ES8302692A1 - Novel n-((2-oxo-1-pyrrolidinyl)acetyl)piperazine, manufacture of same and salts and medicine of therapeutical drug - Google Patents
Novel n-((2-oxo-1-pyrrolidinyl)acetyl)piperazine, manufacture of same and salts and medicine of therapeutical drugInfo
- Publication number
- ES8302692A1 ES8302692A1 ES510759A ES510759A ES8302692A1 ES 8302692 A1 ES8302692 A1 ES 8302692A1 ES 510759 A ES510759 A ES 510759A ES 510759 A ES510759 A ES 510759A ES 8302692 A1 ES8302692 A1 ES 8302692A1
- Authority
- ES
- Spain
- Prior art keywords
- formula
- oxo
- acetyl
- salts
- pyrrolidinyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000003839 salts Chemical class 0.000 title abstract 2
- GLUUGHFHXGJENI-UHFFFAOYSA-N Piperazine Chemical compound C1CNCCN1 GLUUGHFHXGJENI-UHFFFAOYSA-N 0.000 title 2
- 239000003814 drug Substances 0.000 title 2
- 229940079593 drug Drugs 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 2
- 239000002904 solvent Substances 0.000 abstract 2
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 125000000218 acetic acid group Chemical group C(C)(=O)* 0.000 abstract 1
- 238000004821 distillation Methods 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 150000004885 piperazines Chemical class 0.000 abstract 1
- 239000007787 solid Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
Procedure for the obtaining of n - [(2-oxo-1-pirrolidinil) acetyl] substituted piperazines and of their physiologically compatible salts, of formula (I), in which r can be one of various types of radicals and r " it is hydrogen, methyl or ethyl. It consists of the reaction of a mol of an amina of formula (II) with a mol or an excess of ester of formula (III) in which r "'' 'is methyle or ethyl; and r and r "have the same meaning as in formula (I). The reaction is carried out in a solid solvent or in absence of solvents, at temperatures comprised between 170ºc and 190ºc, eliminating the alcohol formed by distillation. (Machine-translation by Google Translate, not legally binding)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES510759A ES8302692A1 (en) | 1982-03-24 | 1982-03-24 | Novel n-((2-oxo-1-pyrrolidinyl)acetyl)piperazine, manufacture of same and salts and medicine of therapeutical drug |
| DE8383400607T DE3361609D1 (en) | 1982-03-24 | 1983-03-23 | New n-((2-oxo-1-pyrrolidinyl)acetyl)piperazines, the methods of producing such new compounds and their salts as well as pharmaceutical preparations for therapeutic use containing these compounds or salts |
| EP83400607A EP0089900B1 (en) | 1982-03-24 | 1983-03-23 | New n-((2-oxo-1-pyrrolidinyl)acetyl)piperazines, the methods of producing such new compounds and their salts as well as pharmaceutical preparations for therapeutic use containing these compounds or salts |
| AT83400607T ATE17120T1 (en) | 1982-03-24 | 1983-03-23 | N-((2-OXO-1-PYRROLIDINYL)ACETYL)PIPERAZINE, PROCESS FOR THEIR PRODUCTION AND THEIR SALTS AND THEIR USE IN PHARMACEUTICAL PREPARATIONS. |
| JP58049659A JPS58174360A (en) | 1982-03-24 | 1983-03-24 | Novel n-((2-oxo-1-pyrrolidinyl)acetyl)piperazine, manufacture of same and salts and medicine of therapeutical drug |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES510759A ES8302692A1 (en) | 1982-03-24 | 1982-03-24 | Novel n-((2-oxo-1-pyrrolidinyl)acetyl)piperazine, manufacture of same and salts and medicine of therapeutical drug |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES510759A0 ES510759A0 (en) | 1983-02-01 |
| ES8302692A1 true ES8302692A1 (en) | 1983-02-01 |
Family
ID=8483886
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES510759A Expired ES8302692A1 (en) | 1982-03-24 | 1982-03-24 | Novel n-((2-oxo-1-pyrrolidinyl)acetyl)piperazine, manufacture of same and salts and medicine of therapeutical drug |
Country Status (2)
| Country | Link |
|---|---|
| JP (1) | JPS58174360A (en) |
| ES (1) | ES8302692A1 (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH075545B2 (en) * | 1988-08-04 | 1995-01-25 | 明治製菓株式会社 | Pyrrolidinone compound and cerebral dysfunction improving agent |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2278340A1 (en) * | 1974-07-17 | 1976-02-13 | Delalande Sa | NEW DERIVATIVE OF N- (TRIMETHOXY-3,4,5 CINNAMOYL) PIPERAZINE, ITS ACID ADDITIONAL SALTS, ITS PREPARATION PROCESS AND ITS THERAPEUTIC APPLICATION |
-
1982
- 1982-03-24 ES ES510759A patent/ES8302692A1/en not_active Expired
-
1983
- 1983-03-24 JP JP58049659A patent/JPS58174360A/en active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| ES510759A0 (en) | 1983-02-01 |
| JPS58174360A (en) | 1983-10-13 |
| JPS6344745B2 (en) | 1988-09-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19970612 |