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EE200100172A - Tetrahüdropüridoeetrid, nende kasutamine ja ravim - Google Patents

Tetrahüdropüridoeetrid, nende kasutamine ja ravim

Info

Publication number
EE200100172A
EE200100172A EEP200100172A EEP200100172A EE200100172A EE 200100172 A EE200100172 A EE 200100172A EE P200100172 A EEP200100172 A EE P200100172A EE P200100172 A EEP200100172 A EE P200100172A EE 200100172 A EE200100172 A EE 200100172A
Authority
EE
Estonia
Prior art keywords
tetrahydropyridoethers
medicine
naphthyridine
imidazo
methoxyethoxy
Prior art date
Application number
EEP200100172A
Other languages
English (en)
Inventor
Senn-Bilfinger J�rg
Postius Stefan
Simon Wolfgang-Alexander
Grundler Gerhard
Hanauer Guido
Huber Reinhard
Kromer Wolfgang
Sturm Ernst
Original Assignee
Byk Gulden Lomberg Chemische Fabrik Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Byk Gulden Lomberg Chemische Fabrik Gmbh filed Critical Byk Gulden Lomberg Chemische Fabrik Gmbh
Publication of EE200100172A publication Critical patent/EE200100172A/et
Publication of EE04677B1 publication Critical patent/EE04677B1/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EEP200100172A 1998-09-23 1999-09-17 Tetrahdropridoeetrid, nende kasutamine ja ravim EE04677B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19843504 1998-09-23
EP98117988 1998-09-23
PCT/EP1999/006899 WO2000017200A1 (en) 1998-09-23 1999-09-17 Tetrahydropyridoethers

Publications (2)

Publication Number Publication Date
EE200100172A true EE200100172A (et) 2002-06-17
EE04677B1 EE04677B1 (et) 2006-08-15

Family

ID=26049024

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100172A EE04677B1 (et) 1998-09-23 1999-09-17 Tetrahdropridoeetrid, nende kasutamine ja ravim

Country Status (31)

Country Link
US (4) US6436953B1 (et)
EP (1) EP1115725B1 (et)
JP (1) JP4145492B2 (et)
KR (1) KR100668400B1 (et)
CN (2) CN100506821C (et)
AT (1) ATE231862T1 (et)
AU (1) AU763463B2 (et)
BG (1) BG65195B1 (et)
BR (1) BR9914044A (et)
CA (1) CA2344251A1 (et)
CZ (1) CZ292335B6 (et)
DE (1) DE69905178T2 (et)
DK (1) DK1115725T3 (et)
EA (1) EA005377B1 (et)
EE (1) EE04677B1 (et)
ES (1) ES2191464T3 (et)
GE (1) GEP20032926B (et)
HK (1) HK1038360B (et)
HR (1) HRP20010224A2 (et)
HU (1) HUP0102990A3 (et)
ID (1) ID28896A (et)
IL (2) IL142063A0 (et)
NO (1) NO317304B1 (et)
NZ (1) NZ510610A (et)
PL (1) PL193616B1 (et)
PT (1) PT1115725E (et)
RS (1) RS50145B (et)
SI (1) SI1115725T1 (et)
SK (1) SK285165B6 (et)
TR (1) TR200100805T2 (et)
WO (1) WO2000017200A1 (et)

