ES2031854T3 - Nuevos acidos 4-quinoloncarboxilicos 1,8-puenteados y medicamentos que les contienen. - Google Patents
Nuevos acidos 4-quinoloncarboxilicos 1,8-puenteados y medicamentos que les contienen.Info
- Publication number
- ES2031854T3 ES2031854T3 ES198787109593T ES87109593T ES2031854T3 ES 2031854 T3 ES2031854 T3 ES 2031854T3 ES 198787109593 T ES198787109593 T ES 198787109593T ES 87109593 T ES87109593 T ES 87109593T ES 2031854 T3 ES2031854 T3 ES 2031854T3
- Authority
- ES
- Spain
- Prior art keywords
- bridged
- quinoloncarboxilicos
- drugs
- contain
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000002253 acid Substances 0.000 title 1
- 150000007513 acids Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- YCAZALSUJDPQPP-UHFFFAOYSA-N 4-oxo-3h-quinoline-3-carboxylic acid Chemical class C1=CC=C2C(=O)C(C(=O)O)C=NC2=C1 YCAZALSUJDPQPP-UHFFFAOYSA-N 0.000 abstract 1
- DFPAKSUCGFBDDF-UHFFFAOYSA-N Nicotinamide Chemical group NC(=O)C1=CC=CN=C1 DFPAKSUCGFBDDF-UHFFFAOYSA-N 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 125000004185 ester group Chemical group 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 125000002560 nitrile group Chemical group 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Quinoline Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Fodder In General (AREA)
Abstract
LA INVENCION SE REFIERE A NUEVOS ACIDOS 4-QUINOLON-3-CARBOXILICOS, PUENTEADOS EN 1,8 Y DERIVADOS DE LA FORMULA (I), EN LA QUE Y, X1, X5, R10 Y R11 TIENEN LA SIGNIFICACION ASIGNADA EN LA DESCRIPCION, AL METODO DE SU OBTENCION, ASI COMO A SU APLICACION COMO MEDICAMENTOS, ESPECIALMENTE COMO ANTIBACTERIANOS, TANTO EN MEDICINA HUMANA COMO VETERINARIA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3623757A DE3623757A1 (de) | 1986-07-15 | 1986-07-15 | Neue 1,8-verbrueckte 4-chinoloncarbonsaeuren und diese enthaltende arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2031854T3 true ES2031854T3 (es) | 1993-01-01 |
Family
ID=6305168
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES198787109593T Expired - Lifetime ES2031854T3 (es) | 1986-07-15 | 1987-07-03 | Nuevos acidos 4-quinoloncarboxilicos 1,8-puenteados y medicamentos que les contienen. |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US4816451A (es) |
| EP (1) | EP0253235B1 (es) |
| JP (1) | JPS6339880A (es) |
| AT (1) | ATE59654T1 (es) |
| DE (2) | DE3623757A1 (es) |
| ES (1) | ES2031854T3 (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0228178A (ja) * | 1988-04-23 | 1990-01-30 | Toyama Chem Co Ltd | 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法 |
| DE3902079A1 (de) * | 1988-04-15 | 1989-10-26 | Bayer Ag | I.m. injektionsformen von gyrase-inhibitoren |
| US4992449A (en) * | 1990-02-01 | 1991-02-12 | American Cyanamid Company | 7-(substituted)cycloalkylamino-1-(substituted)-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids |
| DE4210941A1 (de) * | 1992-04-02 | 1993-10-07 | Bayer Ag | Neue 9-Fluor-7.oxo-7H-pyrido[1,2,3-d,e][1,4]benzoxacin-6-carbonsäuren und -ester |
| DE4210942A1 (de) * | 1992-04-02 | 1993-10-07 | Bayer Ag | 7-Oxo-7H-pyrido[1,2,3-d,e][1,4]benzoxacin-6-carbonsäuren und -ester |
| DE4210939A1 (de) * | 1992-04-02 | 1993-10-07 | Bayer Ag | Verwendung von 7-Oxo-7H-pyrido[1,2,3-de][1,4]benzoxacin-6-carbonsäuren und -estern als Arzneimittel |
| US6022551A (en) * | 1998-01-20 | 2000-02-08 | Ethicon, Inc. | Antimicrobial composition |
| US5972358A (en) * | 1998-01-20 | 1999-10-26 | Ethicon, Inc. | Low tack lotion, gels and creams |
| US5997893A (en) * | 1998-01-20 | 1999-12-07 | Ethicon, Inc. | Alcohol based anti-microbial compositions with cosmetic appearance |
| US6248343B1 (en) | 1998-01-20 | 2001-06-19 | Ethicon, Inc. | Therapeutic antimicrobial compositions |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5746986A (en) * | 1980-09-02 | 1982-03-17 | Dai Ichi Seiyaku Co Ltd | Pyrido(1,2,3-de)(1,4)benzoxazine derivative |
| DE3522405A1 (de) * | 1985-06-22 | 1987-01-02 | Bayer Ag | 1,8-verbrueckte 4-chinolon-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende arzneimittel und ihre verwendung zur herstellung von arzneimitteln |
-
1986
- 1986-07-15 DE DE3623757A patent/DE3623757A1/de not_active Withdrawn
-
1987
- 1987-06-29 US US07/068,074 patent/US4816451A/en not_active Expired - Fee Related
- 1987-07-03 ES ES198787109593T patent/ES2031854T3/es not_active Expired - Lifetime
- 1987-07-03 DE DE8787109593T patent/DE3766903D1/de not_active Expired - Lifetime
- 1987-07-03 AT AT87109593T patent/ATE59654T1/de not_active IP Right Cessation
- 1987-07-03 EP EP87109593A patent/EP0253235B1/de not_active Expired - Lifetime
- 1987-07-15 JP JP62174999A patent/JPS6339880A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| DE3623757A1 (de) | 1988-01-21 |
| JPS6339880A (ja) | 1988-02-20 |
| EP0253235A1 (de) | 1988-01-20 |
| EP0253235B1 (de) | 1991-01-02 |
| ATE59654T1 (de) | 1991-01-15 |
| DE3766903D1 (de) | 1991-02-07 |
| US4816451A (en) | 1989-03-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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