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DK1687288T3 - Substituerede arylcycloalkanoderivater og fremgangsmåder til anvendelse deraf - Google Patents

Substituerede arylcycloalkanoderivater og fremgangsmåder til anvendelse deraf

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Publication number
DK1687288T3
DK1687288T3 DK04795187T DK04795187T DK1687288T3 DK 1687288 T3 DK1687288 T3 DK 1687288T3 DK 04795187 T DK04795187 T DK 04795187T DK 04795187 T DK04795187 T DK 04795187T DK 1687288 T3 DK1687288 T3 DK 1687288T3
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Prior art keywords
derivatives
methods
combinations
fibromyalgia
substituted
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DK04795187T
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Danish (da)
English (en)
Inventor
Eugene John Trybulski
Joseph Peter Sabatucci
An Thien Vu
Arthur Attilio Santilli
Fei Ye
Paige Erin Mahaney
Stephen Todd Cohn
Lori Danielle Krim
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Wyeth Corp
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Publication of DK1687288T3 publication Critical patent/DK1687288T3/da

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    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/092—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings with aromatic radicals attached to the chain
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DK04795187T 2003-10-14 2004-10-13 Substituerede arylcycloalkanoderivater og fremgangsmåder til anvendelse deraf DK1687288T3 (da)

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US51094303P 2003-10-14 2003-10-14
US56130104P 2004-04-12 2004-04-12
US56999604P 2004-05-11 2004-05-11
US10/963,111 US7365076B2 (en) 2003-10-14 2004-10-12 Substituted aryl cycloalkanol derivatives and methods of their use
PCT/US2004/033990 WO2005037809A1 (fr) 2003-10-14 2004-10-13 Derives de cycloalcanoyl aryle substitues et procedes d'utilisation de ceux-ci

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US (2) US7365076B2 (fr)
EP (1) EP1687288B1 (fr)
JP (1) JP2007509076A (fr)
KR (1) KR20070026323A (fr)
AT (1) ATE384055T1 (fr)
AU (1) AU2004282193A1 (fr)
BR (1) BRPI0415380A (fr)
CA (1) CA2540207A1 (fr)
CR (1) CR8313A (fr)
DE (1) DE602004011385T2 (fr)
DK (1) DK1687288T3 (fr)
EC (1) ECSP066505A (fr)
ES (1) ES2300841T3 (fr)
IL (1) IL174539A0 (fr)
MX (1) MXPA06003882A (fr)
NO (1) NO20061383L (fr)
PE (1) PE20050478A1 (fr)
PL (1) PL1687288T3 (fr)
TW (1) TW200526602A (fr)
WO (1) WO2005037809A1 (fr)

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US7517899B2 (en) * 2004-03-30 2009-04-14 Wyeth Phenylaminopropanol derivatives and methods of their use
US7414052B2 (en) * 2004-03-30 2008-08-19 Wyeth Phenylaminopropanol derivatives and methods of their use
GB0513702D0 (en) 2005-07-04 2005-08-10 Sterix Ltd Compound
CA2629807A1 (fr) * 2005-12-05 2007-06-14 Wyeth Procede pour preparer des derives d'arylcycloalcanol substitues
EP1957470A1 (fr) * 2005-12-05 2008-08-20 Wyeth Procede pour la synthese selective d'enantiomeres de 1-(2-amino-1-phenyl-ethyl)-cyclohexanols substitues
CA2648030C (fr) * 2006-03-27 2018-02-13 Children's Hospital & Regional Medical Center Compositions et procedes comprenant l'utilisation d'endonucleases ciblees affichees en surface cellulaire

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EP1687288A1 (fr) 2006-08-09
BRPI0415380A (pt) 2006-12-12
US20050143579A1 (en) 2005-06-30
US20080153826A1 (en) 2008-06-26
ATE384055T1 (de) 2008-02-15
NO20061383L (no) 2006-06-02
AU2004282193A1 (en) 2005-04-28
US7550456B2 (en) 2009-06-23
ECSP066505A (es) 2006-10-10
WO2005037809A1 (fr) 2005-04-28
CR8313A (es) 2006-10-04
TW200526602A (en) 2005-08-16
KR20070026323A (ko) 2007-03-08
IL174539A0 (en) 2006-08-01
JP2007509076A (ja) 2007-04-12
MXPA06003882A (es) 2006-07-03
US7365076B2 (en) 2008-04-29
PE20050478A1 (es) 2005-09-20
DE602004011385T2 (de) 2009-05-14
CA2540207A1 (fr) 2005-04-28
PL1687288T3 (pl) 2008-06-30
ES2300841T3 (es) 2008-06-16
EP1687288B1 (fr) 2008-01-16
DE602004011385D1 (de) 2008-03-06

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