[go: up one dir, main page]

FI910303A7 - Tiatsolidinin johdannaiset, joilla on verenpainetta alentava vaikutus ja niiden terapeuttinen käyttö - Google Patents

Tiatsolidinin johdannaiset, joilla on verenpainetta alentava vaikutus ja niiden terapeuttinen käyttö Download PDF

Info

Publication number
FI910303A7
FI910303A7 FI910303A FI910303A FI910303A7 FI 910303 A7 FI910303 A7 FI 910303A7 FI 910303 A FI910303 A FI 910303A FI 910303 A FI910303 A FI 910303A FI 910303 A7 FI910303 A7 FI 910303A7
Authority
FI
Finland
Prior art keywords
therapeutic use
antihypertensive activity
thiazolidine derivatives
thiazolidine
derivatives
Prior art date
Application number
FI910303A
Other languages
English (en)
Swedish (sv)
Other versions
FI910303A0 (fi
FI910303L (fi
Inventor
Hiroyuki Koike
Takao Yoshioka
Hiroyoshi Horikoshi
Toshihiko Fujiwara
Shinji Yoshioka
Hiroshi Nishino
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of FI910303A0 publication Critical patent/FI910303A0/fi
Publication of FI910303A7 publication Critical patent/FI910303A7/fi
Publication of FI910303L publication Critical patent/FI910303L/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyrrole Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI910303A 1990-01-22 1991-01-21 Derivat av tiazolidin med blodtrycksnedsaenkande effekt och terapeutisk anvaendning av dessa. FI910303L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1232190 1990-01-22

Publications (3)

Publication Number Publication Date
FI910303A0 FI910303A0 (fi) 1991-01-21
FI910303A7 true FI910303A7 (fi) 1991-07-23
FI910303L FI910303L (fi) 1991-07-23

Family

ID=11802053

Family Applications (1)

Application Number Title Priority Date Filing Date
FI910303A FI910303L (fi) 1990-01-22 1991-01-21 Derivat av tiazolidin med blodtrycksnedsaenkande effekt och terapeutisk anvaendning av dessa.

Country Status (11)

Country Link
US (1) US5614542A (fi)
EP (1) EP0439321B1 (fi)
JP (1) JP2826379B2 (fi)
KR (1) KR0163052B1 (fi)
AT (1) ATE119773T1 (fi)
AU (1) AU637182B2 (fi)
CA (1) CA2034616A1 (fi)
DE (1) DE69108067T2 (fi)
DK (1) DK0439321T3 (fi)
ES (1) ES2072536T3 (fi)
FI (1) FI910303L (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5175179A (en) * 1991-09-25 1992-12-29 Pfizer Inc. Method for treating hypertension
CZ283339B6 (cs) * 1993-09-15 1998-03-18 Sankyo Company Limited Použití thiazolidinových derivátů pro výrobu léčivého přípravku pro léčení zhoršené tolerance glukosy pro zabránění nebo zpoždění nástupu diabetes mellitus nezávislé na inzulinu
CZ293016B6 (cs) * 1995-06-01 2004-01-14 Sankyo Company Limited Benzimidazolové deriváty a farmaceutické prostředky s jejich obsahem
ZA973848B (en) * 1996-05-06 1997-12-02 Reddy Research Foundation Novel heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them.
US5801173A (en) * 1996-05-06 1998-09-01 Dr. Reddy's Research Foundation Heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
US5889025A (en) * 1996-05-06 1999-03-30 Reddy's Research Foundation Antidiabetic compounds having hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
US5919782A (en) * 1996-05-06 1999-07-06 Dr. Reddy's Research Foundation Heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
CA2258949C (en) 1996-07-01 2008-05-06 Dr. Reddy's Research Foundation Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
US6372750B2 (en) 1996-07-01 2002-04-16 Dr. Reddy's Research Foundation Heterocyclic compounds, process for their preparation and pharmaceutical compounds containing them and their use in the treatment of diabetes and related diseases
US5885997A (en) * 1996-07-01 1999-03-23 Dr. Reddy's Research Foundation Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
US6114526A (en) 1996-07-01 2000-09-05 Dr. Reddy's Research Foundation Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
USRE39266E1 (en) * 1996-07-01 2006-09-05 Dr. Reddy's Laboratories, Limited Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
TW577875B (en) * 1997-01-31 2004-03-01 Shionogi & Co Pyrrolidine derivatives with inhibitory activity for phospholipase A2
EP0981526B1 (en) * 1997-05-02 2004-02-25 Dr. Reddy's Laboratories Ltd. Novel antidiabetic compounds having hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6051189A (ja) * 1983-08-30 1985-03-22 Sankyo Co Ltd チアゾリジン誘導体およびその製造法
DK173350B1 (da) * 1985-02-26 2000-08-07 Sankyo Co Thiazolidinderivater, deres fremstilling og farmaceutisk paæparat indeholdende dem
US4873255A (en) * 1987-02-04 1989-10-10 Sankyo Company Limited Thiazolidinone derivatives, their preparation and their use
US4933355A (en) * 1988-04-14 1990-06-12 Sankyo Company Limited Thiazole derivatives, their preparation and their use in the treatment of diabetes complications
DE3823533A1 (de) * 1988-07-12 1990-02-08 Beiersdorf Ag Substituierte 4-heterocyclyl-2h-benzo(b)pyrane, verfahren und 4-hydroxy-3-brom-, 3,4-oxiranyl-3,4-dehydro-2h-benzo(b)pyrane als zwischenprodukte zu ihrer herstellung, sowie sie enthaltende pharmazeutsche praeparate
US5053420A (en) * 1989-10-13 1991-10-01 Pershadsingh Harrihar A Thiazolidine derivatives for the treatment of hypertension

