ES557198A0 - Un procedimiento para la preparacion de nuevos derivados de ciclopenta(d)pirimidina - Google Patents

Un procedimiento para la preparacion de nuevos derivados de ciclopenta(d)pirimidina

Info

Publication number: ES557198A0
Authority: ES; Spain
Prior art keywords: sup; procedure; preparation; hydrogen; cyclopenta
Prior art date: 1985-03-07
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

ES557198A

Other languages

English (en)

Other versions

ES8801221A1 (es

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sankyo Co Ltd

Ube Corp

Original Assignee

Sankyo Co Ltd

Ube Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-03-07

Filing date

1986-11-14

Publication date

1988-01-01

1986-11-14 Application filed by Sankyo Co Ltd, Ube Industries Ltd filed Critical Sankyo Co Ltd

1988-01-01 Publication of ES8801221A1 publication Critical patent/ES8801221A1/es

1988-01-01 Publication of ES557198A0 publication Critical patent/ES557198A0/es

Status Expired legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Psychiatry (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Dental Preparations (AREA)
Saccharide Compounds (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)
Luminescent Compositions (AREA)
Soil Working Implements (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
Eyeglasses (AREA)

ES557198A 1985-03-07 1986-11-14 Un procedimiento para la preparacion de nuevos derivados de ciclopenta(d)pirimidina Expired ES8801221A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP4362685		1985-03-07

Publications (2)

Publication Number	Publication Date
ES8801221A1 ES8801221A1 (es)	1988-01-01
ES557198A0 true ES557198A0 (es)	1988-01-01

Family

ID=12669058

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
ES552796A Expired ES8704905A1 (es)	1985-03-07	1986-03-07	Un procedimiento para la preparacion de nuevos derivados de ciclopenta (d) pirimidina.
ES557198A Expired ES8801221A1 (es)	1985-03-07	1986-11-14	Un procedimiento para la preparacion de nuevos derivados de ciclopenta(d)pirimidina
ES557199A Expired ES8801222A1 (es)	1985-03-07	1986-11-14	Un procedimiento para la preparacion de nuevos derivados de ciclopenta(d)pirimidina

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
ES552796A Expired ES8704905A1 (es)	1985-03-07	1986-03-07	Un procedimiento para la preparacion de nuevos derivados de ciclopenta (d) pirimidina.

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
ES557199A Expired ES8801222A1 (es)	1985-03-07	1986-11-14	Un procedimiento para la preparacion de nuevos derivados de ciclopenta(d)pirimidina

Country Status (15)

Country	Link
US (1)	US4749704A (es)
EP (1)	EP0194161B1 (es)
JP (1)	JPS6270A (es)
KR (1)	KR890003839B1 (es)
AT (1)	ATE106077T1 (es)
AU (1)	AU580391B2 (es)
CA (1)	CA1273632A (es)
DE (1)	DE3689848T2 (es)
DK (1)	DK165109C (es)
ES (3)	ES8704905A1 (es)
FI (1)	FI88717C (es)
HK (1)	HK1005450A1 (es)
IE (1)	IE64504B1 (es)
NO (1)	NO168767C (es)
ZA (1)	ZA861708B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5037980A (en) *	1988-04-18	1991-08-06	American Cyanamid Company	Phenyl imidazo[1,2-a]pyrimidines
US5877178A (en) *	1991-04-08	1999-03-02	Duquesne University Of The Holy Ghost	Pyrimidine derivatives and methods of making and using these derivatives
US5234936A (en) *	1991-10-24	1993-08-10	American Home Products Corporation	Pyrimidocycloalkanes as a ii antagonists
JP2007501821A (ja) *	2003-08-12	2007-02-01	エフ．ホフマン−ラ　ロシュ　アーゲー	Ｃｆｒアンタゴニストとしてのテトラヒドロキナゾリン誘導体
US7568556B2 (en)	2005-10-26	2009-08-04	Mitsubishi Electric Corporation	Elevator group management control device
US8063050B2 (en)	2006-07-06	2011-11-22	Array Biopharma Inc.	Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors
WO2008006039A1 (en)	2006-07-06	2008-01-10	Array Biopharma Inc.	Dihydrothieno pyrimidines as akt protein kinase inhibitors
PL2049500T3 (pl)	2006-07-06	2012-02-29	Array Biopharma Inc	Cyklopenta[d]pirymidyny jako inhibitory kinaz białkowych AKT
WO2008006025A1 (en)	2006-07-06	2008-01-10	Array Biopharma Inc.	Dihydrofuro pyrimidines as akt protein kinase inhibitors
WO2008021456A2 (en) *	2006-08-16	2008-02-21	Cytovia, Inc.	N-aryl-5,7-dihydrofuro[3,4-d]pyrimidin-4-amines and analogs as activators of caspases and inducers of apoptosis and the use thereof
BRPI0813999A2 (pt)	2007-07-05	2019-10-01	Array Biopharma Inc	ciclopentanos de pirimidil como inibidores de akt proteína cinase
US8846683B2 (en)	2007-07-05	2014-09-30	Array Biopharma, Inc.	Pyrimidyl cyclopentanes as Akt protein kinase inhibitors
US9409886B2 (en)	2007-07-05	2016-08-09	Array Biopharma Inc.	Pyrimidyl cyclopentanes as AKT protein kinase inhibitors
EP2404907B1 (en)	2007-07-05	2015-01-14	Array Biopharma, Inc.	Pyrimidyl cyclopentanes as AKT protein kinase inhibitors
AU2009204019B2 (en)	2008-01-09	2014-02-20	Array Biopharma Inc.	Hydroxylated pyrimidyl cyclopentane as AKT protein kinase inhibitor
KR101624753B1 (ko)	2008-01-09	2016-05-26	어레이 바이오파마 인크.	Ａｋｔ 단백질 키나제 저해물질로서의 수산화된 피리미딜 시클로펜탄
WO2010047201A1 (ja)	2008-10-20	2010-04-29	三菱電機株式会社	エレベーター群管理装置
BR112013025397A2 (pt)	2011-04-01	2019-09-24	Deepak Sampath	combinação de um composto, composto de fórmula i ou um sal farmaceuticamente aceitável do mesmo, uso, kit, produto, método para tratamento de um distúrbio hiperproliferativo e método para tratamento de uma doença ou afecção modulada por quinase akt em um mamífero
CA2831922C (en)	2011-04-01	2019-12-31	Genentech, Inc.	Combinations of akt inhibitor compounds and vemurafenib, and methods of use
GB201121127D0 (en)	2011-12-08	2012-01-18	Dow Corning	Treatment of filler with silane
CN111303053B (zh) *	2020-03-16	2023-01-17	中国海洋大学	环戊并[d]嘧啶类化合物及其药学上可接受的盐、溶剂合物或者前药以及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3470182A (en) *	1967-02-09	1969-09-30	Sandoz Ag	4-amino-substituted quinazolines
US3980650A (en) *	1972-05-05	1976-09-14	N.V. Koninklijke Pharmaceutische Fabrieken V/H Brocades-Stheeman En Pharmacia	4-Amino-pyrimidine derivatives
US3915976A (en) *	1972-09-01	1975-10-28	Sandoz Ag	Substituted-4-phenyl-5h-cycloalkano(d)pyrimidines
PH20344A (en) *	1981-01-29	1986-12-04	Sankyo Co	Aminopyrimidine derivatives, processes for their preparation, and fungicidal, insecticidal and acaricidal compositions containing them
JPS57203072A (en) *	1981-06-05	1982-12-13	Sankyo Co Ltd	4-anilinopyrimidine derivative, its preparation, antidepressant comprising it as active ingredient

