EA200701409A1 - Новая композиция - Google Patents
Новая композицияInfo
- Publication number
- EA200701409A1 EA200701409A1 EA200701409A EA200701409A EA200701409A1 EA 200701409 A1 EA200701409 A1 EA 200701409A1 EA 200701409 A EA200701409 A EA 200701409A EA 200701409 A EA200701409 A EA 200701409A EA 200701409 A1 EA200701409 A1 EA 200701409A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- drug
- composition
- pharmaceutically acceptable
- dosage form
- new composition
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 5
- 239000003814 drug Substances 0.000 abstract 5
- 229940079593 drug Drugs 0.000 abstract 4
- 239000002552 dosage form Substances 0.000 abstract 2
- 229940126062 Compound A Drugs 0.000 abstract 1
- NLDMNSXOCDLTTB-UHFFFAOYSA-N Heterophylliin A Natural products O1C2COC(=O)C3=CC(O)=C(O)C(O)=C3C3=C(O)C(O)=C(O)C=C3C(=O)OC2C(OC(=O)C=2C=C(O)C(O)=C(O)C=2)C(O)C1OC(=O)C1=CC(O)=C(O)C(O)=C1 NLDMNSXOCDLTTB-UHFFFAOYSA-N 0.000 abstract 1
- 239000003937 drug carrier Substances 0.000 abstract 1
- 239000006186 oral dosage form Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
- A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Пероральная лекарственная форма, включающая первую композицию и вторую композицию, причем каждая композиция включает фармацевтически приемлемое слабое основание, особенно соединение А или его фармацевтически приемлемую соль или сольват («лекарственное средство»), и фармацевтически приемлемый носитель для него, где первая и вторая композиции организованы для высвобождения лекарственного средства с различающимися скоростями высвобождения при введении таким образом, что скорость высвобождения лекарственного средства из лекарственной формы является, по существу, независимой от рН; способ получения такой лекарственной формы и применение такой лекарственной формы в медицине.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49338803P | 2003-08-07 | 2003-08-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EA200701409A1 true EA200701409A1 (ru) | 2007-10-26 |
Family
ID=34135242
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200600377A EA011508B1 (ru) | 2003-08-07 | 2004-08-06 | Пероральная лекарственная форма (варианты) и способ ее получения |
| EA200701409A EA200701409A1 (ru) | 2003-08-07 | 2004-08-06 | Новая композиция |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200600377A EA011508B1 (ru) | 2003-08-07 | 2004-08-06 | Пероральная лекарственная форма (варианты) и способ ее получения |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US20070134326A1 (ru) |
| EP (1) | EP1660049A2 (ru) |
| JP (1) | JP2007501773A (ru) |
| KR (1) | KR20060113650A (ru) |
| CN (2) | CN101239047A (ru) |
| AP (1) | AP2006003488A0 (ru) |
| AR (1) | AR045330A1 (ru) |
| AU (1) | AU2004262926B2 (ru) |
| BR (1) | BRPI0413374A (ru) |
| CA (1) | CA2534546A1 (ru) |
| EA (2) | EA011508B1 (ru) |
| EC (1) | ECSP066318A (ru) |
| IL (1) | IL173176A0 (ru) |
| IS (1) | IS8336A (ru) |
| MA (1) | MA27980A1 (ru) |
| MX (1) | MXPA06001407A (ru) |
| NO (1) | NO20061018L (ru) |
| NZ (1) | NZ544696A (ru) |
| OA (1) | OA13230A (ru) |
| PE (1) | PE20050335A1 (ru) |
| SG (1) | SG145717A1 (ru) |
| TW (1) | TW200517127A (ru) |
| UY (1) | UY28457A1 (ru) |
| WO (1) | WO2005013935A2 (ru) |
| ZA (1) | ZA200600521B (ru) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0203296D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel composition |
