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EA201200019A1 - Соединения, которые селективно модулируют рецептор св2 - Google Patents

Соединения, которые селективно модулируют рецептор св2

Info

Publication number
EA201200019A1
EA201200019A1 EA201200019A EA201200019A EA201200019A1 EA 201200019 A1 EA201200019 A1 EA 201200019A1 EA 201200019 A EA201200019 A EA 201200019A EA 201200019 A EA201200019 A EA 201200019A EA 201200019 A1 EA201200019 A1 EA 201200019A1
Authority
EA
Eurasian Patent Office
Prior art keywords
compounds
receptor
selectively modulate
agonists
useful
Prior art date
Application number
EA201200019A
Other languages
English (en)
Inventor
Алессандра Бартолоцци
Юджин Ричард Хики
Дорис Ритер
Лифэнь Ву
Рене Зинделл
Найджел Блумайр
Моника Эрманн
Эдуард Томас Гленн
Сомейна Кхор
Пшемислав Завадзкий
Original Assignee
Бёрингер Ингельхайм Интернациональ Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42646483&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201200019(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бёрингер Ингельхайм Интернациональ Гмбх filed Critical Бёрингер Ингельхайм Интернациональ Гмбх
Publication of EA201200019A1 publication Critical patent/EA201200019A1/ru

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Immunology (AREA)
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  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
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  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
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  • Transplantation (AREA)
  • Hematology (AREA)
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  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

В заявке описаны соединения формулы (I)Соединения, предлагаемые в настоящем изобретении, связываются с рецептором СВ2, являются агонистами, антагонистами или обратными агонистами рецептора СВ2 и применимы для лечения воспаления. Те соединения, которые являются агонистами, также дополнительно применимы для лечения боли.
EA201200019A 2009-06-15 2010-06-08 Соединения, которые селективно модулируют рецептор св2 EA201200019A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18692009P 2009-06-15 2009-06-15
PCT/US2010/037697 WO2010147792A2 (en) 2009-06-15 2010-06-08 Compounds which selectively modulate the cb2 receptor

Publications (1)

Publication Number Publication Date
EA201200019A1 true EA201200019A1 (ru) 2012-06-29

Family

ID=42646483

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201200019A EA201200019A1 (ru) 2009-06-15 2010-06-08 Соединения, которые селективно модулируют рецептор св2

Country Status (23)

Country Link
US (2) US8299103B2 (ru)
EP (2) EP2443100A2 (ru)
JP (1) JP5492297B2 (ru)
KR (1) KR20120047211A (ru)
CN (1) CN102803235A (ru)
AP (1) AP2011005988A0 (ru)
AR (1) AR077362A1 (ru)
AU (1) AU2010260397A1 (ru)
BR (1) BRPI1011668A2 (ru)
CA (1) CA2765525A1 (ru)
CL (1) CL2011003160A1 (ru)
CO (1) CO6470896A2 (ru)
EA (1) EA201200019A1 (ru)
EC (1) ECSP12011583A (ru)
IL (1) IL216348A0 (ru)
MA (1) MA33362B1 (ru)
MX (1) MX2011013152A (ru)
PE (1) PE20120561A1 (ru)
SG (1) SG176864A1 (ru)
TN (1) TN2011000639A1 (ru)
TW (1) TW201111374A (ru)
WO (1) WO2010147792A2 (ru)
ZA (1) ZA201108258B (ru)

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EP2265585B1 (en) * 2008-02-21 2014-09-17 Boehringer Ingelheim International GmbH Amine and ether compounds which modulate the cb2 receptor
WO2010005782A1 (en) * 2008-07-10 2010-01-14 Boehringer Ingelheim International Gmbh Sulfone compounds which modulate the cb2 receptor
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US8629157B2 (en) 2009-01-05 2014-01-14 Boehringer Ingelheim International Gmbh Pyrrolidine compounds which modulate the CB2 receptor
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US8299103B2 (en) 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
US8383615B2 (en) 2009-06-16 2013-02-26 Boehringer Ingelheim International Gmbh Azetidine 2-carboxamide derivatives which modulate the CB2 receptor
US8383651B2 (en) * 2009-09-22 2013-02-26 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
CA2784710A1 (en) * 2009-12-15 2011-06-23 Shionogi & Co., Ltd. Oxadiazole derivative having endothelial lipase inhibitory activity
EP2523936A1 (en) 2010-01-15 2012-11-21 Boehringer Ingelheim International GmbH Compounds which modulate the cb2 receptor
US8329735B2 (en) 2010-03-05 2012-12-11 Boehringer Ingelheim International Gmbh Tetrazole compounds which selectively modulate the CB2 receptor
EP2595959B1 (en) 2010-07-22 2015-11-04 Boehringer Ingelheim International GmbH Sulfonyl compounds which modulate the cb2 receptor
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