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ES2137170T3 - PROCEDURE FOR PREPARING ALPHA, ALPHA-DISPUTED AROMATIC AND HETEROAROMATIC COMPOUNDS FOR THE IMPROVEMENT OF COGNITIVE FUNCTIONS. - Google Patents

PROCEDURE FOR PREPARING ALPHA, ALPHA-DISPUTED AROMATIC AND HETEROAROMATIC COMPOUNDS FOR THE IMPROVEMENT OF COGNITIVE FUNCTIONS.

Info

Publication number
ES2137170T3
ES2137170T3 ES92115889T ES92115889T ES2137170T3 ES 2137170 T3 ES2137170 T3 ES 2137170T3 ES 92115889 T ES92115889 T ES 92115889T ES 92115889 T ES92115889 T ES 92115889T ES 2137170 T3 ES2137170 T3 ES 2137170T3
Authority
ES
Spain
Prior art keywords
alpha
aromatic
disputed
improvement
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES92115889T
Other languages
Spanish (es)
Inventor
Richard Alan Earl
Melvyn John Myers
Victor Johannes Nickolson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Pharma Co
Original Assignee
DuPont Merck Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/234,382 external-priority patent/US5173489A/en
Application filed by DuPont Merck Pharmaceutical Co filed Critical DuPont Merck Pharmaceutical Co
Application granted granted Critical
Publication of ES2137170T3 publication Critical patent/ES2137170T3/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

SE TRATAN LAS DEFICIENCIAS COGNITIVAS O LA DISFUNCION NEUROLOGICA CON COMPUESTOS O,O-DISUBSTITUIDOS AROMATICOS Y HETERAROMATICOS. LOS COMPUESTOS TIENEN LA FORMULA: O SU SAL EN DONDE X E Y SE TOMAN JUNTOS PARA FORMAR UN PRIMER ANILLO CARBOCICLICO O HETEROCICLICO SATURADO O NO SATURADO Y EL CARBONO MOSTRADO EN DICHO ANILLO ES O RESPECTO, AL MENOS, A UN ANILLO AROMATICO ADICIONAL O A UN ANILLO HETERAROMATICO UNIDO AL PRIMER ANILLO; UNO DE HET1 O HET2 ES 2, 3, O 4 INILO Y EL OTRO SE SELECCIONA A PARTIR DE (A) 2, 3, O 4 DILO (B) 2, 4, O 5 4 ROFURANILO, Y (G) 3 - TIENILO.COGNITIVE DEFICIENCIES OR NEUROLOGICAL DYSFUNCTION WITH COMPOUNDS OR, O-DISUBSTITUTED AROMATIC AND HETERAROMATIC. THE COMPOUNDS HAVE THE FORMULA: OR THEIR SALT WHERE XEY IS TAKEN TOGETHER TO FORM A FIRST CARBON CYCLE OR HETERO-CYCLE RING SATURATED OR NOT SATURATED AND THE CARBON SHOWN IN SUCH A RING ANOIL AROAIL AROIL ATTACHED TO THE FIRST RING; ONE OF HET1 OR HET2 IS 2, 3, OR 4 INIL AND THE OTHER IS SELECTED FROM (A) 2, 3, OR 4 DILO (B) 2, 4, OR 5 4 ROFURANILO, AND (G) 3 - TIENYL .

ES92115889T 1987-10-06 1988-10-04 PROCEDURE FOR PREPARING ALPHA, ALPHA-DISPUTED AROMATIC AND HETEROAROMATIC COMPOUNDS FOR THE IMPROVEMENT OF COGNITIVE FUNCTIONS. Expired - Lifetime ES2137170T3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10515687A 1987-10-06 1987-10-06
US07/234,382 US5173489A (en) 1986-04-10 1988-08-23 α,α-disubstituted aromatics and heteroaromatics as cognition enhancers
EP88116393A EP0311010B1 (en) 1987-10-06 1988-10-04 Alpha,Alpha-disubstituted aromatics and heteroaromatics as cognition enhancers

Publications (1)

Publication Number Publication Date
ES2137170T3 true ES2137170T3 (en) 1999-12-16

Family

ID=27231322

Family Applications (1)

Application Number Title Priority Date Filing Date
ES92115889T Expired - Lifetime ES2137170T3 (en) 1987-10-06 1988-10-04 PROCEDURE FOR PREPARING ALPHA, ALPHA-DISPUTED AROMATIC AND HETEROAROMATIC COMPOUNDS FOR THE IMPROVEMENT OF COGNITIVE FUNCTIONS.

Country Status (3)

Country Link
AT (1) ATE101148T1 (en)
ES (1) ES2137170T3 (en)
GR (1) GR3031080T3 (en)

Also Published As

Publication number Publication date
GR3031080T3 (en) 1999-12-31
ATE101148T1 (en) 1994-02-15

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