| US8637512B2 (en) * | 2002-07-29 | 2014-01-28 | Glaxo Group Limited | Formulations and method of treatment |
| EP1686967A4 (en) * | 2003-11-25 | 2012-08-08 | Smithkline Beecham Cork Ltd | CARVEDILOL-FREE BASE, SALTS, WATER-FREE FORMS OR SOLVATES THEREOF, CORRESPONDING PHARMACEUTICAL COMPOSITIONS, CONTROLLED RELEASE FORMULAS AND TREATMENT OR DISPOSAL PROCEDURES |
| GB0502479D0 (en) * | 2005-02-07 | 2005-03-16 | Sb Pharmco Inc | Novel compositions |
| GB0502475D0 (en) * | 2005-02-07 | 2005-03-16 | Sb Pharmco Inc | Novel compositions |
| US20100323016A1 (en) * | 2008-07-18 | 2010-12-23 | Biljana Nadjsombati | Modified release formulation and methods of use |
| US20100323015A1 (en) * | 2008-07-18 | 2010-12-23 | Biljana Nadjsombati | Modified release formulation and methods of use |
| LT2395840T (lt) | 2009-02-13 | 2020-07-10 | Romark Laboratories, L.C. | Nitazoksanido kontroliuojamo atpalaidavimo farmacinės kompozicijos |
| SG181827A1 (en) | 2010-01-20 | 2012-07-30 | Glaxo Group Ltd | Novel retigabine composition |
| CN103948557A (zh) * | 2014-04-08 | 2014-07-30 | 闻晓光 | 一种新型控释片 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8820353D0 (en) * | 1988-08-26 | 1988-09-28 | Staniforth J N | Controlled release tablet |
| FR2655266B1 (fr) * | 1989-12-05 | 1992-04-03 | Smith Kline French Lab | Compositions pharmaceutiques a base de cimetidine. |
| IT1264517B1 (it) * | 1993-05-31 | 1996-09-24 | Ekita Investments Nv | Compressa farmaceutica atta al rilascio in tempi successivi dei principi attivi in essa veicolati |
| HU213407B (en) * | 1993-12-09 | 1997-06-30 | Egyt Gyogyszervegyeszeti Gyar | Process for producing tablet with diffusive-osmotic release |
| US5407687A (en) * | 1994-02-22 | 1995-04-18 | Glaxo Inc. | Ranitidine solid dosage form |
| US5952509A (en) * | 1996-06-27 | 1999-09-14 | Takeda Chemical Industries, Ltd. | Production of benzaldehyde compounds |
| GB9619757D0 (en) * | 1996-09-21 | 1996-11-06 | Knoll Ag | Chemical process |
| US20010049380A1 (en) * | 1997-06-18 | 2001-12-06 | Smith Stephen Alistair | Treatment of diabetes with thiazolidinedione and sulphonylurea |
| US20020004515A1 (en) * | 1997-06-18 | 2002-01-10 | Smith Stephen Alistair | Treatment of diabetes with thiazolidinedione and metformin |
| US20020006939A1 (en) * | 1997-10-13 | 2002-01-17 | Smithkline Beecham P.L.C. | Use of thiazolidinediones for the treatment of hyperglycaemia |
| US6099859A (en) * | 1998-03-20 | 2000-08-08 | Andrx Pharmaceuticals, Inc. | Controlled release oral tablet having a unitary core |
| US20030153607A1 (en) * | 1998-11-12 | 2003-08-14 | Smithkline Beecham P.L.C. | Novel composition and use |
| US20040102486A1 (en) * | 1998-11-12 | 2004-05-27 | Smithkline Beecham Corporation | Novel method of treatment |
| IL143002A0 (en) * | 1998-11-12 | 2002-04-21 | Smithkline Beecham Plc | Pharmaceutical composition for modified release of an insulin sensitiser and another antidiabetic agent |
| US20040081697A1 (en) * | 1998-11-12 | 2004-04-29 | Smithkline Beecham P.L.C. | Pharmaceutical composition for modified release of an insulin sensitiser and another antidiabetic agent |
| EP1278513B1 (en) * | 2000-05-01 | 2007-07-18 | Aeropharm Technology, LLC | A core formulation |
| GB0117618D0 (en) * | 2001-07-19 | 2001-09-12 | Phoqus Ltd | Pharmaceutical dosage form |
