DK1355906T3 - 2H-1-benzopyranderivater, fremgangsmåder til deres fremstilling og farmaceutiske sammensætninger indeholdende dem - Google Patents

2H-1-benzopyranderivater, fremgangsmåder til deres fremstilling og farmaceutiske sammensætninger indeholdende dem

Info

Publication number: DK1355906T3
Authority: DK; Denmark
Prior art keywords: preparation; processes; pharmaceutical compositions; compositions containing; benzopyran derivatives
Prior art date: 2001-01-24

Application number

DK02703564T

Other languages

English (en)

Inventor

Gabriele Amari

Maurizio Civelli

Maurizio Delcanale

Elisabetta Armani

Elisabetta Galbiati

Original Assignee

Chiesi Farma Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-01-24

Filing date

2002-01-21

Publication date

2005-05-30

2001-01-24 Priority claimed from EP01101521A external-priority patent/EP1229036B1/en

2001-08-03 Priority claimed from EP01118682A external-priority patent/EP1281710A1/en

2002-01-21 Application filed by Chiesi Farma Spa filed Critical Chiesi Farma Spa

2005-05-30 Application granted granted Critical

2005-05-30 Publication of DK1355906T3 publication Critical patent/DK1355906T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Physical Education & Sports Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrane Compounds (AREA)

DK02703564T 2001-01-24 2002-01-21 2H-1-benzopyranderivater, fremgangsmåder til deres fremstilling og farmaceutiske sammensætninger indeholdende dem DK1355906T3 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
EP01101521A EP1229036B1 (en)	2001-01-24	2001-01-24	2H-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
EP01118682A EP1281710A1 (en)	2001-08-03	2001-08-03	2H-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
EP02703564A EP1355906B1 (en)	2001-01-24	2002-01-21	2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
PCT/EP2002/000567 WO2002059113A1 (en)	2001-01-24	2002-01-21	2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof

Publications (1)

Publication Number	Publication Date
DK1355906T3 true DK1355906T3 (da)	2005-05-30

Family

ID=26076450

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK02703564T DK1355906T3 (da)	2001-01-24	2002-01-21	2H-1-benzopyranderivater, fremgangsmåder til deres fremstilling og farmaceutiske sammensætninger indeholdende dem

Country Status (26)

