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FI20030166L - Pysyvästi vapauttava valmiste - Google Patents

Pysyvästi vapauttava valmiste Download PDF

Info

Publication number
FI20030166L
FI20030166L FI20030166A FI20030166A FI20030166L FI 20030166 L FI20030166 L FI 20030166L FI 20030166 A FI20030166 A FI 20030166A FI 20030166 A FI20030166 A FI 20030166A FI 20030166 L FI20030166 L FI 20030166L
Authority
FI
Finland
Prior art keywords
sustained
release preparation
release
preparation
Prior art date
Application number
FI20030166A
Other languages
English (en)
Swedish (sv)
Other versions
FI116196B (fi
Inventor
Shigeru Kamei
Yasutaka Igari
Yasuaki Ogawa
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of FI20030166L publication Critical patent/FI20030166L/fi
Application granted granted Critical
Publication of FI116196B publication Critical patent/FI116196B/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/23Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • A61K38/09Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647Polyesters, e.g. poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Reproductive Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Diabetes (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI20030166A 1992-12-07 2003-02-04 Menetelmä jatkuvasti vapauttavan valmisteen tuottamiseksi FI116196B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP32707092 1992-12-07
JP32707092 1992-12-07
JP1897893 1993-02-05
JP1897893 1993-02-05
JP14513493 1993-06-16
JP14513493 1993-06-16

Publications (2)

Publication Number Publication Date
FI20030166L true FI20030166L (fi) 2003-02-04
FI116196B FI116196B (fi) 2005-10-14

Family

ID=27282444

Family Applications (2)

Application Number Title Priority Date Filing Date
FI935471A FI935471A7 (fi) 1992-12-07 1993-12-07 Pysyvästi vapauttava valmiste
FI20030166A FI116196B (fi) 1992-12-07 2003-02-04 Menetelmä jatkuvasti vapauttavan valmisteen tuottamiseksi

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI935471A FI935471A7 (fi) 1992-12-07 1993-12-07 Pysyvästi vapauttava valmiste

Country Status (23)

Country Link
US (7) US5480868A (fi)
EP (2) EP0601799B1 (fi)
JP (1) JP3725906B2 (fi)
KR (2) KR100305951B1 (fi)
CN (2) CN1099893C (fi)
AT (2) ATE295733T1 (fi)
AU (1) AU669939B2 (fi)
CA (1) CA2110730C (fi)
DE (2) DE69330547T2 (fi)
DK (2) DK0601799T3 (fi)
EE (1) EE03117B1 (fi)
ES (2) ES2158856T3 (fi)
FI (2) FI935471A7 (fi)
GE (1) GEP19991600B (fi)
GR (1) GR3037085T3 (fi)
LV (1) LV10927B (fi)
MX (1) MX9307686A (fi)
NO (1) NO310704B1 (fi)
NZ (1) NZ250349A (fi)
PT (2) PT1088555E (fi)
SG (1) SG46283A1 (fi)
TW (1) TW333456B (fi)
WO (1) WO1994013317A1 (fi)

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* Cited by examiner, † Cited by third party
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US5668111A (en) 1997-09-16
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