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* Cited by examiner, † Cited by third party
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US6436953B1 (en) * 1998-09-23 2002-08-20 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahydropyridoethers
DK1173439T3 (da) * 1999-04-17 2003-09-08 Altana Pharma Ag Halogenalkoxy-imidazonaphthyridiner
CA2721484A1 (en) * 1999-05-12 2000-11-12 President And Fellows Of Harvard College Dopamine transporter imaging agents
JP2003528879A (ja) * 2000-03-29 2003-09-30 アルタナ ファルマ アクチエンゲゼルシャフト 三環式イミダゾピリジン
NZ520837A (en) * 2000-03-29 2005-01-28 Altana Pharma Ag Prodrugs of imidazopyridine derivatives
SK5072003A3 (en) * 2000-10-25 2003-09-11 Altana Pharma Ag Polysubstituted imidazopyridines as gastric secretion inhibitors
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
BR0207762A (pt) * 2001-03-08 2004-06-01 Astrazeneca Ab Uso de um composto ou um sal farmaceuticamente aceitável do mesmo, combinação, formulação farmacêutica, kit, método para a prevenção da úlcera gástrica induzida por medicamento, e, composição farmacêutica oral
EP1414821B1 (en) 2001-08-02 2006-08-16 ALTANA Pharma AG Tricyclic epoxides
EP1417208A1 (en) * 2001-08-03 2004-05-12 ALTANA Pharma AG Amino-substituted imidazopyridines for the treatment of gastrointestinal diseases
NZ531433A (en) * 2001-08-03 2005-09-30 Altana Pharma Ag Alkyl-substituted imidazopyridines for the treatment of gastrointestinal disorders
US7314935B2 (en) 2002-02-15 2008-01-01 Altana Pharma Ag Tricyclic n-acyl compounds
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
EP1506016A2 (en) * 2002-05-07 2005-02-16 ALTANA Pharma AG New combination of reversible proton pump inhibitors and airway therapeutics for treating airway disorders
PL375567A1 (en) 2002-11-19 2005-11-28 Altana Pharma Ag 8-substituted imidazopyridines
EP1572217B1 (en) 2002-12-12 2008-08-20 Nycomed GmbH Combination medicament of r,r-formoterol and ciclesonide
RS20050449A (sr) * 2002-12-20 2007-11-15 Altana Pharma Ag., 8-trialkisiloksi-2-metil-9-fenil-7- okso-7,8,9,10- tetrahidroimidazo /1,2h//1,7/naftiridini
RS20050603A (sr) * 2003-02-17 2007-09-21 Altana Pharma Ag., NOVE KOMBINACIJE I NOVA PRIMENA FARMACEUTSKIH AKTIVNIH JEDINjENjA
KR101179012B1 (ko) 2003-03-10 2012-09-03 니코메드 게엠베하 로플루미라스트 신규한 제조 방법
TW200503783A (en) * 2003-04-11 2005-02-01 Altana Pharma Ag Oral pharmaceutical preparation for proton pump antagonists
SA04250092B1 (ar) * 2003-05-14 2008-05-04 التانا فاروا ايه جي مركب وسيط جديد لتحضير مركبات إيميدازوبيريدين imidazopyridines فعالة علاجياً
US20060241134A1 (en) * 2003-05-27 2006-10-26 Altana Pharma Ga Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
US20050059704A1 (en) * 2003-08-29 2005-03-17 Dynogen Pharmaceuticals, Inc. Compositions useful for treating gastrointestinal motility disorders
ES2452691T5 (es) 2003-09-16 2022-09-14 Covis Pharma Gmbh Uso de ciclesonida para el tratamiento de enfermedades respiratorias
EP1974730A1 (en) 2003-11-03 2008-10-01 AstraZeneca AB Imidazo[1,2-a]pyridine derivatives for use in the treatment of sleep disturbance due to silent gastro-esophageal reflux
US7326784B2 (en) 2003-12-19 2008-02-05 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano-imidazo-pyridines derivatives
AR047605A1 (es) * 2004-02-17 2006-01-25 Altana Pharma Ag Imidazopiridinas triciclicas e intermediarios en la sintesis de las mismas,sus procesos de preparacion,composiciones farmaceuticas que los contienen y usos.
DK1784404T3 (da) 2004-09-03 2012-02-13 Yuhan Corp Pyrrolo[2,3-c]pyridinderivater samt fremgangsmåder til deres fremstilling
WO2006025714A1 (en) 2004-09-03 2006-03-09 Yuhan Corporation PYRROLO[3,2-c]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF
KR100958828B1 (ko) 2004-09-03 2010-05-24 주식회사유한양행 피롤로[3,2-b]피리딘 유도체 및 그의 제조방법
EP1861074B1 (en) * 2005-03-16 2013-04-24 Takeda GmbH Taste masked dosage form containing roflumilast
EP2080513A1 (en) 2008-01-16 2009-07-22 Schraermeyer, Ulrich, Prof. Dr. rer. nat Tetrahydropyridoethers for treatment of AMD
KR101605063B1 (ko) 2009-07-09 2016-03-21 라퀄리아 파마 인코포레이티드 소화관 운동이상이 관여하는 질환의 치료용 산 펌프 길항제
WO2012027240A1 (en) * 2010-08-23 2012-03-01 Schering Corporation Fused tricyclic inhibitors of mammalian target of rapamycin
ES2635067T3 (es) * 2012-06-15 2017-10-02 Bio-Pharm Solutions Co., Ltd. Compuesto de sulfamato de fenilalquilo y composición de relajante muscular que comprende el mismo
WO2015052256A1 (en) 2013-10-08 2015-04-16 Katairo Gmbh Tetrahydropyridoethers for the treatment of stargardt's disease

