ECSP14011505A - BENZYL SULFONAMIDE DERIVATIVES USEFUL AS MOGAT-2 INHIBITORS - Google Patents
BENZYL SULFONAMIDE DERIVATIVES USEFUL AS MOGAT-2 INHIBITORSInfo
- Publication number
- ECSP14011505A ECSP14011505A ECIEPI201411505A ECPI201411505A ECSP14011505A EC SP14011505 A ECSP14011505 A EC SP14011505A EC IEPI201411505 A ECIEPI201411505 A EC IEPI201411505A EC PI201411505 A ECPI201411505 A EC PI201411505A EC SP14011505 A ECSP14011505 A EC SP14011505A
- Authority
- EC
- Ecuador
- Prior art keywords
- mogat
- inhibitors
- derivatives useful
- sulfonamide derivatives
- benzyl sulfonamide
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 1
- ABOYDMHGKWRPFD-UHFFFAOYSA-N phenylmethanesulfonamide Chemical class NS(=O)(=O)CC1=CC=CC=C1 ABOYDMHGKWRPFD-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000006575 hypertriglyceridemia Diseases 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se refiere a compuestos de Fórmula siguiente: y análogos de los mismos donde los varios grupos sustituyentes, R1, R2, R3, R4, R5 A, y X son descritos en la presente; o una sal farmacéutica del mismo; un método para tratar una condición tal como hipertrigliceridemia y un proceso para preparar los compuestos.The present invention relates to compounds of the following Formula: and analogs thereof where the various substituent groups, R1, R2, R3, R4, R5 A, and X are described herein; or a pharmaceutical salt thereof; a method for treating a condition such as hypertriglyceridemia and a process for preparing the compounds.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261592717P | 2012-01-31 | 2012-01-31 | |
| EP12382432 | 2012-11-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP14011505A true ECSP14011505A (en) | 2015-08-31 |
Family
ID=73005793
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECIEPI201411505A ECSP14011505A (en) | 2012-01-31 | 2014-07-30 | BENZYL SULFONAMIDE DERIVATIVES USEFUL AS MOGAT-2 INHIBITORS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP14011505A (en) |
-
2014
- 2014-07-30 EC ECIEPI201411505A patent/ECSP14011505A/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DOP2014000178A (en) | NEW BENCIL SULFONAMIDE DERIVATIVES USEFUL AS MOGAT-2 INHIBITORS | |
| MX375970B (en) | TRIAZOLOPYRIMIDINE COMPOUNDS AND THEIR USES. | |
| EA201401292A3 (en) | NEW THYENOPYRIMIDINE DERIVATIVES, METHOD FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| EA201692114A1 (en) | SUBSTITUTED DIHYDRO-ISOHINOLINE NON COMPOUNDS | |
| UY35818A (en) | COMPOSITIONS AND METHODS TO MODULATE X-FARNESOID RECEPTORS | |
| CO2018000589A2 (en) | Oxiesterols and pharmaceutical compositions containing them | |
| JO3807B1 (en) | New hydroxyacid derivatives, a process for their preparation and pharmaceutical compositions containing them | |
| EA201590879A1 (en) | ARYL-CONDENSED AND HETEROARYL-CONDENSED LACTAMS | |
| CO2019000932A2 (en) | New 7-substituted sulfonimidoylpurinone compounds and derivatives for the treatment and prophylaxis of viral infection. | |
| MX376271B (en) | HETEROCYCLIC COMPOUNDS AND THEIR USES. | |
| DOP2017000278A (en) | PIRIDINES REPLACED AND METHOD OF USE | |
| UY35242A (en) | 3-QUINASA PHOSFATIDYLINOSITOL INHIBITORS | |
| EA201500426A1 (en) | PYRROLOTRIAZINON DERIVATIVES AS PI3K INHIBITORS | |
| DOP2017000034A (en) | IMIDAZOPIRIDAZINE COMPOUNDS | |
| EA201790496A1 (en) | COMPOUNDS 1-ALKYL-6-OXO-1,6-DIHYDROPYRIDIN-3-ELA AND APPLICATION AS SGRM MODULATORS | |
| DOP2014000177A (en) | NEW MOROFOLINYL DERIVATIVES USEFUL AS MOGAT-2 INHIBITORS | |
| CO2017009989A2 (en) | Pyridopyrimidinones and their use as modulators of nmda receptors | |
| NI201200195A (en) | PROCEDURE FOR THE PREPARATION OF THE PERINDOPRYL L-ARGININE SALT | |
| MX2018010177A (en) | COMPOUNDS OF 6,7-DIHIDRO-5H-PIRAZOLO [5,1-B] [1,3] OXAZINA-2-CARBOXA MIDA. | |
| EA201791396A1 (en) | DERIVATIVES OF IMIDAZOPIRIDAZIN AS PI3Kβ INHIBITORS | |
| EA201590656A1 (en) | AZAINDOLINS | |
| EA201650003A1 (en) | CYCLOALCYL-DIGETERO-CYCLIC DERIVATIVES | |
| EA201791397A1 (en) | HYDROCYCLILES RELATED IMIDAZOPIRIDAZIN DERIVATIVES AS PI3Kβ INHIBITORS | |
| ECSP14011505A (en) | BENZYL SULFONAMIDE DERIVATIVES USEFUL AS MOGAT-2 INHIBITORS | |
| ECSP14011506A (en) | NEW MOROFOLINYL DERIVATIVES USEFUL AS INHIBITORS OF MOGAT-2 |