1986
- 1986-03-06 JP JP61049238A patent/JPS6270A/ja not_active Withdrawn
- 1986-03-06 US US06/837,079 patent/US4749704A/en not_active Expired - Lifetime
- 1986-03-07 EP EP86301660A patent/EP0194161B1/en not_active Expired - Lifetime
- 1986-03-07 CA CA000503571A patent/CA1273632A/en not_active Expired - Lifetime
- 1986-03-07 ZA ZA861708A patent/ZA861708B/xx unknown
- 1986-03-07 DE DE3689848T patent/DE3689848T2/de not_active Expired - Fee Related
- 1986-03-07 KR KR1019860001624A patent/KR890003839B1/ko not_active Expired
- 1986-03-07 AT AT86301660T patent/ATE106077T1/de not_active IP Right Cessation
- 1986-03-07 DK DK106586A patent/DK165109C/da not_active IP Right Cessation
- 1986-03-07 IE IE59786A patent/IE64504B1/en not_active IP Right Cessation
- 1986-03-07 FI FI860969A patent/FI88717C/fi not_active IP Right Cessation
- 1986-03-07 ES ES552796A patent/ES8704905A1/es not_active Expired
- 1986-03-07 NO NO860852A patent/NO168767C/no unknown
- 1986-03-07 AU AU54481/86A patent/AU580391B2/en not_active Ceased
- 1986-11-14 ES ES557198A patent/ES8801221A1/es not_active Expired
- 1986-11-14 ES ES557199A patent/ES8801222A1/es not_active Expired
1998
- 1998-05-27 HK HK98104569A patent/HK1005450A1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
IE860597L (en)	1986-09-07
NO860852L (no)	1986-09-08
EP0194161A2 (en)	1986-09-10
IE64504B1 (en)	1995-08-09
DK106586D0 (da)	1986-03-07
EP0194161B1 (en)	1994-05-25
AU5448186A (en)	1986-09-11
DE3689848T2 (de)	1995-01-12
JPS6270A (ja)	1987-01-06
KR890003839B1 (ko)	1989-10-05
US4749704A (en)	1988-06-07
ES557199A0 (es)	1988-01-01
KR860007221A (ko)	1986-10-08
DE3689848D1 (de)	1994-06-30
EP0194161A3 (en)	1987-09-02
FI860969A0 (fi)	1986-03-07
ES8801221A1 (es)	1988-01-01
FI860969L (fi)	1986-09-08
NO168767C (no)	1992-04-01
DK165109C (da)	1993-03-01
ES8704905A1 (es)	1987-04-16
DK106586A (da)	1986-09-08
DK165109B (da)	1992-10-12
CA1273632A (en)	1990-09-04
FI88717C (fi)	1993-06-28
ZA861708B (en)	1986-11-26
FI88717B (fi)	1993-03-15
AU580391B2 (en)	1989-01-12
ATE106077T1 (de)	1994-06-15
NO168767B (no)	1991-12-23
HK1005450A1 (en)	1999-01-08
ES8801222A1 (es)	1988-01-01
ES552796A0 (es)	1987-04-16

Publication	Publication Date	Title
ES552796A0 (es)	1987-04-16	Un procedimiento para la preparacion de nuevos derivados de ciclopenta (d) pirimidina.
ZA858418B (en)	1986-07-30	5-alkyl-1-phenyl-2-piperazinoalkylpyrazoline-3-one compounds and methods for the preparation thereof,intermediates for use in the preparation of said compounds and medicaments containing said compounds
LV10422A (lv)	1995-02-20	Jaunie fluor-naftacendioni to glikozetie atvasinajumi un vinu razosanas panemiens
ES553207A0 (es)	1987-08-01	Un procedimiento para la preparacion de una octahidroindolizina
NO870423L (no)	1987-08-05	5-substituerte oktahydroindolizin-analgetiske forbindelser og 7-keto mellomprodukter.
JO1676B1 (en)	1992-08-09	Extra compounds indinol II
ES8407322A1 (es)	1984-10-01	Procedimiento para la preparacion de 7 -aciltio-15,16-metilen-3-oxo-17 -pregna-1,4-dien-21,17-carbolactonas
DE3572814D1 (en)	1989-10-12	1, 3-benzoxathiole derivatives, their use and their preparation
ATE32216T1 (de)	1988-02-15	Diphenylmethylimin-derivate.
ES550781A0 (es)	1987-10-01	Un procedimiento para preparar un derivado de 1-benzhidril--4-cinamilpiperazina
IE44449L (en)	1977-02-06	Morphanthridines
DE3674250D1 (de)	1990-10-25	Phenylpyrazinderivate, verfahren zu deren herstellung, pharmazeutische zusammensetzung und verwendung.
ATE81465T1 (de)	1992-10-15	Verwendung von 2-oxo-imidazolidin-derivaten zur behandlung von nierenkrankheiten.
ES8302008A1 (es)	1982-12-16	Un procedimiento para la preparacion de derivados de imidazo (2,1-b) tiazol.