Also Published As

Publication number Publication date
HK1006284A1 (en) 1999-02-19
FI910303A0 (fi) 1991-01-21
ES2072536T3 (es) 1995-07-16
AU637182B2 (en) 1993-05-20
AU6948091A (en) 1991-07-25
EP0439321A2 (en) 1991-07-31
DE69108067D1 (de) 1995-04-20
KR910014119A (ko) 1991-08-31
ATE119773T1 (de) 1995-04-15
CA2034616A1 (en) 1991-07-23
FI910303L (fi) 1991-07-23
EP0439321A3 (en) 1992-04-01
DE69108067T2 (de) 1995-11-02
KR0163052B1 (ko) 1998-12-01
DK0439321T3 (da) 1995-07-24
EP0439321B1 (en) 1995-03-15
US5614542A (en) 1997-03-25
JP2826379B2 (ja) 1998-11-18
JPH03251530A (ja) 1991-11-11

Similar Documents

Publication Publication Date Title
FI955248A7 (fi) 1-Bifenyylimetyyli-imitdatsolin johdannaiset, niiden valmistus ja terapeuttinen käyttö
FI934426A7 (fi) Tiatsolidiinidionijohdokset, niiden valmistus ja käyttö
NO910723L (no) Karbapenemderivater med antibiotisk aktivitet, samt fremstilling og anvendelse derav.
NL300038I2 (nl) Thiazolidinedionderivaten, alsmede bereiding en toepassing daarvan.
FI940904A7 (fi) Oksatsolidiinidionijohdannaiset, niiden valmistus ja käyttö
FI951370A7 (fi) Tiatsolidinin ja oksatsolidinin johdannaiset, niiden valmistus ja lääkinnällinen käyttö
NO924401D0 (no) 2-substituerte sakkarinderivater med protedytisk enzyminhiberende aktivitet
FI895689A7 (fi) Substituoituja tiatsoleja ja niiden käyttö fungisideina
FI951731A7 (fi) Heterosykliset yhdisteet, joilla on sokeritautia vastustava vaikutus, niiden valmistus ja käyttö
FI945281A7 (fi) Heterosykliset yhdisteet, niiden valmistus ja käyttö
FI935887L (fi) Tiatzolidiinidionijohdannaiset, niiden valmistus ja käyttö
IT8919730A0 (it) Derivati xantinici ad attivita' broncodilatatrice e loro applicazioni terapeutiche.
FI914611A7 (fi) 2-aminopyrimidiini-4-karboksamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI915099A7 (fi) Tienoimidatsolijohdannaiset, niiden valmistus ja käyttö
FI910303A7 (fi) Tiatsolidinin johdannaiset, joilla on verenpainetta alentava vaikutus ja niiden terapeuttinen käyttö
FI892344A7 (fi) 6-fenyyli-3-piperatsinyylialkyyli-1H,3H-pyrimidiini-2,4-dionin johdannaisia, niiden valmistus ja niiden terapeuttinen käyttö
FI941068A7 (fi) Bentsoksatsiinijohdannaiset, niiden valmistus ja terapeuttinen käyttö
MX9203459A (es) Nuevos derivados de 2'-halometilideno, 2'-etenilideno y 2'-etinilcitidina, uridina y guanosina.
FI922982A7 (fi) 2-aminopyrimidiini-4-karboksamidijohdannaisia, niiden valmistus ja niiden terapeuttinen käyttö
FI934221A7 (fi) Piperidiinijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI923458A7 (fi) 4,5-sykloalkano-3-bentsatsepin-7-olijohdannaiset ja niiden käyttö
FI920663A7 (fi) Polyhydroksisyklopentaanin johdannaiset, niiden valmistus ja terapeuttinen käyttö
FI921814A7 (fi) 2-aminopyrimidiini-4-karboksiamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI895286A7 (fi) Fenyylioksipropanoliamineja, niiden valmistus ja terapeuttinen käyttö
FI894758A7 (fi) 3-Aryylioksimetyyli-kefalosporiinin johdannaiset, niiden valmistus ja lääkinnällinen käyttö

Legal Events

Date Code Title Description
FD Application lapsed