563A patent/DK175200B1/da not_active IP Right Cessation
- 1989-09-15 ZA ZA897049A patent/ZA897049B/xx unknown
- 1989-09-15 IE IE294989A patent/IE61413B1/en not_active IP Right Cessation
1991
- 1991-03-15 NO NO91911042A patent/NO911042L/no unknown

Also Published As

Publication number	Publication date
DK175200B1 (da)	2004-07-05
US5077295A (en)	1991-12-31
JPH02121986A (ja)	1990-05-09
KR900004730A (ko)	1990-04-12
NO911042L (no)	1991-05-15
PT91703B (pt)	1995-07-18
EP0364091A1 (en)	1990-04-18
FI911285A0 (fi)	1991-03-15
ZA897049B (en)	1991-04-24
NO911042D0 (no)	1991-03-15
IL91552A0 (en)	1990-04-29
EP0364091B1 (en)	1993-07-28
PT91703A (pt)	1990-03-30
CA1339314C (en)	1997-08-19
DE68907845D1 (de)	1993-09-02
AU4150689A (en)	1990-03-22
NZ230672A (en)	1990-12-21
KR930002568B1 (ko)	1993-04-03
DK456389D0 (da)	1989-09-15
DE68907845T2 (de)	1993-11-11
IE61413B1 (en)	1994-11-02
DK456389A (da)	1990-03-17
JPH0631231B2 (ja)	1994-04-27
HUT61760A (en)	1993-03-01
ATE92063T1 (de)	1993-08-15
IL91552A (en)	1994-02-27
IE892949L (en)	1990-03-16
MY104207A (en)	1994-02-28
AU607354B2 (en)	1991-02-28
ES2058542T3 (es)	1994-11-01
WO1990002552A1 (en)	1990-03-22

Publication	Publication Date	Title
MA20323A1 (fr)	1985-10-01	Nouvelles 4-(heterocycle bicyclique methyle et -hebbero)-piperidines
NL980022I2 (nl)	1998-11-02	Dibenzothiazepine.
DK247789A (da)	1989-11-24	Piperazinderivater
NO871909D0 (no)	1987-05-07	Fekal inkontinenspose.
DK93887D0 (da)	1987-02-24	Heterocycliske forbindelser
ATA55388A (de)	1990-12-15	Kapazitiver naeherungsgeber
DK292986D0 (da)	1986-06-20	Thiazoler
FI892558L (fi)	1989-05-25	I laoga temperaturer haerdbar cementkomposition.
DE3767816D1 (de)	1991-03-07	1-acylsubstituierte piperidinderivate.
DK575386D0 (da)	1986-11-28	Thiazolderivater
FI871632A0 (fi)	1987-04-14	Heterocykliska karboxamider.
DK674487D0 (da)	1987-12-21	Piperidinderivater
DK287688D0 (da)	1988-05-25	Heterocycliske forbindelser
FI932173L (fi)	1993-05-13	4-(1,2-benzisoxazolyl)piperidinantipsykotiska medel
DK365687A (da)	1988-01-16	Glaskeramiske dielektriske materialer
DK429887A (da)	1988-02-19	Vandigt opvaskemiddel
AT379260B (de)	1985-12-10	Kapazitiver schalter
FI911285A7 (fi)	1991-03-15	Antipsykoottisia bisyklisiä 4-/4-(3-bentsisotiatsolyyli)-1-piperatsiny yli/butyylisiltaimidejä
DK91890A (da)	1990-10-16	Piperazin-derivater
DK499987D0 (da)	1987-09-23	Heterocycliske forbindelser
FI872566A7 (fi)	1987-12-10	Fusionerade heterocykliska imidazofoereningar.
FI861668L (fi)	1986-10-25	Antipsykotisk benzisotiazol-5-oxidfoerening.
DK0395174T3 (da)	1995-02-06	Thiazolderivater
AT379261B (de)	1985-12-10	Kapazitiver schalter
DK365587A (da)	1988-01-16	Glaskeramiske dielektriske materialer

Legal Events

Date	Code	Title	Description
1995-07-24	FD	Application lapsed