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ES2365815T3 - Análogos de arilpropionamida, arilacrilamida, arilpropinamida o arilmetilurea como inhibidores del factor xia. - Google Patents

Análogos de arilpropionamida, arilacrilamida, arilpropinamida o arilmetilurea como inhibidores del factor xia. Download PDF

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Publication number
ES2365815T3
ES2365815T3 ES06846594T ES06846594T ES2365815T3 ES 2365815 T3 ES2365815 T3 ES 2365815T3 ES 06846594 T ES06846594 T ES 06846594T ES 06846594 T ES06846594 T ES 06846594T ES 2365815 T3 ES2365815 T3 ES 2365815T3
Authority
ES
Spain
Prior art keywords
dome
base
housing
antenna
arilpropionamida
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
ES06846594T
Other languages
English (en)
Inventor
Donald J.P. Pinto
Joanne M. Smallheer
James R. Corte
Zilun Hu
Cullen L. Cavallaro
Paul J. Gilligan
Mimi L. Quan
Leon M. Smith Ii
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of ES2365815T3 publication Critical patent/ES2365815T3/es
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Casings For Electric Apparatus (AREA)

Abstract

Un sistema de filtración que comprende: a) un domo (40) de la carcasa conductor eléctrico; b) un conjunto filtrante, que comprende circuitos electrónicos; c) una base (70) de la carcasa; d) una junta aislante eléctricamente (60) interpuesta entre el citado domo (40) y la citada base (70) con el fin de mantenerlos aislados física y eléctricamente; e) un medio para asegurar juntos el citado domo (40), la citada junta (60) y la citada base (70), con el fin de crear una obturación estanca a los líquidos, en el que el citado medio mantiene el aislamiento eléctrico entre el citado domo (40) y la citada base (70 ), y f) un dispositivo externo (100), que incluye una antena, estando el citado domo (40) de la carcasa en comunicación eléctrica con un polo de la citada antena, por medio de lo cual el citado domo (40) de la carcasa conductor eléctrico sirve como una antena por lo que puede transmitir señales desde el citado dispositivo al citado circuito electrónico.
ES06846594T 2005-12-14 2006-12-13 Análogos de arilpropionamida, arilacrilamida, arilpropinamida o arilmetilurea como inhibidores del factor xia. Active ES2365815T3 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US75013005P 2005-12-14 2005-12-14
US750130P 2005-12-14
US821163P 2006-08-02
US865211P 2006-11-10

Publications (1)

Publication Number Publication Date
ES2365815T3 true ES2365815T3 (es) 2011-10-11

Family

ID=40214768

Family Applications (1)

Application Number Title Priority Date Filing Date
ES06846594T Active ES2365815T3 (es) 2005-12-14 2006-12-13 Análogos de arilpropionamida, arilacrilamida, arilpropinamida o arilmetilurea como inhibidores del factor xia.

Country Status (3)

Country Link
CN (1) CN101341129B (es)
ES (1) ES2365815T3 (es)
ZA (1) ZA200805028B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110097666A1 (en) * 2009-10-27 2011-04-28 Celin Savariar-Hauck Lithographic printing plate precursors
PH12012501589A1 (en) 2010-02-11 2012-10-22 Bristol Myers Squibb Co Macrocycles as factor xia inhibitors
GB2494851A (en) * 2011-07-07 2013-03-27 Kalvista Pharmaceuticals Ltd Plasma kallikrein inhibitors
JP6137193B2 (ja) * 2011-12-21 2017-05-31 小野薬品工業株式会社 第XIa因子阻害剤としての新規ピリジノンおよびピリミジノン誘導体
WO2015011087A1 (de) * 2013-07-23 2015-01-29 Bayer Pharma Aktiengesellschaft Substituierte oxopyridin-derivate und ihre verwendung als faktor xia / plasma
CN112028877B (zh) * 2019-06-04 2021-11-26 江西济民可信集团有限公司 烷氧吡啶酮化合物及其制备方法和用途
EP4036087A4 (en) * 2019-09-27 2023-09-20 Shenzhen Salubris Pharmaceuticals Co. Ltd Fxia inhibitors and preparation method therefor and pharmaceutical use thereof
CN117480164B (zh) * 2020-12-11 2024-07-05 上海领泰生物医药科技有限公司 凝血因子XIa抑制剂及其制备方法和应用
TW202246219A (zh) * 2021-03-18 2022-12-01 大陸商深圳信立泰藥業股份有限公司 FXIa抑制劑化合物雜質、其製備方法及其用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU746963B2 (en) * 1998-06-12 2002-05-09 Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) Imidazolyl derivatives
CN1200000C (zh) * 1998-06-16 2005-05-04 研究及应用科学协会股份有限公司 促生长素抑制素类似物
WO2003064440A1 (de) * 2002-01-31 2003-08-07 Morphochem Aktiengesellschaft für kombinatorische Chemie Verbindungen, die faktor xa-aktivät inhibieren
US7371743B2 (en) * 2004-02-28 2008-05-13 Boehringer Ingelheim International Gmbh Carboxylic acid amides, the preparation thereof and their use as medicaments
US7417063B2 (en) * 2004-04-13 2008-08-26 Bristol-Myers Squibb Company Bicyclic heterocycles useful as serine protease inhibitors

Also Published As

Publication number Publication date
ZA200805028B (en) 2009-12-30
CN101341129A (zh) 2009-01-07
CN101341129B (zh) 2011-12-14

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