| GB0127805D0 (en) * | 2001-11-20 | 2002-01-09 | Smithkline Beecham Plc | Pharmaceutical composition |
| GB0203296D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel composition |
| PE20030800A1 (es) * | 2002-02-12 | 2003-10-31 | Glaxo Group Ltd | Forma de dosificacion oral de liberacion controlada |
-
2004
- 2004-08-05 UY UY28457A patent/UY28457A1/es not_active Application Discontinuation
- 2004-08-05 TW TW093123415A patent/TW200517127A/zh unknown
- 2004-08-05 PE PE2004000757A patent/PE20050335A1/es not_active Application Discontinuation
- 2004-08-05 AR ARP040102794A patent/AR045330A1/es not_active Application Discontinuation
- 2004-08-06 EP EP04763874A patent/EP1660049A2/en not_active Withdrawn
- 2004-08-06 SG SG200805824-0A patent/SG145717A1/en unknown
- 2004-08-06 AU AU2004262926A patent/AU2004262926B2/en not_active Ceased
- 2004-08-06 CN CNA2008100088784A patent/CN101239047A/zh active Pending
- 2004-08-06 WO PCT/EP2004/008843 patent/WO2005013935A2/en not_active Ceased
- 2004-08-06 US US10/567,146 patent/US20070134326A1/en not_active Abandoned
- 2004-08-06 KR KR1020067002663A patent/KR20060113650A/ko not_active Ceased
- 2004-08-06 EA EA200600377A patent/EA011508B1/ru not_active IP Right Cessation
- 2004-08-06 NZ NZ544696A patent/NZ544696A/en unknown
- 2004-08-06 CA CA002534546A patent/CA2534546A1/en not_active Abandoned
- 2004-08-06 OA OA1200600040A patent/OA13230A/en unknown
- 2004-08-06 AP AP2006003488A patent/AP2006003488A0/xx unknown
- 2004-08-06 EA EA200701409A patent/EA200701409A1/ru unknown
- 2004-08-06 BR BRPI0413374-9A patent/BRPI0413374A/pt not_active Application Discontinuation
- 2004-08-06 JP JP2006522328A patent/JP2007501773A/ja not_active Withdrawn
- 2004-08-06 CN CNA2004800226534A patent/CN1832729A/zh active Pending
- 2004-08-06 MX MXPA06001407A patent/MXPA06001407A/es unknown
-
2006
- 2006-01-16 IL IL173176A patent/IL173176A0/en unknown
- 2006-01-18 ZA ZA200600521A patent/ZA200600521B/en unknown
- 2006-01-25 EC EC2006006318A patent/ECSP066318A/es unknown
- 2006-02-07 MA MA28777A patent/MA27980A1/fr unknown
- 2006-03-01 NO NO20061018A patent/NO20061018L/no not_active Application Discontinuation
- 2006-03-02 IS IS8336A patent/IS8336A/is unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005013935A3 (en) | 2005-07-14 |
| ZA200600521B (en) | 2007-01-31 |
| PE20050335A1 (es) | 2005-06-01 |
| CN101239047A (zh) | 2008-08-13 |
| BRPI0413374A (pt) | 2006-10-17 |
| AU2004262926B2 (en) | 2009-11-19 |
| JP2007501773A (ja) | 2007-02-01 |
| EA011508B1 (ru) | 2009-04-28 |
| CN1832729A (zh) | 2006-09-13 |
| SG145717A1 (en) | 2008-09-29 |
| OA13230A (en) | 2006-12-13 |
| ECSP066318A (es) | 2006-07-28 |
| MA27980A1 (fr) | 2006-07-03 |
| US20070134326A1 (en) | 2007-06-14 |
| CA2534546A1 (en) | 2005-02-17 |
| AU2004262926A1 (en) | 2005-02-17 |
| NO20061018L (no) | 2006-03-01 |
| MXPA06001407A (es) | 2006-05-15 |
| UY28457A1 (es) | 2005-03-31 |
| AP2006003488A0 (en) | 2006-02-28 |
| EA200600377A1 (ru) | 2006-08-25 |
| IS8336A (is) | 2006-03-02 |
| AR045330A1 (es) | 2005-10-26 |
| WO2005013935A2 (en) | 2005-02-17 |
| IL173176A0 (en) | 2006-06-11 |
| KR20060113650A (ko) | 2006-11-02 |
| TW200517127A (en) | 2005-06-01 |
| EP1660049A2 (en) | 2006-05-31 |
| NZ544696A (en) | 2009-03-31 |
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