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FI872577A7 - Menetelmä terapeuttisesti käyttökelpoisten, hydrofobisen tai niukkaliukoisen aineen mikronisoitujen, hydrofilisoitujen hiukkasten valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten, hydrofobisen tai niukkaliukoisen aineen mikronisoitujen, hydrofilisoitujen hiukkasten valmistamiseksi

Info

Publication number
FI872577A7
FI872577A7 FI872577A FI872577A FI872577A7 FI 872577 A7 FI872577 A7 FI 872577A7 FI 872577 A FI872577 A FI 872577A FI 872577 A FI872577 A FI 872577A FI 872577 A7 FI872577 A7 FI 872577A7
Authority
FI
Finland
Prior art keywords
hydrophobic
sparingly soluble
therapeutically useful
soluble substance
preparing therapeutically
Prior art date
Application number
FI872577A
Other languages
English (en)
Swedish (sv)
Other versions
FI872577A0 (fi
FI90823C (fi
FI90823B (fi
Inventor
Thomas Gergely
Irmgard Gergely
Original Assignee
Gergely Gerhard
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gergely Gerhard filed Critical Gergely Gerhard
Publication of FI872577A0 publication Critical patent/FI872577A0/fi
Publication of FI872577A7 publication Critical patent/FI872577A7/fi
Application granted granted Critical
Publication of FI90823B publication Critical patent/FI90823B/fi
Publication of FI90823C publication Critical patent/FI90823C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5015Organic compounds, e.g. fats, sugars
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5026Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5089Processes

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Glanulating (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fats And Perfumes (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI872577A 1984-12-14 1987-06-09 Menetelmä terapeuttisesti käyttökelpoisten, hydrofobisen tai niukkaliukoisen aineen mikronisoitujen, hydrofilisoitujen hiukkasten valmistamiseksi FI90823C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH594184 1984-12-14
CH594184 1984-12-14
PCT/EP1985/000697 WO1986003675A1 (fr) 1984-12-14 1985-12-12 Particules d'une substance hydrophobe ou difficilement soluble et procede pour les rendre hydrophiles
EP8500697 1985-12-12

Publications (4)

Publication Number Publication Date
FI872577A0 FI872577A0 (fi) 1987-06-09
FI872577A7 true FI872577A7 (fi) 1987-06-09
FI90823B FI90823B (fi) 1993-12-31
FI90823C FI90823C (fi) 1994-04-11

Family

ID=4301863

Family Applications (1)

Application Number Title Priority Date Filing Date
FI872577A FI90823C (fi) 1984-12-14 1987-06-09 Menetelmä terapeuttisesti käyttökelpoisten, hydrofobisen tai niukkaliukoisen aineen mikronisoitujen, hydrofilisoitujen hiukkasten valmistamiseksi

Country Status (8)

