DK3810587T3 - Substituerede alkoxypyridinylindolsulfonamider - Google Patents
Substituerede alkoxypyridinylindolsulfonamider Download PDFInfo
- Publication number
- DK3810587T3 DK3810587T3 DK19731283.8T DK19731283T DK3810587T3 DK 3810587 T3 DK3810587 T3 DK 3810587T3 DK 19731283 T DK19731283 T DK 19731283T DK 3810587 T3 DK3810587 T3 DK 3810587T3
- Authority
- DK
- Denmark
- Prior art keywords
- alkoxypyridinylindolesulfonamides
- substituted
- substituted alkoxypyridinylindolesulfonamides
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP18178773.0A EP3584244A1 (en) | 2018-06-20 | 2018-06-20 | Substituted alkoxypyridinyl indolsulfonamides |
| PCT/EP2019/066148 WO2019243398A1 (en) | 2018-06-20 | 2019-06-19 | Substituted alkoxypyridinyl indolsulfonamides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3810587T3 true DK3810587T3 (da) | 2022-10-31 |
Family
ID=62715911
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK19731283.8T DK3810587T3 (da) | 2018-06-20 | 2019-06-19 | Substituerede alkoxypyridinylindolsulfonamider |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US11976056B2 (da) |
| EP (3) | EP3584244A1 (da) |
| JP (1) | JP7371031B2 (da) |
| CN (1) | CN112292375B (da) |
| CA (1) | CA3101086A1 (da) |
| DK (1) | DK3810587T3 (da) |
| ES (1) | ES2929829T3 (da) |
| HR (1) | HRP20221289T1 (da) |
| HU (1) | HUE060181T2 (da) |
| LT (1) | LT3810587T (da) |
| MX (1) | MX2020012823A (da) |
| PL (1) | PL3810587T3 (da) |
| PT (1) | PT3810587T (da) |
| WO (1) | WO2019243398A1 (da) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP7631235B2 (ja) * | 2019-06-17 | 2025-02-18 | ウーツェーベー ファルマ ゲーエムベーハー | 多発性硬化症のようなcns障害を治療するためのgpr17モジュレーターとしてのn‐(フェニル)‐インドール‐3‐スルホンアミド誘導体及び関連化合物 |
| JP2023531358A (ja) * | 2020-05-01 | 2023-07-24 | ザ チルドレンズ メディカル センター コーポレーション | ミエリン形成を促進する組成物および方法 |
| CN112375027B (zh) * | 2020-12-07 | 2023-03-31 | 中国药科大学 | 吲哚磺酰胺类衍生物及其医药用途 |
| MX2023009045A (es) * | 2021-02-26 | 2023-08-10 | Hoffmann La Roche | Derivados novedosos de pirimidin-2-il sulfonamida. |
| EP4311828A1 (en) * | 2022-07-26 | 2024-01-31 | Basf Se | A process for the photolytic chlorination of 3-halopyridine with molecular chlorine |
| WO2023241960A1 (en) * | 2022-06-15 | 2023-12-21 | Basf Se | A process for the photolytic chlorination of 3-halopyridine with molecular chlorine |
| EP4558496A1 (en) * | 2022-07-20 | 2025-05-28 | F. Hoffmann-La Roche AG | Novel pyrimidinyl and triazinyl sulfonamide derivatives |
| CN119585264A (zh) * | 2022-07-20 | 2025-03-07 | 豪夫迈·罗氏有限公司 | 新颖异噻唑-3-基和异噁唑-3-基磺酰胺化合物 |
| EP4558479A1 (en) * | 2022-07-20 | 2025-05-28 | F. Hoffmann-La Roche AG | Novel naphthyl and isoquinoline sulfonamide derivatives |
| JP2025525574A (ja) | 2022-07-20 | 2025-08-05 | エフ. ホフマン-ラ ロシュ アーゲー | 新規のイミダゾピリジンおよびピラゾロピリジンスルホンアミド誘導体 |
| CN119546576A (zh) | 2022-07-20 | 2025-02-28 | 豪夫迈·罗氏有限公司 | 新颖的异喹啉酮、吡咯并吡啶酮和噻吩并吡啶酮磺酰胺衍生物 |
| JP2025524062A (ja) * | 2022-07-28 | 2025-07-25 | エフ. ホフマン-ラ ロシュ アーゲー | 新規7-置換インドールスルホンアミド誘導体 |
| KR20250042748A (ko) * | 2022-07-28 | 2025-03-27 | 에프. 호프만-라 로슈 아게 | 신규 7-치환 인돌 설폰아미드 유도체 |
| PE20251077A1 (es) * | 2022-08-26 | 2025-04-10 | Hoffmann La Roche | Derivados novedosos deuterados de pirimidin-2-il sulfonamida |
| AU2023401169A1 (en) * | 2022-12-02 | 2025-05-29 | Rewind Therapeutics Nv | Fused pyrrolyl-sulfonamide compounds |
| WO2024153233A1 (en) * | 2023-01-19 | 2024-07-25 | Nanjing Immunophage Biotech Co., Ltd | Compounds and their uses as gpr17 antagonists |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19814084B4 (de) | 1998-03-30 | 2005-12-22 | Lts Lohmann Therapie-Systeme Ag | D2-Agonist enthaltendes transdermales therapeutisches System zur Behandlung des Parkinson-Syndroms und Verfahren zu seiner Herstellung |
| SE9904750D0 (sv) | 1999-12-23 | 1999-12-23 | Pharmacia & Upjohn Ab | New formulation, use and method |
| WO2005103291A1 (ja) | 2004-04-27 | 2005-11-03 | Takeda Pharmaceutical Company Limited | Gタンパク質共役型レセプタータンパク質の新規リガンドとその用途 |
| ITMI20042007A1 (it) | 2004-10-21 | 2005-01-21 | Consiglio Nazionale Ricerche | "modulatori del ricettore gpr17 e loro impieghi terapeutici" |
| MX2008007897A (es) | 2005-12-20 | 2009-03-04 | Teikoku Pharma Usa Inc | Metodos para administrar transdermicamente un agonista de receptor de indol serotonina y composiciones transdermicas para uso con los mismos. |
| EP2162183B1 (de) | 2007-06-25 | 2019-06-26 | AMW GmbH | Elektrophoretisches transdermales applikationssystem |
| US20120172375A1 (en) * | 2008-11-07 | 2012-07-05 | Bruce Trapp | Compounds and methods of promoting oligodendrocyte precursor differentiation |
| WO2011113032A2 (en) | 2010-03-11 | 2011-09-15 | Swinford Jerry L | Method and apparatus for washing dowhole tubulars and equipment |
| EP2567698B1 (en) * | 2011-09-07 | 2014-02-12 | Rheinische Friedrich-Wilhelms-Universität Bonn | GPR 17 agonists and screening assay |
| JP6082457B2 (ja) | 2012-05-09 | 2017-02-15 | ウニヴェルスィタ デッリ ストゥディ ディ ミラノ | Gpr17受容体調節因子 |
| WO2018057989A1 (en) * | 2016-09-24 | 2018-03-29 | Washington University | INHIBITORS OF SARM1 NADase ACTIVITY AND USES THEREOF |
| TWI754702B (zh) * | 2016-12-28 | 2022-02-11 | 德商Ucb製藥有限公司 | (氮雜)吲哚-和苯並呋喃-3-磺醯胺類 |
-
2018
- 2018-06-20 EP EP18178773.0A patent/EP3584244A1/en not_active Ceased
-
2019
- 2019-06-19 PT PT197312838T patent/PT3810587T/pt unknown
- 2019-06-19 CN CN201980039867.9A patent/CN112292375B/zh active Active
- 2019-06-19 JP JP2020570978A patent/JP7371031B2/ja active Active
- 2019-06-19 ES ES19731283T patent/ES2929829T3/es active Active
- 2019-06-19 MX MX2020012823A patent/MX2020012823A/es unknown
- 2019-06-19 HU HUE19731283A patent/HUE060181T2/hu unknown
- 2019-06-19 LT LTEPPCT/EP2019/066148T patent/LT3810587T/lt unknown
- 2019-06-19 CA CA3101086A patent/CA3101086A1/en active Pending
- 2019-06-19 WO PCT/EP2019/066148 patent/WO2019243398A1/en not_active Ceased
- 2019-06-19 DK DK19731283.8T patent/DK3810587T3/da active
- 2019-06-19 EP EP22174561.5A patent/EP4086248A1/en not_active Withdrawn
- 2019-06-19 HR HRP20221289TT patent/HRP20221289T1/hr unknown
- 2019-06-19 EP EP19731283.8A patent/EP3810587B1/en active Active
- 2019-06-19 PL PL19731283.8T patent/PL3810587T3/pl unknown
- 2019-06-19 US US17/058,567 patent/US11976056B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP3810587B1 (en) | 2022-08-10 |
| PT3810587T (pt) | 2022-11-14 |
| CN112292375B (zh) | 2023-12-05 |
| EP3584244A1 (en) | 2019-12-25 |
| LT3810587T (lt) | 2022-11-25 |
| WO2019243398A1 (en) | 2019-12-26 |
| HRP20221289T1 (hr) | 2022-12-23 |
| JP2021527696A (ja) | 2021-10-14 |
| JP7371031B2 (ja) | 2023-10-30 |
| PL3810587T3 (pl) | 2023-02-06 |
| HUE060181T2 (hu) | 2023-02-28 |
| EP3810587A1 (en) | 2021-04-28 |
| CN112292375A (zh) | 2021-01-29 |
| MX2020012823A (es) | 2021-02-15 |
| US11976056B2 (en) | 2024-05-07 |
| CA3101086A1 (en) | 2019-12-26 |
| US20210214337A1 (en) | 2021-07-15 |
| EP4086248A1 (en) | 2022-11-09 |
| ES2929829T3 (es) | 2022-12-01 |
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