FI20011433L - Förfarande för framställning av 2,5-diamino-4,6-diklorpyrimidin - Google Patents

Förfarande för framställning av 2,5-diamino-4,6-diklorpyrimidin Download PDF

Info

Publication number: FI20011433L
Authority: FI; Finland
Prior art keywords: dichloropyrimidine; diamino; preparation
Prior art date: 1994-04-27

Application number

FI20011433A

Other languages

English (en)

Finnish (fi)

Other versions

FI109693B (sv

Inventor

Gerhard Stucky

Rene Imwinkelried

Original Assignee

Lonza Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-04-27

Filing date

2001-07-02

Publication date

2001-07-02

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4207186&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI20011433(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2001-07-02 Application filed by Lonza Ag filed Critical Lonza Ag

2001-07-02 Publication of FI20011433L publication Critical patent/FI20011433L/sv

2002-09-30 Application granted granted Critical

2002-09-30 Publication of FI109693B publication Critical patent/FI109693B/sv

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Virology (AREA)
Communicable Diseases (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Saccharide Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Pyridine Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

FI20011433A 1994-04-27 2001-07-02 Förfarande för framställning av 2,5-diamino-4,6-diklorpyrimidin FI109693B (sv)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH129994		1994-04-27
CH129994		1994-04-27

Publications (2)

Publication Number	Publication Date
FI20011433L true FI20011433L (sv)	2001-07-02
FI109693B FI109693B (sv)	2002-09-30

Family

ID=4207186

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
FI952009A FI109119B (sv)	1994-04-27	1995-04-27	N-(2-amino-4,6-diklor-pyrimidin-5-yl)formamid förfarande för framställning därav samt mellanprodukt därav
FI20011433A FI109693B (sv)	1994-04-27	2001-07-02	Förfarande för framställning av 2,5-diamino-4,6-diklorpyrimidin

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
FI952009A FI109119B (sv)	1994-04-27	1995-04-27	N-(2-amino-4,6-diklor-pyrimidin-5-yl)formamid förfarande för framställning därav samt mellanprodukt därav

Country Status (18)