Country	Link
US (1)	US6951883B2 (da)
EP (1)	EP1355906B1 (da)
JP (1)	JP4332349B2 (da)
CN (1)	CN1261431C (da)
AT (1)	ATE286894T1 (da)
AU (1)	AU2002237282B2 (da)
BR (1)	BR0207066A (da)
CA (1)	CA2435775A1 (da)
CZ (1)	CZ20032014A3 (da)
DE (1)	DE60202590T2 (da)
DK (1)	DK1355906T3 (da)
DZ (1)	DZ3459A1 (da)
EA (1)	EA006158B1 (da)
ES (1)	ES2236485T3 (da)
HU (1)	HUP0401018A3 (da)
IL (2)	IL157065A0 (da)
MA (1)	MA26982A1 (da)
MX (1)	MXPA03006505A (da)
NO (1)	NO327808B1 (da)
NZ (1)	NZ527144A (da)
PL (1)	PL365062A1 (da)
PT (1)	PT1355906E (da)
SI (1)	SI1355906T1 (da)
SK (1)	SK287086B6 (da)
TN (1)	TNSN03043A1 (da)
WO (1)	WO2002059113A1 (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP4976649B2 (ja) *	2004-09-21	2012-07-18	マーシャルエドワーズ，インク．	化合物
ATE532777T1 (de) *	2004-09-21	2011-11-15	Marshall Edwards Inc	Substituierte chromanderivate, medikamente und anwendungen in der therapie
US8080675B2 (en)	2004-09-21	2011-12-20	Marshall Edwards, Inc.	Chroman derivatives, medicaments and use in therapy
EP2436680B1 (en) *	2004-09-21	2016-05-18	Marshall Edwards, Inc.	Chroman derivatives, medicaments and use in therapy
AU2005201855B2 (en) *	2004-09-21	2012-03-29	Marshall Edwards, Inc.	Chroman derived compounds and formulations thereof for use in therapy
ES2377073T3 (es) *	2004-09-21	2012-03-22	Marshall Edwards, Inc.	Derivados de cromano sustituidos, medicamentos y utilización en terapia
CN101444499B (zh) *	2007-11-26	2012-12-05	湘北威尔曼制药股份有限公司	一种化合物及其组合物的新用途
US9663484B2 (en)	2010-11-01	2017-05-30	Mei Pharma, Inc.	Isoflavonoid compounds and methods for the treatment of cancer
JP6576916B2 (ja)	2013-06-19	2019-09-18	セラゴンファーマシューティカルズ，インク．	エストロゲン受容体モジュレーター及びその使用
EP3253208B1 (en)	2015-02-02	2021-05-05	MEI Pharma, Inc.	Combination therapies for use in the treatment of breast cancer
EP3541809B1 (en) *	2016-11-17	2025-06-25	Sanofi	Novel substituted n-(3-fluoropropyl)-pyrrolidine compounds, processes for their preparation and therapeutic uses thereof
US20200215025A1 (en) *	2017-09-15	2020-07-09	Norbio No. 1 Pty Ltd	Treatment of excitotoxicity
CN112225716A (zh) *	2020-10-30	2021-01-15	陕西嘉禾生物科技股份有限公司	一种鹰嘴豆牙素a的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3374245A (en) *	1964-04-01	1968-03-19	Ciba Geigy Corp	Unsaturated oxacycles
DE1518002C3 (de) *	1965-01-02	1975-01-23	Merck Patent Gmbh, 6100 Darmstadt	Isoflavane und Isoflavene und Verfahren zu Ihrer Herstellung sowie diese enthaltende Arzneimittel
US5280040A (en) *	1993-03-11	1994-01-18	Zymogenetics, Inc.	Methods for reducing bone loss using centchroman derivatives
WO1998018774A1 (en)	1996-10-28	1998-05-07	Novo Nordisk A/S	Novel trans-3,4-chroman derivatives useful in the prevention or treatment of estrogen related diseases or syndromes
US5985306A (en) *	1996-10-28	1999-11-16	Novo Nordisk A/S	(+)-enantiomers of cis-3,4-chroman derivatives useful in prevention or treatment of estrogen diseases or syndromes
US6153768A (en) *	1996-12-13	2000-11-28	C & C Research Laboratories	Benzopyran derivatives
KR20000001793A (ko)	1998-06-13	2000-01-15	이경하	신규한 벤조피란 또는 티오벤조피란 유도체
AU765159B2 (en) *	1998-12-30	2003-09-11	Signal Pharmaceuticals, Inc.	Compounds and methods for modulation of estrogen receptors

2002
- 2002-01-21 WO PCT/EP2002/000567 patent/WO2002059113A1/en not_active Ceased
- 2002-01-21 MX MXPA03006505A patent/MXPA03006505A/es active IP Right Grant
- 2002-01-21 IL IL15706502A patent/IL157065A0/xx unknown
- 2002-01-21 CA CA002435775A patent/CA2435775A1/en not_active Abandoned
- 2002-01-21 CZ CZ20032014A patent/CZ20032014A3/cs unknown
- 2002-01-21 US US10/466,118 patent/US6951883B2/en not_active Expired - Fee Related
- 2002-01-21 PL PL02365062A patent/PL365062A1/xx not_active IP Right Cessation
- 2002-01-21 PT PT02703564T patent/PT1355906E/pt unknown
- 2002-01-21 DE DE60202590T patent/DE60202590T2/de not_active Expired - Lifetime
- 2002-01-21 ES ES02703564T patent/ES2236485T3/es not_active Expired - Lifetime
- 2002-01-21 HU HU0401018A patent/HUP0401018A3/hu unknown
- 2002-01-21 SI SI200230096T patent/SI1355906T1/xx unknown
- 2002-01-21 EA EA200300727A patent/EA006158B1/ru not_active IP Right Cessation
- 2002-01-21 EP EP02703564A patent/EP1355906B1/en not_active Expired - Lifetime
- 2002-01-21 SK SK939-2003A patent/SK287086B6/sk not_active IP Right Cessation
- 2002-01-21 DK DK02703564T patent/DK1355906T3/da active
- 2002-01-21 DZ DZ023459A patent/DZ3459A1/fr active
- 2002-01-21 CN CNB02804066XA patent/CN1261431C/zh not_active Expired - Fee Related
- 2002-01-21 AT AT02703564T patent/ATE286894T1/de not_active IP Right Cessation
- 2002-01-21 AU AU2002237282A patent/AU2002237282B2/en not_active Ceased
- 2002-01-21 NZ NZ527144A patent/NZ527144A/en unknown
- 2002-01-21 BR BR0207066-9A patent/BR0207066A/pt not_active IP Right Cessation
- 2002-01-21 JP JP2002559415A patent/JP4332349B2/ja not_active Expired - Fee Related
2003
- 2003-07-08 TN TNPCT/EP2002/000567A patent/TNSN03043A1/en unknown
- 2003-07-15 MA MA27236A patent/MA26982A1/fr unknown
- 2003-07-23 NO NO20033318A patent/NO327808B1/no not_active IP Right Cessation
- 2003-07-23 IL IL157065A patent/IL157065A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
PL365062A1 (en)	2004-12-27
NO20033318D0 (no)	2003-07-23
JP4332349B2 (ja)	2009-09-16
SK287086B6 (sk)	2009-11-05
DZ3459A1 (fr)	2002-08-01
US20040106595A1 (en)	2004-06-03
MXPA03006505A (es)	2004-04-21
EA006158B1 (ru)	2005-10-27
PT1355906E (pt)	2005-05-31
CN1487934A (zh)	2004-04-07
CN1261431C (zh)	2006-06-28
ATE286894T1 (de)	2005-01-15
NO327808B1 (no)	2009-09-28
HK1060558A1 (en)	2004-08-13
JP2004517151A (ja)	2004-06-10
MA26982A1 (fr)	2004-12-20
HUP0401018A3 (en)	2007-05-29
NZ527144A (en)	2005-03-24
AU2002237282B2 (en)	2007-02-15
WO2002059113A1 (en)	2002-08-01
IL157065A0 (en)	2004-02-08
IL157065A (en)	2010-05-17
US6951883B2 (en)	2005-10-04
EP1355906A1 (en)	2003-10-29
SI1355906T1 (en)	2005-06-30
CA2435775A1 (en)	2002-08-01
BR0207066A (pt)	2004-03-30
HUP0401018A2 (hu)	2004-09-28
DE60202590T2 (de)	2005-12-29
EP1355906B1 (en)	2005-01-12
TNSN03043A1 (en)	2005-12-23
SK9392003A3 (en)	2003-12-02
EA200300727A1 (ru)	2004-02-26
ES2236485T3 (es)	2005-07-16
CZ20032014A3 (cs)	2003-12-17
DE60202590D1 (de)	2005-02-17
NO20033318L (no)	2003-09-24

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IS6677A (is)	2003-01-13	Amínóalkýlbensóýl-bensófúran eða bensóþíófenafleiður, aðferð til framleiðslu þeirra og samsetningarsem innihalda þær
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IS6675A (is)	2003-01-13	Amínóalkoxýbensóýl-bensófúran eða bensóþíófenafleiður, aðferð til framleiðslu þeirra og samsetningar sem innihalda þær
WO2001087287A3 (en)	2002-05-16	Use of pyrazole derivatives for treating infertility
AU2002357740A1 (en)	2003-06-23	Pyrazolo-pyridine derivatives as antiherpes agents
NO20012428L (no)	2001-07-17	Substituerte kaprolaktamer, farmasöytiske sammensetninger som inneholder dem og deres anvendelse ved behandling av tumorer
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AP2001002369A0 (en)	2001-12-31	Pharmaceutical complex.
PL368040A1 (en)	2005-03-21	Substituted 4-aminocyclohexanol derivatives
NO20035215D0 (no)	2003-11-24	Tricykliske dihydrokinolinforbindelser, fremgangsmåte for deres fremstilling og farmasöytiske sammensetninger inneholdende dem
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DE60108354D1 (de)	2005-02-17	2H-1-Benzopyran-Derivative, Prozesse zu ihrer Herstellung und Pharmazeutische Zusammensetzungen
TW200503672A (en)	2005-02-01	2-aminobenzoyl derivatives
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NO20035214D0 (no)	2003-11-24	Tricykliske dihydrokinolinforbindelser, fremgangsmåte for deres fremstilling og farmasöytiske sammensetninger inneholdende dem