ES2373901A1 - Energizing composition and dietetic supplement that contains it. (Machine-translation by Google Translate, not legally binding) - Google Patents

Abstract

Energizing composition and dietary supplement that contains it. The present invention describes a new energizing and revitalizing composition comprising: 1.82% -59.76% vitamin c; 0.34% -40.87% thiamine hydrochloride; 0.34% -40.87% pyridoxine hydrochloride; 1.89% -51.00 of N-acetyl-l-cysteine; 3.82% -61.41% l-asparagine; 0.21% -30.34% vitamin e; 0.38% -43.54% l-glutamic acid; and 0.32% -11.73% caffeine. The composition is useful for the preparation of a dietary or nutritional supplement such as a beverage. The food supplement obtained has antioxidant properties and hepato-, neuro- and nephroprotective effects. (Machine-translation by Google Translate, not legally binding)

Description

Energizing composition and dietary supplement that contains it.

Field of the Invention

The present invention fits within the field of energizing and revitalizing products intended for human consumption in general, and more particularly in situations of high physical and / or mental performance.

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Background of the invention

Various are known in the state of the art energetic and revitalizing compositions, particularly in form of drinks. Among the many drinks that exist in the market It is worth mentioning, for example, the Red Bull ® drink.

The composition of this product contains: water, saccharin and sugars, such as glucose; glucuronolactone, which it consists of a derivative of glucose that is part of the tissue connective; stimulants, such as taurine, an amino acid; Caffeine in an amount of 32 mg / 100 cc equivalent to one cup of coffee expresso and vitamins of group B, such as niacin (vitamin B3), the pantothenic acid (vitamin B5), and vitamins B6 and B12.

These components are characterized by their Different functionalities Thus, hydrocarbon substrates they provide energy; the stimulants are psychostimulants and metabolism accelerators; and the vitamins of group B are all of them related to metabolism so that they optimize the increase in metabolic speed in a very general way.

According to the manufacturers of these drinks, these have a revitalizing and detoxifying effect as well as properties that increase physical capabilities and enhance the mental speed It is therefore functional drinks, not to remove thirst, which have been designed for consumption in moments of high physical and mental demand; such as during driving on very long highways that can induce sleep, on a lot of work days, before practicing a lot of activity physical wear or before an exam.

However this type of energy drinks in In general, they have a significant disadvantage and they produce a increased metabolism, which inexorably leads to increased production of free radicals and therefore at a imbalance in oxidative metabolism.

In this sense the need still exists in the state of the art of providing an alternative composition that satisfactorily meets the desirable properties of this type of energizing and revitalizing compositions without the Associated disadvantage mentioned.

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Description of the invention

The present invention relates in one aspect to a new composition that includes:

1.82% -59.76% of vitamin C;

0.34% -40.87% of thiamine hydrochloride;

0.34% -40.87% of pyridoxine hydrochloride;

1.89% -51.00 of N-acetyl-L-cysteine;

3.82% -61.41% of L-asparagine;

0.21% -30.34% of Vitamin E;

0.38% -43.54% of L-glutamic acid; Y

0.32% -11.73% of caffeine.

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The components that are used for the Preparation of the composition of the invention can be found in neutral form or pharmaceutically acceptable derivative salts. The Vitamin E can be in principle any of the 8 ways called tocopherols or trocotrienols, preferably α-tocopherol. The composition of the invention. It is prepared in a simple way by a procedure that includes The mixture of the ingredients.

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In a particular embodiment the composition understands:

15.65% of vitamin C;

9.39% of thiamine hydrochloride;

9.39% of pyridoxine hydrochloride;

18.79% of N-acetyl-L-cysteine;

21.29% of L-asparagine;

4.17% of Vitamin E;

18.79% acid L-glutamic; Y

2.50% of caffeine.

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This composition, hereinafter the composition of the invention, provides biological substrates that optimize routes important metabolic in energy metabolism, all mediated by the improvement of the redox balance, favoring an environment reducer in the cell cytoplasm.

An advantage of the composition of the invention resides in that its stimulating effect, with the use of accelerators metabolic of group B vitamin group (vitamin B1 and vitamin B6) along with caffeine and amino acids, such as asparagine and L-glutamic acid, is found balanced with a very powerful antioxidant composition based on N-acetyl-Cysteine, vitamin C and Vitamin E.

In comparison to other compositions state of the art energizers considered stimulants and metabolic accelerators, the composition of the present invention consists of a metabolic balancer in high situations performance. In this sense the antioxidant composition gives it to the composition of the invention properties that are extremely beneficial in situations of metabolic stress both physical and psychic, as are their ability to protect organs especially sensitive to oxidative imbalance (nervous system central, liver, kidneys), although it is clear that their ability to performance at the level of organs and devices is systemic, that is, widespread throughout the economy.

Therefore in another aspect the composition is relates to its use in the preparation of a dietary supplement or energizing or revitalizing food composition with antioxidant, neuroprotective, hepatoprotective and Nephroprotective as well as anti-aging.

In a further aspect the invention relates to a dietary supplement or food composition comprising the composition of the invention Said dietary supplement or food composition, hereinafter supplement of the invention, it comprises a quantity of the composition of the invention and a pharmaceutically acceptable excipient or vehicle combinable with said composition that has no adverse effect on the treated organism The supplement of the invention may comprise excipients such as fructose, water, aromas, dyes, etc.