Country	Link
US (4)	US5583226A (sv)
EP (2)	EP0684236B2 (sv)
JP (2)	JP3811966B2 (sv)
KR (1)	KR100327996B1 (sv)
CN (2)	CN1065862C (sv)
AT (2)	ATE167672T1 (sv)
CA (1)	CA2145928C (sv)
CZ (1)	CZ287261B6 (sv)
DE (2)	DE59510726D1 (sv)
DK (2)	DK0684236T4 (sv)
ES (2)	ES2120099T5 (sv)
FI (2)	FI109119B (sv)
HU (3)	HU219716B (sv)
NO (2)	NO306461B1 (sv)
PL (1)	PL190855B1 (sv)
PT (1)	PT816344E (sv)
SK (1)	SK282208B6 (sv)
TW (1)	TW442474B (sv)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9402161D0 (en) *	1994-02-04	1994-03-30	Wellcome Found	Chloropyrimidine intermediates
CA2145928C (en) *	1994-04-27	2007-10-09	Gerhard Stucky	N-(2-amino-4,6-dichloropyrimidin-5-yl)formamide, and a process for its preparation
HK1042474B (zh)	1998-10-30	2003-11-21	Lonza Ag	制备4-[(2'，5'-二胺基-6'-卤代咪啶-4'-)胺]-环戊-2-烯-甲醇的方法
WO2000026193A1 (de) *	1998-10-30	2000-05-11	Lonza Ag	Verfahren zur herstellung von 4-[(2',5'-diamino-6'-halogenpyrimidin-4'-yl)amino]-cyclopent-2-enylmethanolen
ES2204798T3 (es)	1998-12-21	2004-05-01	Lonza Ag	Procedimiento para la preparacion de 2,5-diamino-4,6-dihalogenopirimidina.
US6608199B2 (en)	2000-07-07	2003-08-19	Syngenta Limited	Synthesis of chlorinated pyrimidines
JP2002223094A (ja) *	2001-01-25	2002-08-09	Yokohama Rubber Co Ltd:The	電波吸収体の構造
US6982331B2 (en) *	2001-06-08	2006-01-03	Syngenta Crop Protection, Inc.	Synthesis of chlorinated pyrimidines
FR2849030A1 (fr) *	2002-12-20	2004-06-25	Isochem Sa	Procede de preparation des n-(2-amino-4, 6-dihalogenopyrimidin-5-yl) formamides
JPWO2004103979A1 (ja) *	2003-05-26	2006-07-20	住友化学株式会社	Ｎ−（２−アミノ−４，６−ジクロロピリミジン−５−イル）ホルムアミドの製造方法
DE102004002055A1 (de) *	2004-01-15	2005-08-11	Degussa Ag	Verfahren zur Herstellung von 2-Amino-4,6-dichlor-5-formamidopyrimidin
CN101003511B (zh) *	2007-01-19	2010-06-09	中国科学院上海有机化学研究所	制备2-氨基-4,6-二氯-5-甲酰氨基嘧啶的方法
CN102127022A (zh) *	2010-12-30	2011-07-20	苏州开元民生科技股份有限公司	2-氨基-4,6-二氯-5-甲酰胺基嘧啶的合成方法
CZ305457B6 (cs)	2011-02-28	2015-09-30	Ústav organické chemie a biochemie, Akademie věd ČR v. v. i.	Pyrimidinové sloučeniny inhibující tvorbu oxidu dusnatého a prostaglandinu E2, způsob výroby a použití
CZ305750B6 (cs) *	2012-01-26	2016-03-02	Ústav Organické Chemie A Biochemie Akademie Věd Čr, V.V.I.	Způsob výroby N-9 substituovaných analogů purinu
CN102702110A (zh) *	2012-05-24	2012-10-03	盛世泰科生物医药技术(苏州)有限公司	一种4-氨基-5,6-二氯嘧啶的制备方法
EP2882720A1 (en) *	2012-08-06	2015-06-17	Enantia, S.L.	A process for the preparation of an intermediate for a triazolopyrimidine carbonucleoside

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8916698D0 (en) *	1989-07-21	1989-09-06	Beecham Group Plc	Novel process
SK279618B6 (sk) *	1992-01-22	1999-01-11	Lonza A.G. (Dir.:Basel)	N-5-chránené 2,5-diamino-4,6-dichlórpyrimidíny a s
GB9402161D0 (en) *	1994-02-04	1994-03-30	Wellcome Found	Chloropyrimidine intermediates
CA2145928C (en) *	1994-04-27	2007-10-09	Gerhard Stucky	N-(2-amino-4,6-dichloropyrimidin-5-yl)formamide, and a process for its preparation

