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ES2160955T3 - Derivados del acido 4-arilbutirico sustituido como inhibidores de la metaloproteasa de matriz. - Google Patents

Derivados del acido 4-arilbutirico sustituido como inhibidores de la metaloproteasa de matriz.

Info

Publication number
ES2160955T3
ES2160955T3 ES97923625T ES97923625T ES2160955T3 ES 2160955 T3 ES2160955 T3 ES 2160955T3 ES 97923625 T ES97923625 T ES 97923625T ES 97923625 T ES97923625 T ES 97923625T ES 2160955 T3 ES2160955 T3 ES 2160955T3
Authority
ES
Spain
Prior art keywords
ilo
rent
phenyl
bencilo
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES97923625T
Other languages
English (en)
Inventor
Harold C E Kluender
Brian R Dixon
David R Brittelli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Bayer Corp
Original Assignee
Bayer AG
Bayer Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG, Bayer Corp filed Critical Bayer AG
Application granted granted Critical
Publication of ES2160955T3 publication Critical patent/ES2160955T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/76Unsaturated compounds containing keto groups
    • C07C59/84Unsaturated compounds containing keto groups containing six membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/76Unsaturated compounds containing keto groups
    • C07C59/90Unsaturated compounds containing keto groups containing singly bound oxygen-containing groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/30Phthalazines
    • C07D237/32Phthalazines with oxygen atoms directly attached to carbon atoms of the nitrogen-containing ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D253/00Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/041,2,3-Triazines

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

LA INVENCION SE REFIERE A INHIBIDORES DE LA METALOPROTEASA DE LA MATRIZ, A COMPOSICIONES FARMACEUTICAS QUE LOS CONTIENEN, Y A UN PROCEDIMIENTO DE UTILIZACION DE LOS MISMOS PARA TRATAR DIVERSOS ESTADOS FISIOLOGICOS. LOS COMPUESTOS DE LA INVENCION PRESENTAN LA FORMULA GENERAL (I), DONDE R 1 REPRESENTA ALQUILO C 6 C 12 ; ALCOXI C 5 - C 12 ; ALQUILT IO C 5 C 12 ; UN POLIETER DE FORMULA R 2 O(C 2 H 4 O) A -, EN DONDE A ES 1 O 2; Y R 2 ES ALQU ILO C 1 - C 5 , FENILO O BENCILO; Y ALQUINILO SUSTITUIDO DE FORMULA R 3 (CH 2 ) B - C C -; EN DONDE B ES 1-10 Y R 3 ES H -, HO - O R 4 O -, EN DONDE R 4 ES ALQUILO C 1 - C 3 , FENILO O BENCILO. LAS FRACC IONES ALQUILO, FENILO Y BENCILO DE R 1 PUEDEN LLEVAR AL MENOS UN SUSTITUYENTE FARMACEUTICAMENTE ACEPTABLE. EL SUBINDICE N ES 2-4. R 5 REPRESENTA FENILO; IMIDOILO DE 4-12 ATOMOS DE CARBONO; (3H) - BENZO - 1,2,3 - TRIAZIN - 4 - ON - 3 - ILO; N - SACARINILO; (2H) - FTALACIN - 1 -ON - 2 - ILO; 2 - BENZOXAZOLIN - 2 - ON - 3 ILO; 5,5 - DIMETILOXAZOLIDINA - 2,4 -DION - 3 - ILO; Y TIAZOLIDIN 2,4 - DION - 3 - ILO; PUDIENDO LLEVAR LAS FRACCIONES FENILO Y BENZO DE R 5 AL MENOS UN SUSTITUYENTE FARMACEUTICAMENTE ACEPTABLE. SE INCLUYEN ASIMISMO LAS SALES FARMACEUTICAMENTE ACEPTABLES DE DICHOS MATERIALES.
ES97923625T 1996-05-15 1997-05-12 Derivados del acido 4-arilbutirico sustituido como inhibidores de la metaloproteasa de matriz. Expired - Lifetime ES2160955T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US64768296A 1996-05-15 1996-05-15

Publications (1)

Publication Number Publication Date
ES2160955T3 true ES2160955T3 (es) 2001-11-16

Family

ID=24597888

Family Applications (1)

Application Number Title Priority Date Filing Date
ES97923625T Expired - Lifetime ES2160955T3 (es) 1996-05-15 1997-05-12 Derivados del acido 4-arilbutirico sustituido como inhibidores de la metaloproteasa de matriz.