Preferably the composition of the invention is present in the supplement of the invention in an amount effective to provide an antioxidant effect, as well as neuro-, hepato- and nephroprotective in a mammal, in particular a human. He vehicle or excipient must be pharmaceutically tolerable, Combinable with the composition of the invention and having no effect adverse on the treated organism. The supplement can present in the form of unit doses. It is prepared according to procedures well known in the state of the art in the field of pharmacology and / or food. The appropriate amount of composition of the invention included in the supplement of the invention may vary depending on the nature of the supplement of so that in general this is between 5 and 95% by weight with respect to the total weight of the supplement.

The supplement of the invention may be adapted for oral administration in liquid or solid form. It can be among others a drink, or a candy, a gum etc. In a particular embodiment the supplement of the invention consists of a drink comprising fructose as an excipient.

The supplement can have any form Regular pharmacist adapted to your oral administration. The excipients in each case and their preparation procedure are well known to a person skilled in the art. Between the ways of oral administration include tablets, tablets optionally film coated, effervescent powders, suspensions, syrups, ampoules, etc.

In a particular embodiment the supplement of The invention comprises:

50 mg to 4 gr of vitamin C,

10 mg to 2 gr of thiamine hydrochloride;

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10 mg to 2 gr of pyridoxine hydrochloride;

50 mg to 2.7 gr of N-acetyl cysteine;

100 mg to 4 gr of L-asparagine;

10 Ul to 4 gr (2000 Ul) of vitamin E (alpha-tocopherol);

10 mg to 2 gr of L-glutamic acid;

10 mg to 600 mg of caffeine; Y

between 0.00 and 70 gr of fructose

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In a preferred embodiment the supplement of The invention comprises:

500 mg of vitamin C,

300 mg of thiamine hydrochloride;

300 mg of pyridoxine hydrochloride;

600 mg of N-acetyl cysteine;

680 mg of L-asparagine;

200 ul of vitamin E (alpha-tocopherol);

600 mg of acid L-glutamic;

80 mg of caffeine.

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In another more preferred embodiment the supplement it presents, in addition to these indicated quantities, 25 gr of fructose.

In another particular embodiment the supplement of the invention is a liquid composition, preferably in the form of a drink of typically 200-250 ml.

Below are examples illustrative of the invention set forth for a better understanding of the invention and in no case should be considered a Limitation of its scope.

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Examples Example 1

Unit composition of 250 ml drinkable according to invention comprising:

500 mg of vitamin C,

300 mg of thiamine hydrochloride;

300 mg of pyridoxine hydrochloride;

600 mg of N-acetyl cysteine;

680 mg of L-asparagine;

200 ul of vitamin E (α-tocopherol);

600 mg of acid L-glutamic;

80 mg of caffeine; Y

25 grams of fructose.

Claims (9)

1. New composition comprising:

1.82% -59.76% of vitamin C;

0.34% -40.87% of thiamine hydrochloride;

0.34% -40.87% of pyridoxine hydrochloride;

1.89% -51.00 of N-acetyl-L-cysteine;

3.82% -61.41% of L-asparagine;

0.21% -30.34% of Vitamin E;

0.38% -43.54% of L-glutamic acid; Y

0.32% -11.73% of caffeine.

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2. Composition according to claim 1, in the that the composition comprises:

15.65% of vitamin C;

9.39% of thiamine hydrochloride;

9.39% of pyridoxine hydrochloride;

18.79% of N-acetyl-L-cysteine;

21.29% of L-asparagine;

4.17% of Vitamin E;

18.79% acid L-glutamic; Y

2.50% of caffeine.

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3. Use of the composition according to any one of claims 1 or 2, in the preparation of a supplement dietary. 4. Dietary supplement comprising the composition according to any one of claims 1 or 2, and at less a pharmaceutically acceptable excipient. 5. Dietary supplement comprising:

50 mg to 4 gr of vitamin C,

10 mg to 2 gr of thiamine hydrochloride;

10 mg to 2 gr of pyridoxine hydrochloride;

50 mg to 2.7 gr of N-acetyl cysteine;

100 mg to 4 gr of L-asparagine;

10 Ul to 4 gr (2000 Ul) of vitamin E (alpha-tocopherol);

10 mg to 2 gr of L-glutamic acid;

10 mg to 600 mg of caffeine

and optionally between 0.00 mg and 70 mg of fructose.

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6. Supplement according to claim 5 that understands:

500 mg of vitamin C,

300 mg of thiamine hydrochloride;

300 mg of pyridoxine hydrochloride;

600 mg of N-acetyl cysteine;

680 mg of L-asparagine;

200 ul of vitamin E (alpha-tocopherol);

600 mg of acid L-glutamic;

80 mg of caffeine and optionally 25 mg of fructose.

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7. Supplement according to claim 6 that It consists of 250 ml of drinkable unit composition. 8. Supplement according to claim 4 or 5, in form of a drink, a candy, a gum or a form of liquid or solid oral administration. 9. Supplement according to claim 4 or 5 in which the supplement is selected from among a dragee, a compressed, optionally film coated, powders Effervescent, suspension, syrup, and blister.