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EP3177365A4 - Agonistes de la voie du récepteur ahr ayant une activité sébosuppressive et procédé d'identification desdits agonistes - Google Patents

Agonistes de la voie du récepteur ahr ayant une activité sébosuppressive et procédé d'identification desdits agonistes Download PDF

Info

Publication number
EP3177365A4
EP3177365A4 EP15830204.2A EP15830204A EP3177365A4 EP 3177365 A4 EP3177365 A4 EP 3177365A4 EP 15830204 A EP15830204 A EP 15830204A EP 3177365 A4 EP3177365 A4 EP 3177365A4
Authority
EP
European Patent Office
Prior art keywords
agonists
identifying
receptor pathway
ahr receptor
sebosuppressive activity
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP15830204.2A
Other languages
German (de)
English (en)
Other versions
EP3177365A1 (fr
Inventor
Jean Hilaire Saurat
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
THESAN PHARMACEUTICALS Inc
Original Assignee
THESAN PHARMACEUTICALS Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by THESAN PHARMACEUTICALS Inc filed Critical THESAN PHARMACEUTICALS Inc
Publication of EP3177365A1 publication Critical patent/EP3177365A1/fr
Publication of EP3177365A4 publication Critical patent/EP3177365A4/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/08—Antiseborrheics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EP15830204.2A 2014-08-06 2015-08-05 Agonistes de la voie du récepteur ahr ayant une activité sébosuppressive et procédé d'identification desdits agonistes Withdrawn EP3177365A4 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462034005P 2014-08-06 2014-08-06
US201462041751P 2014-08-26 2014-08-26
PCT/US2015/043833 WO2016022703A1 (fr) 2014-08-06 2015-08-05 Agonistes de la voie du récepteur ahr ayant une activité sébosuppressive et procédé d'identification desdits agonistes

Publications (2)

Publication Number Publication Date
EP3177365A1 EP3177365A1 (fr) 2017-06-14
EP3177365A4 true EP3177365A4 (fr) 2018-01-10

Family

ID=55264515

Family Applications (1)

Application Number Title Priority Date Filing Date
EP15830204.2A Withdrawn EP3177365A4 (fr) 2014-08-06 2015-08-05 Agonistes de la voie du récepteur ahr ayant une activité sébosuppressive et procédé d'identification desdits agonistes

Country Status (2)

Country Link
EP (1) EP3177365A4 (fr)
WO (1) WO2016022703A1 (fr)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009093207A1 (fr) * 2008-01-23 2009-07-30 Jean Hilaire Saurat Composition a usage topique

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU84491A1 (fr) * 1982-11-26 1984-06-13 Oreal Composition anti-acneique contenant en tant que compose actif un derive d'isothiazolo-(5,4b) pyridine one-3
US6008254A (en) * 1997-05-09 1999-12-28 Kligman; Douglas E. Method of treating skin disorders with high-strength tretinoin
BRPI0318498B1 (pt) * 2002-07-01 2016-07-05 Maria Villani composições terapêuticas à base de porifera para o tratamento e a prevenção de doenças da pele
US20120328670A1 (en) * 2011-06-03 2012-12-27 Allergan, Inc. Targeted Delivery of Retinoid Compounds to the Sebaceous Glands
EP2664919A1 (fr) * 2012-05-15 2013-11-20 Jean Hilaire Saurat Une méthode pour identifier les ligands du récepteur AhR possédant une activité sebosuppressive thérapeutique

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009093207A1 (fr) * 2008-01-23 2009-07-30 Jean Hilaire Saurat Composition a usage topique

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
GRIMALT R ET AL: "Premature familial sebaceous hyperplasia: Successful response to oral isotretinoin in three patients", JOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY, MOSBY, INC, US, vol. 37, no. 6, 1 December 1997 (1997-12-01), pages 996 - 998, XP027420679, ISSN: 0190-9622, [retrieved on 19971201], DOI: 10.1016/S0190-9622(97)70082-3 *
See also references of WO2016022703A1 *

Also Published As

Publication number Publication date
EP3177365A1 (fr) 2017-06-14
WO2016022703A1 (fr) 2016-02-11

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Effective date: 20170301

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Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

AX Request for extension of the european patent

Extension state: BA ME

DAV Request for validation of the european patent (deleted)
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A4 Supplementary search report drawn up and despatched

Effective date: 20171207

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Ipc: A61P 17/08 20060101AFI20171201BHEP

STAA Information on the status of an ep patent application or granted ep patent

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Effective date: 20180714