ES406297A1 - A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) - Google Patents
A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding)Info
- Publication number
- ES406297A1 ES406297A1 ES406297A ES406297A ES406297A1 ES 406297 A1 ES406297 A1 ES 406297A1 ES 406297 A ES406297 A ES 406297A ES 406297 A ES406297 A ES 406297A ES 406297 A1 ES406297 A1 ES 406297A1
- Authority
- ES
- Spain
- Prior art keywords
- compound
- formula
- procedure
- translation
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 238000000034 method Methods 0.000 title abstract 3
- 150000003839 salts Chemical class 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000005277 alkyl imino group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000001118 alkylidene group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000003236 benzoyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C(*)=O 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 150000002431 hydrogen Chemical group 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 239000011593 sulfur Substances 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
A procedure for the preparation of an acyloxyalkylheterocyclic compound of formula: **(See formula)** where 2 is sulfur, oxygen or (lower) alkyl imino, each of groups A1 and A2 is lower alkylene or lower alkylidene, R1 is hydrogen, halogen or trifluoromethyl, R2 is acyl selected from the group consisting of higher aliphatic acyl, phenylalkanoyl lower or benzoyl in which the phenyl portion can carry no more than 3 halogen atoms, lower alkyl groups and/or lower alkoxy groups and n is 2 or 3, and their addition salts with acids; whose procedure is to react a compound of formula: **(See formula)** where Z, A1 and R1 are defined above, or their reactive derivatives, with an amine of formula: **(See formula)** where A2, R2 and n are as defined above, or their salts. Whereby the resulting compound is optionally converted into the acid addition salt thereof. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2144869 | 1969-03-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES406297A1 true ES406297A1 (en) | 1975-09-16 |
Family
ID=12055228
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES377689A Expired ES377689A1 (en) | 1969-03-20 | 1970-03-18 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
| ES406298A Expired ES406298A1 (en) | 1969-03-20 | 1972-09-01 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
| ES406297A Expired ES406297A1 (en) | 1969-03-20 | 1972-09-01 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
| ES406296A Expired ES406296A1 (en) | 1969-03-20 | 1972-09-01 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES377689A Expired ES377689A1 (en) | 1969-03-20 | 1970-03-18 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
| ES406298A Expired ES406298A1 (en) | 1969-03-20 | 1972-09-01 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES406296A Expired ES406296A1 (en) | 1969-03-20 | 1972-09-01 | A procedure for the preparation of an aciloxialquilheterociclico compound. (Machine-translation by Google Translate, not legally binding) |
Country Status (11)
| Country | Link |
|---|---|
| AT (1) | AT301539B (en) |
| BE (1) | BE747274R (en) |
| CH (3) | CH554363A (en) |
| DE (1) | DE2012667C3 (en) |
| DK (1) | DK134023B (en) |
| ES (4) | ES377689A1 (en) |
| FI (1) | FI52088C (en) |
| NL (1) | NL7004067A (en) |
| NO (1) | NO128822B (en) |
| SE (1) | SE360869B (en) |
| SU (3) | SU420180A3 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GR65270B (en) * | 1978-10-10 | 1980-07-31 | Fujisawa Pharmaceutical Co | Isatin derivatives and processes for the preparation thereof |
| US4411900A (en) * | 1980-01-03 | 1983-10-25 | Fujisawa Pharmaceutical Co., Ltd. | Benzhydrylpiperozinyl thiazole derivatives and pharmaceutical composition comprising the same |
| FR2637286A1 (en) * | 1988-10-04 | 1990-04-06 | Adir | NOVEL BENZOXAZOLINON DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL108409C (en) * | 1958-10-29 |
-
1970
- 1970-03-12 BE BE747274D patent/BE747274R/en active
- 1970-03-13 FI FI68870A patent/FI52088C/en active
- 1970-03-17 DE DE19702012667 patent/DE2012667C3/en not_active Expired
- 1970-03-18 ES ES377689A patent/ES377689A1/en not_active Expired
- 1970-03-19 NO NO100670A patent/NO128822B/no unknown
- 1970-03-19 SE SE371670A patent/SE360869B/xx unknown
- 1970-03-19 AT AT259670A patent/AT301539B/en not_active IP Right Cessation
- 1970-03-20 SU SU1413002A patent/SU420180A3/en active
- 1970-03-20 CH CH1496673A patent/CH554363A/en not_active IP Right Cessation
- 1970-03-20 DK DK141070A patent/DK134023B/en unknown
- 1970-03-20 NL NL7004067A patent/NL7004067A/xx not_active Application Discontinuation
- 1970-03-20 CH CH427470A patent/CH565174A5/xx not_active IP Right Cessation
- 1970-03-20 SU SU1620557A patent/SU416947A3/en active
- 1970-03-20 CH CH1496773A patent/CH554364A/en not_active IP Right Cessation
- 1970-03-20 SU SU1620554A patent/SU400104A3/ru active
-
1972
- 1972-09-01 ES ES406298A patent/ES406298A1/en not_active Expired
- 1972-09-01 ES ES406297A patent/ES406297A1/en not_active Expired
- 1972-09-01 ES ES406296A patent/ES406296A1/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| SU400104A3 (en) | 1973-10-03 |
| SE360869B (en) | 1973-10-08 |
| DE2012667C3 (en) | 1981-11-26 |
| DE2012667B2 (en) | 1981-02-26 |
| ES406296A1 (en) | 1975-09-16 |
| AT301539B (en) | 1972-09-11 |
| FI52088C (en) | 1977-06-10 |
| CH565174A5 (en) | 1975-08-15 |
| BE747274R (en) | 1970-08-17 |
| DK134023C (en) | 1977-03-21 |
| DK134023B (en) | 1976-08-30 |
| DE2012667A1 (en) | 1970-10-01 |
| CH554363A (en) | 1974-09-30 |
| ES377689A1 (en) | 1973-01-01 |
| FI52088B (en) | 1977-02-28 |
| NL7004067A (en) | 1970-09-22 |
| SU420180A3 (en) | 1974-03-15 |
| CH554364A (en) | 1974-09-30 |
| SU416947A3 (en) | 1974-02-25 |
| ES406298A1 (en) | 1975-09-16 |
| NO128822B (en) | 1974-01-14 |
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