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EA200700600A1 - Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агент - Google Patents

Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агент

Info

Publication number
EA200700600A1
EA200700600A1 EA200700600A EA200700600A EA200700600A1 EA 200700600 A1 EA200700600 A1 EA 200700600A1 EA 200700600 A EA200700600 A EA 200700600A EA 200700600 A EA200700600 A EA 200700600A EA 200700600 A1 EA200700600 A1 EA 200700600A1
Authority
EA
Eurasian Patent Office
Prior art keywords
agent
pharmaceutical composition
betumepholic
composition containing
cholinergic
Prior art date
Application number
EA200700600A
Other languages
English (en)
Inventor
Амар Лулла
Джина Малхотра
Original Assignee
Сипла Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Сипла Лимитед filed Critical Сипла Лимитед
Publication of EA200700600A1 publication Critical patent/EA200700600A1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/468-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Фармацевтическая композиция в дозированной форме, приемлемой для ингаляции, содержащая терапевтически эффективный изомер бета-миметического агента или его соль, сольват, эфир, производное или полиморф, по существу, свободный от менее терапевтически эффективного(ых) изомера(ов) указанного агента и необязательно антихолинергический агент или его соль, сольват, эфир, производное, изомер или полиморф. Предпочтительно композиция содержит сульфат R-сальбутамола и бромид ипратропия. Также представлены способы получения композиций по изобретению.
EA200700600A 2004-09-09 2005-09-09 Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агент EA200700600A1 (ru)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
IN970MU2004 2004-09-09
IN1004MU2004 2004-09-17
IN1077MU2004 2004-10-08
IN1088MU2004 2004-10-11
IN1089MU2004 2004-10-11
IN93MU2005 2005-01-31
IN222MU2005 2005-02-28
PCT/GB2005/003475 WO2006027595A1 (en) 2004-09-09 2005-09-09 Pharmaceutical composition comprising an isomer of a betamimetic agent and an anti-cholinergic agent

Publications (1)

Publication Number Publication Date
EA200700600A1 true EA200700600A1 (ru) 2008-02-28

Family

ID=35311711

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200700600A EA200700600A1 (ru) 2004-09-09 2005-09-09 Фармацевтическая композиция, содержащая изомер бета-миметического агента и антихолинергический агент

Country Status (11)

Country Link
US (1) US20070264202A1 (ru)
EP (1) EP1791534A1 (ru)
JP (1) JP2008512434A (ru)
KR (1) KR20070102659A (ru)
AU (1) AU2005281511B2 (ru)
BR (1) BRPI0515103A (ru)
CA (1) CA2580019A1 (ru)
EA (1) EA200700600A1 (ru)
IL (1) IL181828A0 (ru)
MX (1) MX2007002899A (ru)
WO (1) WO2006027595A1 (ru)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0501956D0 (en) * 2005-01-31 2005-03-09 Arrow Internat Nebulizer formulation
CA2652699C (en) 2006-05-19 2014-11-04 Boehringer Ingelheim International Gmbh Propellant-free inhalation aerosol formulation containing ipratropium bromide and salbutamol sulfate
US20100144784A1 (en) * 2006-05-19 2010-06-10 Boehringer Ingelheim International Gmbh Aerosol formulation
US20070286814A1 (en) * 2006-06-12 2007-12-13 Medispray Laboratories Pvt. Ltd. Stable aerosol pharmaceutical formulations
EP2077132A1 (en) 2008-01-02 2009-07-08 Boehringer Ingelheim Pharma GmbH & Co. KG Dispensing device, storage device and method for dispensing a formulation
CA2741078A1 (en) * 2008-10-23 2010-04-29 Sunovion Pharmaceuticals Inc. Arformoterol and tiotropium compositions and methods for use
US10011906B2 (en) 2009-03-31 2018-07-03 Beohringer Ingelheim International Gmbh Method for coating a surface of a component
JP5763053B2 (ja) 2009-05-18 2015-08-12 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング アダプタ、吸入器具及びアトマイザ
EP2504051B1 (en) 2009-11-25 2019-09-04 Boehringer Ingelheim International GmbH Nebulizer
US10016568B2 (en) 2009-11-25 2018-07-10 Boehringer Ingelheim International Gmbh Nebulizer
AP3141A (en) 2009-11-25 2015-02-28 Boehringer Ingelheim Int Nebulizer
JP5874724B2 (ja) 2010-06-24 2016-03-02 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ネブライザ
WO2012130757A1 (de) 2011-04-01 2012-10-04 Boehringer Ingelheim International Gmbh Medizinisches gerät mit behälter
US9827384B2 (en) 2011-05-23 2017-11-28 Boehringer Ingelheim International Gmbh Nebulizer
WO2013152894A1 (de) 2012-04-13 2013-10-17 Boehringer Ingelheim International Gmbh Zerstäuber mit kodiermitteln
ES2836977T3 (es) 2013-08-09 2021-06-28 Boehringer Ingelheim Int Nebulizador
US9744313B2 (en) 2013-08-09 2017-08-29 Boehringer Ingelheim International Gmbh Nebulizer
CN106255554B (zh) 2014-05-07 2021-05-04 勃林格殷格翰国际有限公司 容器、喷雾器及用途
PE20210959A1 (es) 2014-05-07 2021-05-25 Boehringer Ingelheim Int Nebulizador, dispositivo indicador y recipiente
ES2874029T3 (es) 2014-05-07 2021-11-04 Boehringer Ingelheim Int Nebulizador
EP3569221A1 (en) * 2018-05-17 2019-11-20 Notoxins IP B.V. Aqueous formulations comprising ipratropium for topical treatment of hyperhidrosis
CN113018280A (zh) * 2021-03-01 2021-06-25 石家庄四药有限公司 一种异丙托溴铵吸入用溶液制剂及其制备方法