1995
- 1995-03-30 CA CA002145928A patent/CA2145928C/en not_active Expired - Fee Related
- 1995-04-25 PT PT97114001T patent/PT816344E/pt unknown
- 1995-04-25 DK DK95106220T patent/DK0684236T4/da active
- 1995-04-25 AT AT95106220T patent/ATE167672T1/de active
- 1995-04-25 AT AT97114001T patent/ATE243200T1/de active
- 1995-04-25 DE DE59510726T patent/DE59510726D1/de not_active Expired - Lifetime
- 1995-04-25 ES ES95106220T patent/ES2120099T5/es not_active Expired - Lifetime
- 1995-04-25 EP EP95106220A patent/EP0684236B2/de not_active Expired - Lifetime
- 1995-04-25 US US08/428,916 patent/US5583226A/en not_active Expired - Lifetime
- 1995-04-25 JP JP10149995A patent/JP3811966B2/ja not_active Expired - Fee Related
- 1995-04-25 ES ES97114001T patent/ES2201229T3/es not_active Expired - Lifetime
- 1995-04-25 DK DK97114001T patent/DK0816344T3/da active
- 1995-04-25 EP EP97114001A patent/EP0816344B1/de not_active Expired - Lifetime
- 1995-04-25 DE DE59502637T patent/DE59502637D1/de not_active Expired - Lifetime
- 1995-04-26 HU HU9501194A patent/HU219716B/hu not_active IP Right Cessation
- 1995-04-26 NO NO951594A patent/NO306461B1/no not_active IP Right Cessation
- 1995-04-26 SK SK541-95A patent/SK282208B6/sk not_active IP Right Cessation
- 1995-04-26 CZ CZ19951067A patent/CZ287261B6/cs not_active IP Right Cessation
- 1995-04-26 HU HU0003724A patent/HU219986B/hu not_active IP Right Cessation
- 1995-04-26 HU HU0003725A patent/HU219712B/hu not_active IP Right Cessation
- 1995-04-27 CN CN95106201A patent/CN1065862C/zh not_active Expired - Fee Related
- 1995-04-27 CN CNB991234553A patent/CN1193991C/zh not_active Expired - Fee Related
- 1995-04-27 FI FI952009A patent/FI109119B/sv not_active IP Right Cessation
- 1995-04-27 PL PL308394A patent/PL190855B1/pl not_active IP Right Cessation
- 1995-04-27 KR KR1019950010196A patent/KR100327996B1/ko not_active Expired - Fee Related
- 1995-05-06 TW TW084104525A patent/TW442474B/zh not_active IP Right Cessation
1996
- 1996-08-08 US US08/693,521 patent/US5693800A/en not_active Expired - Lifetime
- 1996-08-08 US US08/693,520 patent/US5663340A/en not_active Expired - Lifetime
1997
- 1997-05-12 US US08/854,378 patent/US5744601A/en not_active Expired - Lifetime
1998
- 1998-10-01 NO NO984588A patent/NO306859B1/no not_active IP Right Cessation
2001
- 2001-07-02 FI FI20011433A patent/FI109693B/sv not_active IP Right Cessation
2006
- 2006-04-03 JP JP2006102585A patent/JP4525625B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
EP0684236B1 (de)	1998-06-24
FI109693B (sv)	2002-09-30
JP3811966B2 (ja)	2006-08-23
HU0003724D0 (sv)	2000-11-28
EP0816344A1 (de)	1998-01-07
SK282208B6 (sk)	2001-12-03
JP4525625B2 (ja)	2010-08-18
HUT70700A (en)	1995-10-30
PT816344E (pt)	2003-10-31
ATE243200T1 (de)	2003-07-15
DK0684236T3 (da)	1998-11-02
JP2006199707A (ja)	2006-08-03
HU9501194D0 (en)	1995-06-28
US5663340A (en)	1997-09-02
NO984588L (no)	1995-10-30
CN1065862C (zh)	2001-05-16
NO951594L (no)	1995-10-30
EP0816344B1 (de)	2003-06-18
ES2201229T3 (es)	2004-03-16
CA2145928C (en)	2007-10-09
DE59502637D1 (de)	1998-07-30
KR100327996B1 (ko)	2002-07-27
CN1113237A (zh)	1995-12-13
ES2120099T5 (es)	2008-05-16
HU219986B (hu)	2001-10-28
NO984588D0 (no)	1998-10-01
US5744601A (en)	1998-04-28
US5583226A (en)	1996-12-10
DK0816344T3 (da)	2003-10-06
EP0684236B2 (de)	2007-12-26
CN1193991C (zh)	2005-03-23
NO306461B1 (no)	1999-11-08
NO306859B1 (no)	2000-01-03
HU0003725D0 (sv)	1995-04-26
CA2145928A1 (en)	1995-10-28
US5693800A (en)	1997-12-02
FI109119B (sv)	2002-05-31
TW442474B (en)	2001-06-23
CZ287261B6 (en)	2000-10-11
DK0684236T4 (da)	2008-05-05
ATE167672T1 (de)	1998-07-15
KR950032143A (ko)	1995-12-20
HU219716B (hu)	2001-06-28
SK54195A3 (en)	1995-11-08
EP0684236A3 (de)	1996-07-17
EP0684236A2 (de)	1995-11-29
FI952009L (sv)	1995-10-28
HU219712B (hu)	2001-06-28
FI952009A0 (sv)	1995-04-27
ES2120099T3 (es)	1998-10-16
PL308394A1 (en)	1995-10-30
CN1259517A (zh)	2000-07-12
CZ106795A3 (en)	1995-11-15
PL190855B1 (pl)	2006-02-28
NO951594D0 (no)	1995-04-26
DE59510726D1 (de)	2003-07-24
JPH07300466A (ja)	1995-11-14