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) * 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
CA1327796C (en) 1987-07-16 1994-03-15 Jorg Senn-Bilfinger Diazoles
SE9401197D0 (sv) * 1994-04-11 1994-04-11 Astra Ab Active compounds
CA2196076A1 (en) * 1994-07-28 1996-02-08 Gerhard Grundler Acyl imidazopyridines
CZ290548B6 (cs) * 1997-03-24 2002-08-14 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahydropyridinové deriváty a farmaceutický prostředek
HUP0001555A3 (en) * 1997-10-30 2001-01-29 Altana Pharma Ag Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation
US6436953B1 (en) 1998-09-23 2002-08-20 Byk Gulden Lomberg Chemische Fabrik Gmbh Tetrahydropyridoethers

Also Published As

Publication number Publication date
US7105676B2 (en) 2006-09-12
EP1115725A1 (en) 2001-07-18
NO20011243D0 (no) 2001-03-12
TR200100805T2 (tr) 2001-08-21
PL193616B1 (pl) 2007-02-28
DK1115725T3 (da) 2003-06-23
ID28896A (id) 2001-07-12
NO317304B1 (no) 2004-10-04
CN1155598C (zh) 2004-06-30
IL142063A (en) 2007-10-31
AU6192099A (en) 2000-04-10
EE04677B1 (et) 2006-08-15
CZ20011082A3 (cs) 2001-09-12
DE69905178D1 (de) 2003-03-06
NO20011243L (no) 2001-03-12
KR100668400B1 (ko) 2007-01-17
US6436953B1 (en) 2002-08-20
ATE231862T1 (de) 2003-02-15
CN1319101A (zh) 2001-10-24
DE69905178T2 (de) 2003-07-17
US6696460B2 (en) 2004-02-24
GEP20032926B (en) 2003-03-25
KR20010075223A (ko) 2001-08-09
PL346617A1 (en) 2002-02-25
CN1560055A (zh) 2005-01-05
RS50145B (sr) 2009-03-25
WO2000017200A1 (en) 2000-03-30
BG65195B1 (bg) 2007-06-29
IL142063A0 (en) 2002-03-10
JP2002526499A (ja) 2002-08-20
AU763463B2 (en) 2003-07-24
PT1115725E (pt) 2003-06-30
BR9914044A (pt) 2001-12-04
JP4145492B2 (ja) 2008-09-03
SI1115725T1 (en) 2003-06-30
SK3992001A3 (en) 2001-12-03
BG105270A (en) 2001-11-30
EA200100315A1 (ru) 2001-10-22
US7393860B1 (en) 2008-07-01
ES2191464T3 (es) 2003-09-01
CN100506821C (zh) 2009-07-01
NZ510610A (en) 2003-07-25
EP1115725B1 (en) 2003-01-29
EA005377B1 (ru) 2005-02-24
HK1038360B (en) 2003-05-16
HUP0102990A2 (hu) 2002-01-28
US20020169320A1 (en) 2002-11-14
CZ292335B6 (cs) 2003-09-17
HUP0102990A3 (en) 2002-09-30
CA2344251A1 (en) 2000-03-30
YU21401A (sh) 2004-03-12
US20040162310A1 (en) 2004-08-19
SK285165B6 (sk) 2006-07-07
HK1038360A1 (en) 2002-03-15
HRP20010224A2 (en) 2002-04-30

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Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20061231

KB4A Valid patent at the end of a year

Effective date: 20071231

KB4A Valid patent at the end of a year

Effective date: 20081231

KB4A Valid patent at the end of a year

Effective date: 20101231

MM4A Lapsed by not paying the annual fees

Effective date: 20100917