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5192528A (en) * 1985-05-22 1993-03-09 Liposome Technology, Inc. Corticosteroid inhalation treatment method
US5919827A (en) * 1990-07-11 1999-07-06 Sepracor Inc. Method for treating asthma using optically pure R(-) salmeterol
US6299863B1 (en) * 1992-04-03 2001-10-09 Sepracor Inc. Aerosol formulations containing micronized optically pure (R,R) formoterol for bronchodilating therapy
US5795564A (en) * 1991-04-05 1998-08-18 Sepracor, Inc. Methods and compositions for treating pulmonary disorders using optically pure (R,R)-formoterol
US6423298B2 (en) * 1998-06-18 2002-07-23 Boehringer Ingelheim Pharmaceuticals, Inc. Pharmaceutical formulations for aerosols with two or more active substances
GB9827200D0 (en) * 1998-12-11 1999-02-03 Glaxo Group Ltd Dry powder inhaler
AU4831801A (en) * 2000-03-01 2001-09-12 Glaxo Group Limited Metered dose inhaler
US20040019025A1 (en) * 2000-04-18 2004-01-29 Gavin Brian Charles Medical compositions comprising (r,r)-formoterol and rofleponide
GB0009607D0 (en) * 2000-04-18 2000-06-07 Glaxo Group Ltd Medical compositions
AU2001278115A1 (en) * 2000-08-04 2002-02-18 Longwood Pharmaceutical Research, Inc. Formulations of mometasone and a bronchodilator for pulmonary administration
JP2004512101A (ja) * 2000-10-20 2004-04-22 グラクソ グループ リミテッド 吸入器
GB0030171D0 (en) * 2000-12-11 2001-01-24 Cipla Ltd Process for preparing isomers of salbutamol
US20020189610A1 (en) * 2001-02-01 2002-12-19 Karl-Heinz Bozung Pharmaceutical compositions containing an ipratropium salt and a betamimetic
GB0105560D0 (en) * 2001-03-07 2001-04-25 Glaxo Group Ltd Pharmaceutical formulations
US6667344B2 (en) * 2001-04-17 2003-12-23 Dey, L.P. Bronchodilating compositions and methods
JP2003221335A (ja) * 2001-10-26 2003-08-05 Dey Lp 慢性閉塞性肺疾患の症状を緩和するためのアルブテロールおよびイプラトロピウム吸入溶液、システム、キットおよび方法
DK1572622T3 (da) * 2002-12-10 2006-08-28 Sepracor Inc Anvendelse af levalbuterol-L-tartrat ved fremstilling af en doseringsinhalator
US20040191176A1 (en) * 2003-03-28 2004-09-30 Kaplan Leonard W Formulations for treatment of pulmonary disorders

Also Published As

Publication number Publication date
CA2580019A1 (en) 2006-03-16
AU2005281511A1 (en) 2006-03-16
US20070264202A1 (en) 2007-11-15
WO2006027595A1 (en) 2006-03-16
IL181828A0 (en) 2007-07-04
EP1791534A1 (en) 2007-06-06
BRPI0515103A (pt) 2008-07-08
KR20070102659A (ko) 2007-10-19
AU2005281511B2 (en) 2011-03-31
JP2008512434A (ja) 2008-04-24
MX2007002899A (es) 2007-05-16

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