Country Link
US (1) US5158779A (fi)
EP (1) EP0241469B1 (fi)
JP (1) JPH07106977B2 (fi)
AT (1) ATE68695T1 (fi)
AU (1) AU5356986A (fi)
DE (1) DE3584522D1 (fi)
FI (1) FI90823C (fi)
WO (1) WO1986003675A1 (fi)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8630273D0 (en) * 1986-12-18 1987-01-28 Til Medical Ltd Pharmaceutical delivery systems
JPH02500591A (ja) * 1987-05-27 1990-03-01 アクゾ・エヌ・ヴエー β‐ラクタム抗生物質の乾燥した急速溶解性の組成物
US4971804A (en) * 1989-02-02 1990-11-20 Warner-Lambert Company Water dispersible gemfibrozil compositions
US5213800A (en) * 1989-02-09 1993-05-25 Diamond Scientific Company Chlorhexidine disinfectant granules
US5064656A (en) * 1989-11-14 1991-11-12 Dr. Gergely & Co. Uncoated pharmaceutical reaction tablet
FR2682874B1 (fr) * 1991-10-24 1993-12-10 Rinrone Ets Procede pour la preparation d'un extrait de principes actifs sous forme seche adsorbable et microgranules adsorbables ainsi obtenus.
FR2708853A1 (fr) * 1993-06-30 1995-02-17 Salsarulo Gilles Composition à base d'acide acétylsalicylique à biodisponibilité améliorée et procédé pour la produire.
CH686865A5 (de) * 1994-06-15 1996-07-31 Gergely Gerhard Pharmazeutische Zubereitung mit einem hydrophoben Wirkstoff und einem Brausesystem, sowie Verfahren zur Herstellung der Zubereitung.
US20030109503A1 (en) * 1995-06-06 2003-06-12 Smithkline Beecham P.L.C. Pharmaceutical formulations comprising clavulanic acid alone or in combination with other beta-lactam antibiotics
US6974595B1 (en) * 1996-05-17 2005-12-13 Proethic Pharmaceuticals, Inc. Pharmaceutical compositions based on Diclofenae
US20030124187A1 (en) * 1997-02-14 2003-07-03 Smithkline Beecham Laboratoires Pharmaceutiques, Pharmaceutical formulations comprising amoxycillin and clavulanate
PT1023050E (pt) * 1997-06-27 2013-12-04 Abraxis Bioscience Llc Novas formulações de agentes farmacológicos, métodos para a sua preparação e métodos para a sua utilização
BR9909434A (pt) * 1998-04-09 2000-12-12 Eurand Int Microcápsulas umectáveis tendo núcleos revestidos de polìmero hidrofóbico
US6294199B1 (en) * 1999-04-13 2001-09-25 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising administering amoxycillin
US7250176B1 (en) * 1999-04-13 2007-07-31 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection
US6878386B1 (en) 1999-04-13 2005-04-12 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising amoxycillin and potassium clavulanate
EP1116485A3 (de) * 2000-01-10 2002-01-16 Gerhard Dr. Gergely Instant-Granulat und Verfahren zu seiner Herstellung
AU2001292185A1 (en) 2000-10-12 2002-04-22 Beecham Pharmaceuticals (Pte) Limited Formulation containing amoxicillin
US6756057B2 (en) 2000-10-12 2004-06-29 Beecham Pharmaceuticals (Pte) Limited Amoxicillin and potassium clavulanate dosage form
AU2003302579B2 (en) * 2002-12-02 2008-09-18 Bharat Serums And Vaccines Ltd. Ifosfamide compositions for parenteral administration and a process for their preparation
US7199111B2 (en) * 2002-12-02 2007-04-03 Bharat Serums & Vaccines Ltd. Aqueous ifosfamide compositions for parenteral administration and a process for their preparations
US6874708B2 (en) * 2003-02-13 2005-04-05 Illinois Tool Works Inc. Automatic air-assisted manifold mounted gun
US8216610B2 (en) 2004-05-28 2012-07-10 Imaginot Pty Ltd. Oral paracetamol formulations
JP2008500288A (ja) * 2004-05-28 2008-01-10 イメイジノット ピーティーワイ エルティーディー 経口治療用化合物の供給系
US9757455B2 (en) * 2005-11-28 2017-09-12 Johnson & Johnson Consumer Inc. Oral therapeutic compound delivery system
US20070267859A1 (en) * 2006-05-19 2007-11-22 Milman David A Service order payment and receipt form set

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB970462A (en) * 1962-05-02 1964-09-23 Monsanto Co Free-flowing acid compositions
US3887700A (en) * 1969-11-28 1975-06-03 Aspro Nicholas Ltd Analgesic formulations
US3920442A (en) * 1972-09-18 1975-11-18 Du Pont Water-dispersible pesticide aggregates
ZA739543B (en) * 1973-02-16 1975-03-26 Hoffmann La Roche Free-flowing, directly tablettable, pharmaceutically active substances
US4344934A (en) * 1978-11-20 1982-08-17 American Home Products Corporation Therapeutic compositions with enhanced bioavailability
AT368880B (de) * 1980-05-02 1982-11-25 Gergely Gerhard Verfahren zur herstellung eines zur weiterverarbeitung zu einer waesserigen suspension dienenden wasserunloeslichen trockeninstantpr[parates
AT376147B (de) * 1980-12-15 1984-10-10 Gergely Gerhard Verfahren und vorrichtung zum granulieren eines pulvergemisches

Also Published As

Publication number Publication date
EP0241469B1 (de) 1991-10-23
AU5356986A (en) 1986-07-22
ATE68695T1 (de) 1991-11-15
WO1986003675A1 (fr) 1986-07-03
FI872577A0 (fi) 1987-06-09
DE3584522D1 (de) 1991-11-28
JPH07106977B2 (ja) 1995-11-15
EP0241469A1 (de) 1987-10-21
JPS62501421A (ja) 1987-06-11
FI90823C (fi) 1994-04-11
FI90823B (fi) 1993-12-31
US5158779A (en) 1992-10-27

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Legal Events

Date Code Title Description
BB Publication of examined application
FG Patent granted

Owner name: GERGELY, GERHARD

MA Patent expired