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DK475388D0 - BENZAZEPINE DERIVATIVES AND THEIR USE AS CARDIOVASCULAR AGENTS - Google Patents

BENZAZEPINE DERIVATIVES AND THEIR USE AS CARDIOVASCULAR AGENTS

Info

Publication number
DK475388D0
DK475388D0 DK475388A DK475388A DK475388D0 DK 475388 D0 DK475388 D0 DK 475388D0 DK 475388 A DK475388 A DK 475388A DK 475388 A DK475388 A DK 475388A DK 475388 D0 DK475388 D0 DK 475388D0
Authority
DK
Denmark
Prior art keywords
cardiovascular agents
benzazepine derivatives
benzazepine
derivatives
cardiovascular
Prior art date
Application number
DK475388A
Other languages
Danish (da)
Other versions
DK163121C (en
DK163121B (en
DK475388A (en
Inventor
Jagabandhu Das
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of DK475388D0 publication Critical patent/DK475388D0/en
Publication of DK475388A publication Critical patent/DK475388A/en
Publication of DK163121B publication Critical patent/DK163121B/en
Application granted granted Critical
Publication of DK163121C publication Critical patent/DK163121C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16Benzazepines; Hydrogenated benzazepines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK475388A 1987-08-26 1988-08-25 1-BENZAZEPIN-2-ON DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING SUCH PRODUCTS AND USING THEM FOR THE PREPARATION OF THE PREPARATIONS DK163121C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/089,479 US4774239A (en) 1987-08-26 1987-08-26 Benzazepine derivatives
US8947987 1987-08-26

Publications (4)

Publication Number Publication Date
DK475388D0 true DK475388D0 (en) 1988-08-25
DK475388A DK475388A (en) 1989-02-27
DK163121B DK163121B (en) 1992-01-20
DK163121C DK163121C (en) 1992-06-15

Family

ID=22217878

Family Applications (1)

Application Number Title Priority Date Filing Date
DK475388A DK163121C (en) 1987-08-26 1988-08-25 1-BENZAZEPIN-2-ON DERIVATIVES, PHARMACEUTICAL PREPARATIONS CONTAINING SUCH PRODUCTS AND USING THEM FOR THE PREPARATION OF THE PREPARATIONS

Country Status (8)

Country Link
US (1) US4774239A (en)
EP (1) EP0304918A1 (en)
JP (1) JPS6471859A (en)
AU (1) AU609169B2 (en)
DK (1) DK163121C (en)
HU (1) HU201308B (en)
NZ (1) NZ225613A (en)
ZA (1) ZA885606B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4952692A (en) * 1989-04-04 1990-08-28 E. R. Squibb & Sons, Inc. Benzazepine derivatives
US4946840A (en) * 1989-04-06 1990-08-07 E. R. Squibb & Sons, Inc. Benzazepine and benzothiazepine derivatives
US5559017A (en) * 1989-08-09 1996-09-24 E. R. Squibb & Sons, Inc. Microbial reduction of benzazepines and benzothiazepine derivatives
JP4202250B2 (en) 2001-07-25 2008-12-24 バイオマリン ファーマシューティカル インコーポレイテッド Compositions and methods for modulating blood brain barrier transport
CA2789262C (en) 2005-04-28 2016-10-04 Proteus Digital Health, Inc. Pharma-informatics system
US8795627B2 (en) 2007-03-21 2014-08-05 Raptor Pharmaceuticals Inc. Treatment of liver disorders by administration of RAP conjugates
ES2919563T3 (en) 2009-02-20 2022-07-27 Enhanx Biopharm Inc Glutathione-based drug delivery system
CN110075069A (en) 2009-05-06 2019-08-02 实验室护肤股份有限公司 Include activating agent-calcium phosphate granules compound dermal delivery composition and its application
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
JP2022055368A (en) * 2019-02-19 2022-04-08 株式会社三和化学研究所 Method for producing benzoazepine derivative and intermediate thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3312691A (en) * 1963-08-23 1967-04-04 Ciba Geigy Corp 2, 3, 4, 5-tetrahydro-1-benzazepin-2-ones
US3330823A (en) * 1964-12-16 1967-07-11 Squibb & Sons Inc N-amino-loweralkylene-benzo-lactams
US3395150A (en) * 1965-02-26 1968-07-30 Squibb & Sons Inc Benzothiazepine carboxamides and derivatives thereof
US3562257A (en) * 1967-10-28 1971-02-09 Tanabe Seiyaku Co Benzothiazepine derivatives
DE2850078A1 (en) * 1978-11-18 1980-05-29 Basf Ag AMINOPROPANOL DERIVATIVES OF 6-HYDROXY-2,3,4,5-TETRAHYDRO-1H-1-BENZAZEPIN-2-ONS
US4748239A (en) * 1985-06-12 1988-05-31 E. R. Squibb & Sons, Inc. Benzazepine derivatives
CA1271747C (en) * 1985-06-12 1990-07-17 Benzazepines derivatives
CA1271748A (en) * 1985-12-12 1990-07-17 Jagabandhu Das Benzazepine derivatives

Also Published As

Publication number Publication date
JPS6471859A (en) 1989-03-16
HU201308B (en) 1990-10-28
DK163121C (en) 1992-06-15
DK163121B (en) 1992-01-20
US4774239A (en) 1988-09-27
AU2058288A (en) 1989-03-02
NZ225613A (en) 1990-09-26
AU609169B2 (en) 1991-04-26
ZA885606B (en) 1989-04-26
HUT48601A (en) 1989-06-28
DK475388A (en) 1989-02-27
EP0304918A1 (en) 1989-03-01

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Legal Events

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