ECSP003378A - ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEM - Google Patents
ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEMInfo
- Publication number
- ECSP003378A ECSP003378A ECSP003378A ECSP003378A EC SP003378 A ECSP003378 A EC SP003378A EC SP003378 A ECSP003378 A EC SP003378A EC SP003378 A ECSP003378 A EC SP003378A
- Authority
- EC
- Ecuador
- Prior art keywords
- combinations
- methods
- pain
- compounds
- directed
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 230000003556 anti-epileptic effect Effects 0.000 title abstract 2
- 239000001961 anticonvulsive agent Substances 0.000 title abstract 2
- 230000000202 analgesic effect Effects 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 241000124008 Mammalia Species 0.000 abstract 1
- 229940099433 NMDA receptor antagonist Drugs 0.000 abstract 1
- 229940035676 analgesics Drugs 0.000 abstract 1
- 239000000730 antalgic agent Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 239000003703 n methyl dextro aspartic acid receptor blocking agent Substances 0.000 abstract 1
- 239000000041 non-steroidal anti-inflammatory agent Substances 0.000 abstract 1
- 229940021182 non-steroidal anti-inflammatory drug Drugs 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención está dirigida a combinaciones nuevas de compuestos antiepilépticos que demuestran propiedades para aliviar el dolor, con compuestos seleccionados del grupo que consiste en analgésicos antagonistas del receptor de NMDA, NSAID y combinanciones de las mismas, y composiciones farmacéuticas que las comprenden. Se ha descubierto que la administarción de compuestos antiepiléptidos que demuestran propiedades que alivian el dolor de estas combinaciones nuevas da como resultado una reducción mejorada en la fracuencia y severidad del dolor. También se cree que estas combinaciones nuevas pueden reducir la incidencia de efectso colaterales no deseados en comparación con el uso de dosis más elevadas de un tratamiento de un solo agente para lograr un efecto terapéutico similar. La presente invención también está dirigida a métodos para usar cantidades efectivas de las composiciones farmacéuticas para tratar el dolor en mamíferos.The present invention is directed to novel combinations of antiepileptic compounds demonstrating pain relieving properties, with compounds selected from the group consisting of NMDA receptor antagonist analgesics, NSAIDs and combinations thereof, and pharmaceutical compositions comprising them. Administration of antiepileptide compounds demonstrating pain relieving properties of these new combinations has been found to result in an improved reduction in pain severity and frequency. These new combinations are also believed to reduce the incidence of unwanted side effects compared to using higher doses of a single agent treatment to achieve a similar therapeutic effect. The present invention is also directed to methods of using effective amounts of pharmaceutical compositions to treat pain in mammals.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003378 ECSP003378A (en) | 2000-03-08 | 2000-03-08 | ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEM |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003378 ECSP003378A (en) | 2000-03-08 | 2000-03-08 | ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEM |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003378A true ECSP003378A (en) | 2000-05-08 |
Family
ID=42041008
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003378 ECSP003378A (en) | 2000-03-08 | 2000-03-08 | ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEM |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003378A (en) |
-
2000
- 2000-03-08 EC ECSP003378 patent/ECSP003378A/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY26052A1 (en) | ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEM | |
| CU23226B7 (en) | ANALGESTIC COMPOSITIONS THAT INCLUDE NON-STEROID ANTI-EPILEPTIC AND ANTI-INFLAMMATORY COMPOUNDS | |
| PA8515001A1 (en) | A PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF ACUTE, CHRONIC AND / OR NEUROPATHIC PAIN AND MIGRAINE PAIN | |
| CL2004000452A1 (en) | USE OF AN ANTIEPILEPTIC COMPOUND CONTAINING PAIN RELIEF PROPERTIES AND TWO OR MORE COMPOUNDS OF THE GROUP FORMED BY ANDAGONIST OF THE NMDA SELECTIVES OF SUBTIPO, ANALGESICOS, NSAID, AND COMBINATIONS OF THEM, FOR THE PREPARATION OF A MEDICINAL PRODUCT | |
| CO6241105A2 (en) | "PHARMACEUTICAL COMPOSITIONS THAT YOU INCLUDE {4- (6-FLUORO-7-METHYLAMINE-2,4-DIOXO-1,4-DIHYDRO-2H-QUINAZOLIN-3-IL) -FENIL} -5-CHLORINE-THIOFEN-2-IL -SULFONILUREA AND AN ANTICOAGULANT OR ANOTHER ANTIPLAQUETARY AGENT " | |
| ECSP066312A (en) | PIRIDILO DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS | |
| CY1116215T1 (en) | Combination therapy for the therapeutic treatment of Protein Deficiency Disorders | |
| AR044007A1 (en) | METHODS FOR THE TREATMENT OF PARKINSON'S DISEASE | |
| EA200400689A1 (en) | PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING AROMATIC ALDEHYDES CONTAINING OXYGROUP | |
| AR022252A1 (en) | ORAL ADMINISTRATION COMPOSITION. | |
| CO5670327A2 (en) | PROCEDURE FOR THE TREATMENT OF DEPRESSION AND ANXIETY DISORDERS THROUGH COMBINATION THERAPY | |
| AR074313A1 (en) | METHOD TO TREAT OR PREVENT THROMBOSIS USING DABIGATRAN ETEXYLATE OR A SALT OF THE SAME. USE. KIT | |
| BR0111207A (en) | Combinations of an endothelin receptor antagonist and an antiepileptic compound having pain relieving or analgesic properties | |
| CR6962A (en) | COMBINATION OF GABA AGONISTS AND INHIBITORS OF ALDOSA-REDUCTASA | |
| EA202191079A1 (en) | METHODS FOR TREATMENT OF RETTA SYNDROME WITH FENFLURAMINE | |
| EA200870469A1 (en) | NEW, CONTAINING NIMESULIDE, PHARMACEUTICAL COMPOSITIONS WITH LOW DOSE, THEIR RECEPTION AND APPLICATION | |
| IS6558A (en) | Mixed disease treatment with vasoconstrictor | |
| DE602004020494D1 (en) | ANALGETIC COMPOUNDS, THE SYNTHESIS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
| ECSP003378A (en) | ANALGESIC COMPOSITIONS INCLUDING ANTI-EPILEPTIC COMPOUNDS AND METHODS FOR USING THEM | |
| AR045423A1 (en) | COMBINATIONS OF ANALYTICS AND ANTIDEPRESSANTS | |
| Liu et al. | Comparative study between three analgesic agents for the pain management during extracorporeal shock wave lithotripsy | |
| AR052830A1 (en) | CLADRIBINE REGIME TO TREAT MULTIPLE SCLEROSIS | |
| CL2004000767A1 (en) | ORAL DOSING UNIT INCLUDING AN ANTAGONIST AGENT FOR PUMPS OF PROTONS AND EXCIPIENTS OF BASIC CHARACTER; PROCEDURE FOR PREPARATION, USEFUL TO TREAT DISEASES CAUSED BY AN INCREASED SECRETION OF GASTRIC ACIDS. | |
| EA200300430A1 (en) | NEW PHARMACEUTICAL COMPOSITIONS CONTAINING EPINASTINES AND PSEVDOEDFEDRIN | |
| FR2809725B1 (en) | PROPANOLAMINOTETRALINS, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME |