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DK1732534T3 - Anvendelse af methylenamidderivater ved cardiovaskulære sygdomme - Google Patents

Anvendelse af methylenamidderivater ved cardiovaskulære sygdomme

Info

Publication number
DK1732534T3
DK1732534T3 DK05716814T DK05716814T DK1732534T3 DK 1732534 T3 DK1732534 T3 DK 1732534T3 DK 05716814 T DK05716814 T DK 05716814T DK 05716814 T DK05716814 T DK 05716814T DK 1732534 T3 DK1732534 T3 DK 1732534T3
Authority
DK
Denmark
Prior art keywords
derivatives
methylenamide
cardiovascular diseases
prevention
formula
Prior art date
Application number
DK05716814T
Other languages
English (en)
Inventor
Van Huijsduijnen Rob Hooft
Vincent Richard
Original Assignee
Serono Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Serono Lab filed Critical Serono Lab
Application granted granted Critical
Publication of DK1732534T3 publication Critical patent/DK1732534T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK05716814T 2004-02-27 2005-02-25 Anvendelse af methylenamidderivater ved cardiovaskulære sygdomme DK1732534T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04100778 2004-02-27
PCT/EP2005/050823 WO2005082347A1 (en) 2004-02-27 2005-02-25 Use of methylene amide derivatives in cardiovascular disorders

Publications (1)

Publication Number Publication Date
DK1732534T3 true DK1732534T3 (da) 2008-11-17

Family

ID=34896106

Family Applications (1)

Application Number Title Priority Date Filing Date
DK05716814T DK1732534T3 (da) 2004-02-27 2005-02-25 Anvendelse af methylenamidderivater ved cardiovaskulære sygdomme

Country Status (23)

Country Link
US (1) US20070185118A1 (da)
EP (1) EP1732534B1 (da)
JP (1) JP5001138B2 (da)
KR (1) KR101188940B1 (da)
CN (1) CN1933827B (da)
AT (1) ATE401877T1 (da)
AU (1) AU2005216649B2 (da)
BR (1) BRPI0508080A (da)
CA (1) CA2554919C (da)
CY (1) CY1108252T1 (da)
DE (1) DE602005008412D1 (da)
DK (1) DK1732534T3 (da)
EA (1) EA011811B1 (da)
ES (1) ES2308458T3 (da)
HR (1) HRP20080367T3 (da)
IL (1) IL177494A (da)
NO (1) NO20064295L (da)
PL (1) PL1732534T3 (da)
PT (1) PT1732534E (da)
RS (1) RS50596B (da)
SI (1) SI1732534T1 (da)
UA (1) UA84453C2 (da)
WO (1) WO2005082347A1 (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA012260B1 (ru) * 2002-01-29 2009-08-28 Лаборатуар Сероно Са ЗАМЕЩЁННЫЕ ПРОИЗВОДНЫЕ МЕТИЛЕНАМИДА В КАЧЕСТВЕ МОДУЛЯТОРОВ ПРОТЕИНТИРОЗИНФОСФАТАЗ (PTPs)
EP1654247B1 (en) 2003-07-21 2010-01-20 Merck Serono SA Alkynyl aryl carboxamides
US7884234B2 (en) * 2006-10-12 2011-02-08 Institute Of Medicinal Molecular Design, Inc. N-phenyloxamide derivatives
US8633245B2 (en) * 2008-04-11 2014-01-21 Institute Of Medicinal Molecular Design, Inc. PAI-1 inhibitor
TW201319023A (zh) 2011-08-29 2013-05-16 Ticona Llc 具改良低剪切黏度之熱向性液晶聚合物
TW201319223A (zh) 2011-08-29 2013-05-16 Ticona Llc 高流量液晶聚合物組合物
US9045685B2 (en) 2011-08-29 2015-06-02 Ticona Llc Cast molded parts formed from a liquid crystalline polymer
TW201313884A (zh) 2011-08-29 2013-04-01 Ticona Llc 液晶聚合物之固態聚合
CN103764793B (zh) 2011-08-29 2016-09-14 提克纳有限责任公司 高流动液晶聚合物组合物
JP2014529627A (ja) 2011-08-29 2014-11-13 ティコナ・エルエルシー 芳香族アミド化合物
US9057016B2 (en) 2011-08-29 2015-06-16 Ticona Llc Melt polymerization of low melt viscosity liquid crystalline polymers
WO2013032971A1 (en) 2011-08-29 2013-03-07 Ticona Llc Melt-extruded substrate for use in thermoformed articles
JP2014525499A (ja) 2011-08-29 2014-09-29 ティコナ・エルエルシー 低い融解温度をもつ耐熱性液晶ポリマー組成物
WO2014095815A1 (en) 2012-12-17 2014-06-26 Shell Internationale Research Maatschappij B.V. Integrated gas-to-liquid condensate process
WO2014130275A2 (en) 2013-02-22 2014-08-28 Ticona Llc High performance polymer composition with improved flow properties
CN113912988A (zh) 2013-06-07 2022-01-11 提克纳有限责任公司 高强度热致液晶聚合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6985200A (en) * 1999-09-10 2001-04-17 Novo Nordisk A/S Modulators of protein tyrosine phosphatases (ptpases)
US6627767B2 (en) * 2000-08-29 2003-09-30 Abbott Laboratories Amino(oxo) acetic acid protein tyrosine phosphatase inhibitors
DE10117823A1 (de) * 2001-04-10 2002-10-17 Merck Patent Gmbh Oxalsäurederivate
AR034374A1 (es) * 2001-06-07 2004-02-18 Wyeth Corp Combinacion de un inhibidor de ptpasa y un inhibidor de ace
WO2002098408A1 (en) * 2001-06-07 2002-12-12 Wyeth Ptpase inhibitors for improving cardiovascular risk profile
EA012260B1 (ru) * 2002-01-29 2009-08-28 Лаборатуар Сероно Са ЗАМЕЩЁННЫЕ ПРОИЗВОДНЫЕ МЕТИЛЕНАМИДА В КАЧЕСТВЕ МОДУЛЯТОРОВ ПРОТЕИНТИРОЗИНФОСФАТАЗ (PTPs)

Also Published As

Publication number Publication date
US20070185118A1 (en) 2007-08-09
UA84453C2 (ru) 2008-10-27
JP2007524701A (ja) 2007-08-30
IL177494A (en) 2011-06-30
KR101188940B1 (ko) 2012-10-08
HRP20080367T3 (en) 2008-09-30
ATE401877T1 (de) 2008-08-15
JP5001138B2 (ja) 2012-08-15
ES2308458T3 (es) 2008-12-01
CA2554919A1 (en) 2005-09-09
CN1933827B (zh) 2011-07-27
AU2005216649B2 (en) 2010-09-09
IL177494A0 (en) 2006-12-31
CA2554919C (en) 2013-04-16
PL1732534T3 (pl) 2008-12-31
RS50596B (sr) 2010-05-07
EA011811B1 (ru) 2009-06-30
EP1732534B1 (en) 2008-07-23
BRPI0508080A (pt) 2007-07-17
PT1732534E (pt) 2008-08-08
AU2005216649A1 (en) 2005-09-09
HK1098073A1 (en) 2007-07-13
WO2005082347A1 (en) 2005-09-09
CY1108252T1 (el) 2014-02-12
KR20060129066A (ko) 2006-12-14
CN1933827A (zh) 2007-03-21
EP1732534A1 (en) 2006-12-20
EA200601511A1 (ru) 2007-02-27
SI1732534T1 (sl) 2008-10-31
NO20064295L (no) 2006-09-22
DE602005008412D1 (de) 2008-09-04

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