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EA200600925A1 - DERIVATIVES OF TRIAZOLE AS ANTAGONISTS VAZOPRESSIN - Google Patents

DERIVATIVES OF TRIAZOLE AS ANTAGONISTS VAZOPRESSIN

Info

Publication number
EA200600925A1
EA200600925A1 EA200600925A EA200600925A EA200600925A1 EA 200600925 A1 EA200600925 A1 EA 200600925A1 EA 200600925 A EA200600925 A EA 200600925A EA 200600925 A EA200600925 A EA 200600925A EA 200600925 A1 EA200600925 A1 EA 200600925A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
vazopressin
triazole
antagonists
ring
Prior art date
Application number
EA200600925A
Other languages
Russian (ru)
Other versions
EA010132B1 (en
Inventor
Джастин Стивен Брайанс
Патрик Стивен Джонсон
Ли Ричард Робертс
Томас Рикманс
Original Assignee
Пфайзер Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0329693A external-priority patent/GB0329693D0/en
Priority claimed from GB0408789A external-priority patent/GB0408789D0/en
Application filed by Пфайзер Инк. filed Critical Пфайзер Инк.
Publication of EA200600925A1 publication Critical patent/EA200600925A1/en
Publication of EA010132B1 publication Critical patent/EA010132B1/en

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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  • Health & Medical Sciences (AREA)
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Abstract

Соединения формулы (I) или их фармацевтически приемлемые производные, где: V представляет собой прямую связь или -О-; кольцо А представляет собой возможно замещенное 5-7-членное насыщенное гетероциклическое кольцо или фениленовую группу.Compounds of formula (I) or pharmaceutically acceptable derivatives thereof, wherein: V is a direct bond or —O—; ring A is a possibly substituted 5-7 membered saturated heterocyclic ring or phenylene group.

EA200600925A 2003-12-22 2004-12-09 Triazole derivatives as vasopressin antagonists EA010132B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0329693A GB0329693D0 (en) 2003-12-22 2003-12-22 Compounds useful in therapy
GB0408789A GB0408789D0 (en) 2004-04-20 2004-04-20 Triazole derivatives
PCT/IB2004/004059 WO2005063754A1 (en) 2003-12-22 2004-12-09 Triazole derivatives as vasopressin antagonists

Publications (2)

Publication Number Publication Date
EA200600925A1 true EA200600925A1 (en) 2006-12-29
EA010132B1 EA010132B1 (en) 2008-06-30

Family

ID=34740750

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200600925A EA010132B1 (en) 2003-12-22 2004-12-09 Triazole derivatives as vasopressin antagonists

Country Status (24)

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EP (1) EP1701959A1 (en)
JP (1) JP4698604B2 (en)
KR (1) KR100854872B1 (en)
AP (1) AP2331A (en)
AR (1) AR047340A1 (en)
AU (1) AU2004309164B2 (en)
BR (1) BRPI0417267A (en)
CA (1) CA2551038C (en)
CR (1) CR8481A (en)
DO (1) DOP2004001062A (en)
EA (1) EA010132B1 (en)
EC (1) ECSP066647A (en)
GE (1) GEP20084571B (en)
IL (1) IL176349A (en)
IS (1) IS8472A (en)
MA (1) MA28393B1 (en)
NL (1) NL1027833C2 (en)
NO (1) NO20063380L (en)
OA (1) OA13347A (en)
PA (1) PA8620501A1 (en)
PE (1) PE20051051A1 (en)
TW (1) TWI287541B (en)
UY (1) UY28693A1 (en)
WO (1) WO2005063754A1 (en)

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