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FI900801A0 - Melantonianaloger. - Google Patents

Melantonianaloger.

Info

Publication number
FI900801A0
FI900801A0 FI900801A FI900801A FI900801A0 FI 900801 A0 FI900801 A0 FI 900801A0 FI 900801 A FI900801 A FI 900801A FI 900801 A FI900801 A FI 900801A FI 900801 A0 FI900801 A0 FI 900801A0
Authority
FI
Finland
Prior art keywords
melantonianaloger
Prior art date
Application number
FI900801A
Other languages
English (en)
Other versions
FI900801A7 (fi
Inventor
Margarita L Dubocovich
James V Peck
Atef A Helmy
Vithal J Rajadhyaksha
Original Assignee
Nelson Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nelson Res & Dev filed Critical Nelson Res & Dev
Publication of FI900801A7 publication Critical patent/FI900801A7/fi
Publication of FI900801A0 publication Critical patent/FI900801A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Saccharide Compounds (AREA)
FI900801A 1987-08-17 1988-05-20 Melantonianaloger. FI900801A0 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8606287A 1987-08-17 1987-08-17
US8629087A 1987-08-17 1987-08-17
PCT/US1988/001859 WO1989001472A1 (en) 1987-08-17 1988-05-20 Melatonin analogues

Publications (2)

Publication Number Publication Date
FI900801A7 FI900801A7 (fi) 1990-02-16
FI900801A0 true FI900801A0 (fi) 1990-02-16

Family

ID=26774333

Family Applications (1)

Application Number Title Priority Date Filing Date
FI900801A FI900801A0 (fi) 1987-08-17 1988-05-20 Melantonianaloger.

Country Status (7)

Country Link
EP (1) EP0375726A4 (fi)
KR (1) KR910006124B1 (fi)
AU (1) AU616907B2 (fi)
DK (1) DK42490A (fi)
FI (1) FI900801A0 (fi)
NO (1) NO173732C (fi)
WO (1) WO1989001472A1 (fi)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK108022C (da) * 1964-10-15 1967-07-31 Svend Anton Hansen Wexel Fremgangsmåde til hel eller delvis udskæring af rygbenet af opskårne slagtekroppe, navnlig grisekroppe, og anlæg til udførelse af denne fremgangsmåde.
AU644367B2 (en) * 1989-05-17 1993-12-09 Applied Medical Research Ltd Use of melatonin derivatives for effecting contraception
US5071875A (en) * 1989-09-25 1991-12-10 Northwestern University Substituted 2-amidotetralins as melatonin agonists and antagonists
IT1251544B (it) * 1991-05-13 1995-05-17 Gabriele Biella Composizioni farmaceutiche attive nella terapia dei disturbi del sonno comprendenti melatonina o un suo derivato in associazione con un derivato benzodiazepinico
FR2680366B1 (fr) * 1991-08-13 1995-01-20 Adir Nouveaux derives d'arylethylamines, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
JPH07503232A (ja) * 1991-10-18 1995-04-06 アルザ・コーポレーション メラトニンの制御経皮投与
US5206377A (en) * 1991-12-05 1993-04-27 Whitby Research, Inc. Compounds useful as antiproliferative agents
IT1255199B (it) * 1992-07-01 1995-10-20 Franco Fraschini Farmaco sintetizzato analogo della melatonina particolarmente efficacenelle patologie che interferiscono con i ritmi circadiani
US5300481A (en) * 1993-05-05 1994-04-05 The Regents Of The University Of California Methods for controlling flowering in plants
US5654325A (en) * 1993-11-18 1997-08-05 Eli Lilly And Company Melatonin derivatives for use in treating sleep disorders
US6180657B1 (en) 1993-11-18 2001-01-30 Eli Lilly And Company Melatonin derivatives for use in treating desynchronization disorders
FR2713636B1 (fr) * 1993-12-07 1996-01-05 Adir Nouveaux dérivés naphtaléniques, leur procédé de préparation, et les compositions pharmaceutiques qui les contiennent.
US5403851A (en) * 1994-04-05 1995-04-04 Interneuron Pharmaceuticals, Inc. Substituted tryptamines, phenalkylamines and related compounds
FR2724170B1 (fr) * 1994-09-02 1997-05-30 Cemaf Nouveaux derives de spiro(indole-pyrrolidine) agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament
CN1047386C (zh) * 1994-04-07 1999-12-15 西玛夫公司 新型褪黑激素拮抗物螺旋[吲哚吡咯烷丁]衍生物,其制备方法及其作为药物产品的用途
FR2718445B1 (fr) * 1994-04-07 1996-06-28 Cemaf Nouveaux dérivés de spiro [indole-pyrrolidine] agonistes de la mélatonine, leur procédé de préparation et leur utilisation à titre de médicament.
ES2172415B2 (es) * 2000-07-28 2003-11-16 Univ Madrid Complutense Tratamiento del glaucoma y la hipertension ocular por medio de un analogo de la melatonina.
AR035651A1 (es) * 2000-07-28 2004-06-23 Univ Madrid Complutense Uso de derivados de indol para la manufactura de un medicamento para reducir la presion intraocular y una composicion
WO2002072145A1 (en) 2001-03-14 2002-09-19 Ono Pharmaceutical Co., Ltd. Remedies for depression containing ep1 antagonist as the active ingredient
FR2874611B1 (fr) * 2004-08-31 2006-11-17 Servier Lab Nouveaux derives d'imidazopyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2010012789A1 (en) 2008-07-30 2010-02-04 Ferrer Internacional S. A. 1,6-dihydro-2h-3-oxa-6-aza-as-indacene compounds
KR101534523B1 (ko) * 2013-04-30 2015-07-09 경희대학교 산학협력단 1,2,3,4-테트라히드로-6-메톡시-1-옥소-베타-카르볼린을 포함하는 피부 미백용 화장료 조성물
FR3065225B1 (fr) 2017-04-12 2024-04-05 Patrick Choay Sas Adjuvants depourvus de cytokines pour milieux de culture cellulaire, notamment pour fecondation in vitro, ou pour la culture de follicules, cellules germinales males ou embryons

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3370063A (en) * 1964-10-05 1968-02-20 Mcneilab Inc Substituted dimethoxy indoles and method of making the same
US3915990A (en) * 1973-03-13 1975-10-28 Nelson Res & Dev Tryptamines
US4087444A (en) * 1976-09-08 1978-05-02 Eli Lilly And Company Amides as ovulation inhibitors

Also Published As

Publication number Publication date
NO173732C (no) 1994-01-26
FI900801A7 (fi) 1990-02-16
KR890701558A (ko) 1989-12-20
KR910006124B1 (ko) 1991-08-13
EP0375726A1 (en) 1990-07-04
NO173732B (no) 1993-10-18
NO900790D0 (no) 1990-02-19
WO1989001472A1 (en) 1989-02-23
AU2309788A (en) 1989-03-09
DK42490A (da) 1990-04-17
NO900790L (no) 1990-03-26
EP0375726A4 (en) 1991-01-30
AU616907B2 (en) 1991-11-14
DK42490D0 (da) 1990-02-16

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Legal Events

Date Code Title Description
FD Application lapsed
MM Patent lapsed

Owner name: NELSON RESEARCH & DEVELOPMENT CO.