Publication	Publication Date	Title
DK0719788T3 (da)	1999-11-01	Fremgangsmåde til fremstilling af 1-(2'-deoxy-2',2'-difluor-D-ribofuranosyl)-4-aminopyrimidin-2-on-hydrochlorid
NO981800L (no)	1998-06-11	FremgangsmÕte for fremstilling av 1,1,1,3,3-pentafluorpentan
FI971268A7 (sv)	1997-03-26	Förfarande för framställning av 1,3-alkandioler och 3-hydroxialdehyder
FI20011433L (sv)	2001-07-02	Förfarande för framställning av 2,5-diamino-4,6-diklorpyrimidin
FI952424L (sv)	1995-11-20	11,21-bisfenyl-19-norpregnanderivat
DE59507222D1 (de)	1999-12-16	Substituierte 1,2,3,4-tetrahydro-5-nitro-pyrimidine
MA24182A1 (fr)	1997-12-31	Procede pour la preparation de 2,4-diaminopyrimidines substituees
EP1023250A4 (en)	2001-03-21	METHOD FOR PRODUCING 2,6-DIALKYLNAPHTHALINE
FI972742A0 (sv)	1997-06-25	Lösningsmedelsfritt förfarande för framställning av 2,6-difluorbensonitril
DK0815092T3 (da)	1999-12-06	Fremgangsmåde til fremstilling af 1,2-benzisothiazolin-3-oner
NO985535L (no)	1999-01-27	FremgangsmÕte for fremstilling av 1,3-alkandioler
FI971267A7 (sv)	1997-03-26	Förfarande för framställning av 1,3-alkandioler och 3-hydroxialdehyder
DK0735043T3 (da)	1998-10-07	Fremgangsmåde til fremstilling af 2-substitueret 3,3-difluorfuran
FI952145L (sv)	1995-11-07	Förfarande för framställning av alfa-D-glukopyrano-sido-1,6-mannitol och -sorbitol från alfa-D-glukopyranosido-1,6-fruktos
FI964410A7 (sv)	1996-11-01	Förfarande för framställning av 4-amino-delta4-3-ketosteroider genom 4 -nitro-delta4-3-ketosteroider
FI952287A7 (sv)	1995-11-14	Förfarande för framställning av 2-amino-4,6-diklor-pyrimidin
FI943833A0 (sv)	1994-08-19	Förfarande för framställning av 2,3,5,6-tetraklorpyridin
FI964278L (sv)	1996-12-20	Förfarande för framställning av 5,6-dihydroxi-2-amino-1,2,3,4-tetrahydronaftalenderivat
FI930237A7 (sv)	1993-07-24	Förfarande för framställning av 4,6-dialkoxipyrimidiner
BR9508248A (pt)	1997-11-04	1,2,4,6-Tiatriazinas herbicidas
FI970039A7 (sv)	1997-01-03	Förfarande för framställning av 5-aryl-2,4-dialkyl-3H-1,2,3-triazol-3- tioner
FI971964L (sv)	1997-05-07	Förfarande för framställning av 1-halo-3-trialkylsilanylbensenderivat
ITMI941144A0 (it)	1994-06-02	Procedimento per la formazione di timbri
DK0783491T3 (da)	2002-01-21	Fremgangsmåde til fremstilling af 3,3,5-trichlorglutarimid
FI973631L (sv)	1999-03-09	1,3-diolbaserade etrar, förfarande för framställning av 1,3-diolbaserade etrar samt användningen av etrarna

Legal Events

Date	Code	Title	Description
2012-12-11	MM	Patent lapsed