[go: up one dir, main page]

ES2586740A1 - Cyclic boamids with antifungal, antibiotic, antiviral and antitumor activity. (Machine-translation by Google Translate, not legally binding) - Google Patents

Cyclic boamids with antifungal, antibiotic, antiviral and antitumor activity. (Machine-translation by Google Translate, not legally binding) Download PDF

Info

Publication number
ES2586740A1
ES2586740A1 ES201530510A ES201530510A ES2586740A1 ES 2586740 A1 ES2586740 A1 ES 2586740A1 ES 201530510 A ES201530510 A ES 201530510A ES 201530510 A ES201530510 A ES 201530510A ES 2586740 A1 ES2586740 A1 ES 2586740A1
Authority
ES
Spain
Prior art keywords
antifungal
antibiotic
translation
cyclic
machine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES201530510A
Other languages
Spanish (es)
Other versions
ES2586740B1 (en
Inventor
Víctor TENA PÉREZ
Ángel RUMBERO SANCHEZ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
VICTOR TENA PEREZ
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Priority to ES201530510A priority Critical patent/ES2586740B1/en
Priority to PCT/EP2016/058396 priority patent/WO2016166319A1/en
Publication of ES2586740A1 publication Critical patent/ES2586740A1/en
Application granted granted Critical
Publication of ES2586740B1 publication Critical patent/ES2586740B1/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/04—Esters of boric acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention consists of the application of the cyclic boramide (figure 1) as antitumor and antimicrobial agent (antifungal, anti-hiv and antibiotic). It is a new structure based on the boron element (b) that consists of four rings of six fused members. In these, boron has a tetrahedral arrangement and forms an amide bond. The molecule is composed of the elements hydrogen (h), halides (cloro -cl-, bromo -br- and fluor-f-) or the radical methoxy (-ome) in the positions r3 and r'3 while the rest of r positions are composed of the hydrogen element (h). (Machine-translation by Google Translate, not legally binding)

Description

imagen1image 1

imagen2image2

imagen3image3

imagen4image4

imagen5image5

imagen6image6

imagen7image7

imagen8image8

imagen9image9

imagen10image10

imagen11image11

imagen12image12

imagen13image13

imagen14image14

imagen15image15

imagen16image16

imagen17image17

imagen18image18

Claims (1)

imagen1image 1 imagen2image2 imagen3image3 imagen4image4 imagen5image5 imagen6image6 imagen7image7 imagen8image8 imagen9image9
ES201530510A 2015-04-15 2015-04-15 Cyclic boramides with antifungal, antibiotic, antiviral and antitumor activity. Active ES2586740B1 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
ES201530510A ES2586740B1 (en) 2015-04-15 2015-04-15 Cyclic boramides with antifungal, antibiotic, antiviral and antitumor activity.
PCT/EP2016/058396 WO2016166319A1 (en) 2015-04-15 2016-04-15 Boramides for treating diseases

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES201530510A ES2586740B1 (en) 2015-04-15 2015-04-15 Cyclic boramides with antifungal, antibiotic, antiviral and antitumor activity.

Publications (2)

Publication Number Publication Date
ES2586740A1 true ES2586740A1 (en) 2016-10-18
ES2586740B1 ES2586740B1 (en) 2017-08-16

Family

ID=55754301

Family Applications (1)

Application Number Title Priority Date Filing Date
ES201530510A Active ES2586740B1 (en) 2015-04-15 2015-04-15 Cyclic boramides with antifungal, antibiotic, antiviral and antitumor activity.

Country Status (2)

Country Link
ES (1) ES2586740B1 (en)
WO (1) WO2016166319A1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111139189A (en) * 2020-01-14 2020-05-12 浙江工业大学 Aspergillus WBX-38 and application thereof in production of cyclopiazonic acid

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT109941B (en) 2017-03-02 2021-02-09 Hovione Farmaciência, S.A. MULTIFUNCTIONAL BORON CONJUGATES WITH A TRIPODAL STRUCTURE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PROCESSES FOR THE SAME

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013084199A1 (en) * 2011-12-07 2013-06-13 Universidade De Lisboa Boron heterocycles as new inhibitors of human neutrophil elastase

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111139189A (en) * 2020-01-14 2020-05-12 浙江工业大学 Aspergillus WBX-38 and application thereof in production of cyclopiazonic acid
CN111139189B (en) * 2020-01-14 2022-04-19 浙江工业大学 Aspergillus WBX-38 and application thereof in production of cyclopiazonic acid

Also Published As

Publication number Publication date
WO2016166319A1 (en) 2016-10-20
ES2586740B1 (en) 2017-08-16

Similar Documents

Publication Publication Date Title
EP3787734A4 (en) WEARABLE, ERGONOMIC NEUROSTIMULATION SYSTEM
JP2019046670A5 (en)
JP2019207083A5 (en)
ES2586740A1 (en) Cyclic boamids with antifungal, antibiotic, antiviral and antitumor activity. (Machine-translation by Google Translate, not legally binding)
JP2021062522A5 (en)
JP2019181899A5 (en)
JP2019094024A5 (en)
EP3361911A4 (en) PERMEABLE FOLDABLE MATTRESS
DK3886834T3 (en) PROCESSES FOR PREPARING NITROSYLATED PROPANEDIOLS, COMPOSITIONS COMPRISING THE SAME, AND MEDICAL USE THEREOF
JP2019058493A5 (en)
JP2021101083A5 (en)
JP2020175713A5 (en)
JP2020089637A5 (en)
JP2019183589A5 (en)
JP2019119952A5 (en)
EP4054790C0 (en) TOOLLESS ROTARY INDEXING TABLE ARRANGEMENT
FI12640U1 (en) Blowpipe
UA45180S (en) 1.-2. SUBWOOFER
JP2021101084A5 (en)
TH184370S (en) pillow
UA118271U (en) INFORMATION SYSTEM
RU2018141495A (en) ANTIDEPRESSANT
TH188432S (en) Headphones
JP2019058494A5 (en)
RU2018139641A (en) CELL LINE IN SUSPENSION

Legal Events

Date Code Title Description
PC2A Transfer of patent

Owner name: VICTOR TENA PEREZ

Effective date: 20150817

FG2A Definitive protection

Ref document number: 2586740

Country of ref document: ES

Kind code of ref document: B1

Effective date: 20170816