Country Status (21)

Country Link
EP (1) EP0923529B1 (es)
JP (1) JP3354941B2 (es)
CN (1) CN1225620A (es)
AR (1) AR007101A1 (es)
AT (1) ATE205822T1 (es)
AU (1) AU727468B2 (es)
BR (1) BR9709075A (es)
CA (1) CA2253795C (es)
CO (1) CO5011113A1 (es)
DE (1) DE69706874T2 (es)
ES (1) ES2160955T3 (es)
HR (1) HRP970247B1 (es)
ID (1) ID17326A (es)
MY (1) MY116903A (es)
PA (1) PA8429501A1 (es)
SV (1) SV1997000033A (es)
TN (1) TNSN97086A1 (es)
TW (1) TW442468B (es)
WO (1) WO1997043237A1 (es)
YU (1) YU18897A (es)
ZA (1) ZA974033B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CO5080759A1 (es) 1996-05-15 2001-09-25 Bayer Corp Biarilacetilenos como inhibidores de la metaloproteasa de matriz
US6288063B1 (en) 1998-05-27 2001-09-11 Bayer Corporation Substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors
FR2832925B1 (fr) * 2001-12-03 2006-07-14 Lipha Utilisation de derives de l'acide 4-oxobutanoique dans le traitement de l'inflammation
JP2012087113A (ja) * 2010-09-22 2012-05-10 Daicel Corp フェニル酢酸化合物
EP3126340A2 (de) 2014-04-03 2017-02-08 Bayer Pharma Aktiengesellschaft Chirale 2,5-disubstituierte cyclopentancarbonsäure-derivate und ihre verwendung
CA2944614A1 (en) 2014-04-03 2015-10-08 Bayer Pharma Aktiengesellschaft 2,5-disubstituted cyclopentane carboxylic acids for the treatment of respiratoy tract diseases
WO2015150363A1 (de) 2014-04-03 2015-10-08 Bayer Pharma Aktiengesellschaft 2,5-disubstituierte cyclopentancarbonsäuren und ihre verwendung
WO2015150364A1 (de) * 2014-04-03 2015-10-08 Bayer Pharma Aktiengesellschaft Substituierte benzotriazinonbutansäuren und ihre verwendung
US20170121315A1 (en) * 2014-06-12 2017-05-04 Bayer Pharma Aktiengesellschaft Heterobicyclically substituted 4-oxobutane acid derivatives and use thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE650081A (es) * 1963-07-03
FR2378741A1 (fr) * 1977-02-01 1978-08-25 Fabre Sa Pierre Acides garyl goxo isovaleriques doues de proprietes antiphlogistiques et antalgiques
JP2000502343A (ja) 1995-12-22 2000-02-29 ワーナー―ランバート・コンパニー マトリックスメタロプロテイナーゼのインヒビターとしての芳香族ケト酸およびその誘導体
TNSN97081A1 (fr) 1996-05-15 2005-03-15 Bayer Corp Inhibition des matrices metalloproteinases par 2- (w-aroylkyl) -4-biaryl-4-des acides oxubutyriques

Also Published As

Publication number Publication date
JPH11510518A (ja) 1999-09-14
CO5011113A1 (es) 2001-02-28
SV1997000033A (es) 1999-01-14
ID17326A (id) 1997-12-18
PA8429501A1 (es) 2000-05-24
HRP970247A2 (en) 1998-04-30
YU18897A (en) 1999-11-22
DE69706874T2 (de) 2002-03-28
JP3354941B2 (ja) 2002-12-09
HRP970247B1 (en) 2002-02-28
WO1997043237A1 (en) 1997-11-20
ZA974033B (en) 1998-02-19
ATE205822T1 (de) 2001-10-15
EP0923529B1 (en) 2001-09-19
TNSN97086A1 (fr) 2005-03-15
AU727468B2 (en) 2000-12-14
AR007101A1 (es) 1999-10-13
TW442468B (en) 2001-06-23
AU2938997A (en) 1997-12-05
CA2253795A1 (en) 1997-11-20
CA2253795C (en) 2002-10-15
DE69706874D1 (en) 2001-10-25
MY116903A (en) 2004-04-30
BR9709075A (pt) 1999-08-03
EP0923529A1 (en) 1999-06-23
CN1225620A (zh) 1999-08-11

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